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Items: 7

1.

Allosteric modulation of caspases.

Häcker HG, Sisay MT, Gütschow M.

Pharmacol Ther. 2011 Nov;132(2):180-95. doi: 10.1016/j.pharmthera.2011.07.003. Epub 2011 Jul 23. Review.

PMID:
21807025
2.

Solid-phase synthesis of disubstituted N-acylureas from resin-bound ureas and acyl chlorides.

Häcker HG, Meusel M, Aschfalk M, Gütschow M.

ACS Comb Sci. 2011 Jan 10;13(1):59-64. doi: 10.1021/co100020b. Epub 2010 Nov 10.

PMID:
21247126
3.

Direct formation of ring-fused 1,3-thiazine-2,4-dithiones from aromatic o-amino carboxylic acids: observation of a carbon disulfide mediated thionation.

Ottersbach PA, Elsinghorst PW, Häcker HG, Gütschow M.

Org Lett. 2010 Aug 20;12(16):3662-5. doi: 10.1021/ol101471g.

PMID:
20666472
4.

Analogs of a 4-aminothieno[2,3-d]pyrimidine lead (QB13) as modulators of P-glycoprotein substrate specificity.

Häcker HG, de la Haye A, Sterz K, Schnakenburg G, Wiese M, Gütschow M.

Bioorg Med Chem Lett. 2009 Nov 1;19(21):6102-5. doi: 10.1016/j.bmcl.2009.09.023. Epub 2009 Sep 11.

PMID:
19783433
5.

Aromatic 2-(thio)ureidocarboxylic acids as a new family of modulators of multidrug resistance-associated protein 1: synthesis, biological evaluation, and structure-activity relationships.

Häcker HG, Leyers S, Wiendlocha J, Gütschow M, Wiese M.

J Med Chem. 2009 Aug 13;52(15):4586-95. doi: 10.1021/jm900688v.

PMID:
19580319
6.

2-Amino- and 2-alkylthio-4H-3,1-benzothiazin-4-ones: synthesis, interconversion and enzyme inhibitory activities.

Häcker HG, Grundmann F, Lohr F, Ottersbach PA, Zhou J, Schnakenburg G, Gütschow M.

Molecules. 2009 Jan 14;14(1):378-402. doi: 10.3390/molecules14010378.

7.

A 4-aminobenzoic acid derivative as novel lead for selective inhibitors of multidrug resistance-associated proteins.

Leyers S, Häcker HG, Wiendlocha J, Gütschow M, Wiese M.

Bioorg Med Chem Lett. 2008 Sep 1;18(17):4761-3. doi: 10.1016/j.bmcl.2008.07.127. Epub 2008 Aug 3.

PMID:
18707884

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