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Items: 1 to 20 of 51

1.

Targeting an EGFR water network using novel 4-anilinoquin(az)olines inhibitors for chordoma.

Asquith CRM, Maffuid KA, Laitinen T, Torrice C, Tizzard GJ, Crona DJ, Zuercher WJ.

ChemMedChem. 2019 Aug 19. doi: 10.1002/cmdc.201900428. [Epub ahead of print]

PMID:
31424613
2.

Novel epidithiodiketopiperazines as anti-viral zinc ejectors of the Feline Immunodeficiency Virus (FIV) nucleocapsid protein as a model for HIV infection.

Asquith CRM, Sil BC, Laitinen T, Tizzard GJ, Coles SJ, Poso A, Hofmann-Lehmann R, Hilton ST.

Bioorg Med Chem. 2019 Sep 15;27(18):4174-4184. doi: 10.1016/j.bmc.2019.07.047. Epub 2019 Jul 30.

PMID:
31395510
3.

Solvent-Free Synthesis and Key Intermediate Isolation in Ni2Dy2 Catalyst Development in the Domino Ring-Opening Electrocyclization Reaction of Furfural and Amines.

Sampani SI, McGown A, Vargas A, Abdul-Sada A, Tizzard GJ, Coles SJ, Spencer J, Kostakis GE.

J Org Chem. 2019 Jun 7;84(11):6858-6867. doi: 10.1021/acs.joc.9b00608. Epub 2019 May 22.

PMID:
31074278
4.

A synthetic approach to chrysophaentin F.

Vendeville JB, Matters RF, Chen A, Light ME, Tizzard GJ, Chai CLL, Harrowven DC.

Chem Commun (Camb). 2019 Apr 18;55(33):4837-4840. doi: 10.1039/c9cc01666j.

PMID:
30950475
5.

Twists to the Spin Structure of the Ln9-diabolo Motif Exemplified in Two {Zn2Ln2}[Ln9]{Zn2} Coordination Clusters.

Griffiths K, Kühne IA, Tizzard GJ, Coles SJ, Kostakis GE, Powell AK.

Inorg Chem. 2019 Feb 18;58(4):2483-2490. doi: 10.1021/acs.inorgchem.8b03048. Epub 2019 Jan 31.

PMID:
30702868
6.

Stopping Hydrogen Migration in Its Tracks: The First Successful Synthesis of Group Ten Scorpionate Complexes Based on Azaindole Scaffolds.

da Costa RC, Rawe BW, Iannetelli A, Tizzard GJ, Coles SJ, Guwy AJ, Owen GR.

Inorg Chem. 2019 Jan 7;58(1):359-367. doi: 10.1021/acs.inorgchem.8b02456. Epub 2018 Dec 10.

PMID:
30525534
7.

Modulation of σ-Alkane Interactions in [Rh(L2)(alkane)]+ Solid-State Molecular Organometallic (SMOM) Systems by Variation of the Chelating Phosphine and Alkane: Access to η22-σ-Alkane Rh(I), η1-σ-Alkane Rh(III) Complexes, and Alkane Encapsulation.

Martínez-Martínez AJ, Tegner BE, McKay AI, Bukvic AJ, Rees NH, Tizzard GJ, Coles SJ, Warren MR, Macgregor SA, Weller AS.

J Am Chem Soc. 2018 Nov 7;140(44):14958-14970. doi: 10.1021/jacs.8b09364. Epub 2018 Oct 24.

PMID:
30351014
8.

Probing the Anticancer Action of Novel Ferrocene Analogues of MNK Inhibitors.

Sansook S, Lineham E, Hassell-Hart S, Tizzard GJ, Coles SJ, Spencer J, Morley SJ.

Molecules. 2018 Aug 23;23(9). pii: E2126. doi: 10.3390/molecules23092126.

9.

Synthesis and Reactivity of N-Allenyl Cyanamides.

Ayres JN, Williams MTJ, Tizzard GJ, Coles SJ, Ling KB, Morrill LC.

Org Lett. 2018 Sep 7;20(17):5282-5285. doi: 10.1021/acs.orglett.8b02225. Epub 2018 Aug 14.

10.

Combining Sanford Arylations on Benzodiazepines with the Nuisance Effect.

Khan R, Boonseng S, Kemmitt PD, Felix R, Coles SJ, Tizzard GJ, Williams G, Simmonds O, Harvey JL, Atack J, Cox H, Spencer J.

Adv Synth Catal. 2017 Sep 18;359(18):3261-3269. doi: 10.1002/adsc.201700626. Epub 2017 Aug 2.

11.

Preparation and reactivity of rhodium and iridium complexes containing a methylborohydride based unit supported by two 7-azaindolyl heterocycles.

Da Costa RC, Rawe BW, Tsoureas N, Haddow MF, Sparkes HA, Tizzard GJ, Coles SJ, Owen GR.

Dalton Trans. 2018 Aug 14;47(32):11047-11057. doi: 10.1039/c8dt02311e.

PMID:
30027202
12.

Copper(ii)-benzotriazole coordination compounds in click chemistry: a diagnostic reactivity study.

Loukopoulos E, Abdul-Sada A, Csire G, Kállay C, Brookfield A, Tizzard GJ, Coles SJ, Lykakis IN, Kostakis GE.

Dalton Trans. 2018 Aug 21;47(31):10491-10508. doi: 10.1039/c8dt01256c. Epub 2018 May 24.

PMID:
29796447
13.

Synergistic effects of inhibiting the MNK-eIF4E and PI3K/AKT/ mTOR pathways on cell migration in MDA-MB-231 cells.

Lineham E, Tizzard GJ, Coles SJ, Spencer J, Morley SJ.

Oncotarget. 2018 Jan 31;9(18):14148-14159. doi: 10.18632/oncotarget.24354. eCollection 2018 Mar 6.

14.

Dinucleating Schiff base ligand in Zn/4f coordination chemistry: synthetic challenges and catalytic activity evaluation.

Sampani SI, Aubert S, Cattoen M, Griffiths K, Abdul-Sada A, Akien GR, Tizzard GJ, Coles SJ, Arseniyadis S, Kostakis GE.

Dalton Trans. 2018 Mar 26;47(13):4486-4493. doi: 10.1039/c8dt00538a.

PMID:
29505050
15.

Synthesis and biological evaluation of ferrocene-based cannabinoid receptor 2 ligands.

Sansook S, Tuo W, Bollier M, Barczyk A, Dezitter X, Klupsch F, Leleu-Chavain N, Farce A, Tizzard GJ, Coles SJ, Spencer J, Millet R.

Future Med Chem. 2018 Mar 1;10(6):631-638. doi: 10.4155/fmc-2017-0200. Epub 2018 Feb 8.

PMID:
29419319
16.

Correction: Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety.

Sansook S, Ocasio CA, Day IJ, Tizzard GJ, Coles SJ, Fedorov O, Bennett JM, Elkins JM, Spencer J.

Org Biomol Chem. 2018 Jan 3;16(2):336. doi: 10.1039/c7ob90195j.

PMID:
29256564
17.

Noncovalent Interactions of π Systems with Sulfur: The Atomic Chameleon of Molecular Recognition.

Motherwell WB, Moreno RB, Pavlakos I, Arendorf JRT, Arif T, Tizzard GJ, Coles SJ, Aliev AE.

Angew Chem Int Ed Engl. 2018 Jan 26;57(5):1193-1198. doi: 10.1002/anie.201708485. Epub 2017 Dec 28.

PMID:
29194884
18.

Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase.

Asquith CRM, Laitinen T, Bennett JM, Godoi PH, East MP, Tizzard GJ, Graves LM, Johnson GL, Dornsife RE, Wells CI, Elkins JM, Willson TM, Zuercher WJ.

ChemMedChem. 2018 Jan 8;13(1):48-66. doi: 10.1002/cmdc.201700663. Epub 2017 Nov 27.

19.

Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety.

Sansook S, Ocasio CA, Day IJ, Tizzard GJ, Coles SJ, Fedorov O, Bennett JM, Elkins JM, Spencer J.

Org Biomol Chem. 2017 Oct 18;15(40):8655-8660. doi: 10.1039/c7ob02289a. Erratum in: Org Biomol Chem. 2018 Jan 3;16(2):336.

20.

Base-Controlled Diastereoselective Synthesis of Either anti- or syn-β-Aminonitriles.

Anderson JC, Campbell IB, Campos S, Rundell CD, Shannon J, Tizzard GJ.

Org Lett. 2017 Apr 7;19(7):1918-1921. doi: 10.1021/acs.orglett.7b00679. Epub 2017 Mar 21.

PMID:
28322059

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