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Items: 1 to 20 of 49

1.

Intramolecular Metal Free N-N Bond Formation with Heteroaromatic Amines: Mild Access to Fused-Triazapentalene Derivatives.

Daniel M, Hiebel MA, Guillaumet G, Pasquinet E, Suzenet F.

Chemistry. 2019 Dec 24. doi: 10.1002/chem.201905558. [Epub ahead of print]

PMID:
31872461
2.

Bis(het)aryl-1,2,3-triazole quinuclidines as α7 nicotinic acetylcholine receptor ligands: Synthesis, structure affinity relationships, agonism activity, [18F]-radiolabeling and PET study in rats.

Ouach A, Vercouillie J, Bertrand E, Rodrigues N, Pin F, Serriere S, Boiaryna L, Chartier A, Percina N, Tangpong P, Gulhan Z, Mothes C, Deloye JB, Guilloteau D, Page G, Suzenet F, Buron F, Chalon S, Routier S.

Eur J Med Chem. 2019 Oct 1;179:449-469. doi: 10.1016/j.ejmech.2019.06.049. Epub 2019 Jun 27.

PMID:
31271958
3.

An original class of small sized molecules as versatile fluorescent probes for cellular imaging.

Sirbu D, Diharce J, Martinić I, Chopin N, Eliseeva SV, Guillaumet G, Petoud S, Bonnet P, Suzenet F.

Chem Commun (Camb). 2019 Jul 2;55(54):7776-7779. doi: 10.1039/c9cc03765a.

PMID:
31210218
4.

Organocatalytic aza-Michael Reaction to 3-Vinyl-1,2,4-triazines as a Valuable Bifunctional Platform.

Buttard F, Berthonneau C, Hiebel MA, Brière JF, Suzenet F.

J Org Chem. 2019 Mar 15;84(6):3702-3714. doi: 10.1021/acs.joc.9b00141. Epub 2019 Mar 1.

PMID:
30791682
5.

Palladium-Catalyzed C3-Arylations of 1 H- and 2 H-Pyrazolo[4,3- b]pyridines on Water.

Faarasse S, El Kazzouli S, Suzenet F, Guillaumet G.

J Org Chem. 2018 Oct 19;83(20):12847-12854. doi: 10.1021/acs.joc.8b01728. Epub 2018 Oct 4.

PMID:
30240222
6.

A Novel Polyaminocarboxylate Compound To Treat Murine Pulmonary Aspergillosis by Interfering with Zinc Metabolism.

Laskaris P, Vicentefranqueira R, Helynck O, Jouvion G, Calera JA, du Merle L, Suzenet F, Buron F, de Sousa RA, Mansuy D, Cavaillon JM, Latgé JP, Munier-Lehmann H, Ibrahim-Granet O.

Antimicrob Agents Chemother. 2018 May 25;62(6). pii: e02510-17. doi: 10.1128/AAC.02510-17. Print 2018 Jun.

7.

Efficient synthesis and first regioselective C-6 direct arylation of imidazo[2,1-c][1,2,4]triazine scaffold and their evaluation in H2O2-induced oxidative stress.

Loubidi M, Jouha J, Tber Z, Khouili M, Suzenet F, Akssira M, Erdogan MA, Köse FA, Dagcı T, Armagan G, Saso L, Guillaumet G.

Eur J Med Chem. 2018 Feb 10;145:113-123. doi: 10.1016/j.ejmech.2017.12.081. Epub 2017 Dec 27.

PMID:
29324335
8.

"On Water" Direct C-3 Arylation of 2H-Pyrazolo[3,4-b]pyridines.

Faarasse S, El Kazzouli S, Naas M, Jouha J, Suzenet F, Guillaumet G.

J Org Chem. 2017 Dec 1;82(23):12300-12306. doi: 10.1021/acs.joc.7b02136. Epub 2017 Nov 13.

PMID:
29090922
9.

Dual role of mitochondria in producing melatonin and driving GPCR signaling to block cytochrome c release.

Suofu Y, Li W, Jean-Alphonse FG, Jia J, Khattar NK, Li J, Baranov SV, Leronni D, Mihalik AC, He Y, Cecon E, Wehbi VL, Kim J, Heath BE, Baranova OV, Wang X, Gable MJ, Kretz ES, Di Benedetto G, Lezon TR, Ferrando LM, Larkin TM, Sullivan M, Yablonska S, Wang J, Minnigh MB, Guillaumet G, Suzenet F, Richardson RM, Poloyac SM, Stolz DB, Jockers R, Witt-Enderby PA, Carlisle DL, Vilardaga JP, Friedlander RM.

Proc Natl Acad Sci U S A. 2017 Sep 19;114(38):E7997-E8006. doi: 10.1073/pnas.1705768114. Epub 2017 Sep 5.

10.

Domino Aza-Michael-ih-Diels-Alder Reaction to Various 3-Vinyl-1,2,4-triazines: Access to Polysubstituted Tetrahydro-1,6-naphthyridines.

Jouha J, Buttard F, Lorion M, Berthonneau C, Khouili M, Hiebel MA, Guillaumet G, Brière JF, Suzenet F.

Org Lett. 2017 Sep 15;19(18):4770-4773. doi: 10.1021/acs.orglett.7b02132. Epub 2017 Aug 31.

PMID:
28857570
11.

Design and validation of the first cell-impermeant melatonin receptor agonist.

Gbahou F, Cecon E, Viault G, Gerbier R, Jean-Alphonse F, Karamitri A, Guillaumet G, Delagrange P, Friedlander RM, Vilardaga JP, Suzenet F, Jockers R.

Br J Pharmacol. 2017 Jul;174(14):2409-2421. doi: 10.1111/bph.13856. Epub 2017 Jun 11.

12.

Synthesis of new heterocyclic compounds based on pyrazolopyridine scaffold and evaluation of their neuroprotective potential in MPP+-induced neurodegeneration.

Jouha J, Loubidi M, Bouali J, Hamri S, Hafid A, Suzenet F, Guillaumet G, Dagcı T, Khouili M, Aydın F, Saso L, Armagan G.

Eur J Med Chem. 2017 Mar 31;129:41-52. doi: 10.1016/j.ejmech.2017.02.019. Epub 2017 Feb 11.

PMID:
28214632
13.

Nitroimidazole derivatives of polypyridyl ruthenium complexes: Towards understanding their anticancer activity and mode of action.

Mazuryk O, Krysiak-Foria O, Żak A, Suzenet F, Ptak-Belowska A, Brzozowski T, Stochel G, Brindell M.

Eur J Pharm Sci. 2017 Apr 1;101:43-55. doi: 10.1016/j.ejps.2017.01.020. Epub 2017 Jan 28.

PMID:
28137470
14.

30ièmes Journées Franco-Belges de Pharmacochimie.

Aci-Sèche S, Buron F, Plé K, Robin L, Suzenet F, Routier S.

Pharmaceuticals (Basel). 2016 Nov 18;9(4). pii: E73.

15.

Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity.

Couhert A, Delagrange P, Caignard DH, Chartier A, Suzenet F, Guillaumet G.

Eur J Med Chem. 2016 Feb 15;109:268-75. doi: 10.1016/j.ejmech.2016.01.008. Epub 2016 Jan 12.

PMID:
26785296
16.

Design of α7 nicotinic acetylcholine receptor ligands using the (het)Aryl-1,2,3-triazole core: Synthesis, in vitro evaluation and SAR studies.

Ouach A, Pin F, Bertrand E, Vercouillie J, Gulhan Z, Mothes C, Deloye JB, Guilloteau D, Suzenet F, Chalon S, Routier S.

Eur J Med Chem. 2016 Jan 1;107:153-64. doi: 10.1016/j.ejmech.2015.11.001. Epub 2015 Nov 10.

PMID:
26580980
17.

Rational Design, Pharmacomodulation, and Synthesis of Dual 5-Hydroxytryptamine 7 (5-HT7)/5-Hydroxytryptamine 2A (5-HT2A) Receptor Antagonists and Evaluation by [(18)F]-PET Imaging in a Primate Brain.

Deau E, Robin E, Voinea R, Percina N, Satała G, Finaru AL, Chartier A, Tamagnan G, Alagille D, Bojarski AJ, Morisset-Lopez S, Suzenet F, Guillaumet G.

J Med Chem. 2015 Oct 22;58(20):8066-96. doi: 10.1021/acs.jmedchem.5b00874. Epub 2015 Oct 5.

PMID:
26348247
18.

Sequential Michael Addition and Enamine-Promoted Inverse Electron Demanding Diels-Alder Reaction upon 3-Vinyl-1,2,4-triazine Platforms.

Lorion M, Guillaumet G, Brière JF, Suzenet F.

Org Lett. 2015 Jun 19;17(12):3154-7. doi: 10.1021/acs.orglett.5b01487. Epub 2015 Jun 11.

PMID:
26066589
19.

A Pyridine-Based Ligand with Two Hydrazine Functions for Lanthanide Chelation: Remarkable Kinetic Inertness for a Linear, Bishydrated Complex.

Bonnet CS, Laine S, Buron F, Tircsó G, Pallier A, Helm L, Suzenet F, Tóth É.

Inorg Chem. 2015 Jun 15;54(12):5991-6003. doi: 10.1021/acs.inorgchem.5b00804. Epub 2015 Jun 1.

PMID:
26030671
20.

The biological effect of the nitroimidazole derivative of a polypyridyl ruthenium complex on cancer and endothelial cells.

Mazuryk O, Suzenet F, Kieda C, Brindell M.

Metallomics. 2015 Mar;7(3):553-66. doi: 10.1039/c5mt00037h.

PMID:
25711770

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