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Items: 18

1.

Novel derivatives of anaplastic lymphoma kinase inhibitors: Synthesis, radiolabeling, and preliminary biological studies of fluoroethyl analogues of crizotinib, alectinib, and ceritinib.

Radaram B, Pisaneschi F, Rao Y, Yang P, Piwnica-Worms D, Alauddin MM.

Eur J Med Chem. 2019 Aug 9;182:111571. doi: 10.1016/j.ejmech.2019.111571. [Epub ahead of print]

PMID:
31425908
2.

The 3S Enantiomer Drives Enolase Inhibitory Activity in SF2312 and Its Analogues.

Pisaneschi F, Lin YH, Leonard PG, Satani N, Yan VC, Hammoudi N, Raghavan S, Link TM, K Georgiou D, Czako B, Muller FL.

Molecules. 2019 Jul 9;24(13). pii: E2510. doi: 10.3390/molecules24132510.

3.

Multiwalled Carbon Nanotubes for Combination Therapy: a Biodistribution and Efficacy Pilot Study.

Biagiotti G, Pisaneschi F, Gammon ST, Machetti F, Ligi MC, Giambastiani G, Tuci G, Powell E, Piwnica-Worms H, Pranzini E, Paoli P, Cicchi S, Piwnica-Worms D.

J Mater Chem B. 2019 Apr 28;7(16):2678-2687. doi: 10.1039/C8TB03299H. Epub 2019 Mar 12.

PMID:
31073405
4.

Development of a Potential Gallium-68-Labelled Radiotracer Based on DOTA-Curcumin for Colon-Rectal Carcinoma: From Synthesis to In Vivo Studies.

Orteca G, Pisaneschi F, Rubagotti S, Liu TW, Biagiotti G, Piwnica-Worms D, Iori M, Capponi PC, Ferrari E, Asti M.

Molecules. 2019 Feb 12;24(3). pii: E644. doi: 10.3390/molecules24030644.

5.

Caspase-3 Substrates for Noninvasive Pharmacodynamic Imaging of Apoptosis by PET/CT.

Engel BJ, Gammon ST, Chaudhari R, Lu Z, Pisaneschi F, Yang H, Ornelas A, Yan V, Kelderhouse L, Najjar AM, Tong WP, Zhang S, Piwnica-Worms D, Bast RC Jr, Millward SW.

Bioconjug Chem. 2018 Sep 19;29(9):3180-3195. doi: 10.1021/acs.bioconjchem.8b00514. Epub 2018 Aug 31.

6.

Automated, Resin-Based Method to Enhance the Specific Activity of Fluorine-18 Clicked PET Radiotracers.

Pisaneschi F, Kelderhouse LE, Hardy A, Engel BJ, Mukhopadhyay U, Gonzalez-Lepera C, Gray JP, Ornelas A, Takahashi TT, Roberts RW, Fiacco SV, Piwnica-Worms D, Millward SW.

Bioconjug Chem. 2017 Feb 15;28(2):583-589. doi: 10.1021/acs.bioconjchem.6b00678. Epub 2017 Feb 2.

7.

SF2312 is a natural phosphonate inhibitor of enolase.

Leonard PG, Satani N, Maxwell D, Lin YH, Hammoudi N, Peng Z, Pisaneschi F, Link TM, Lee GR 4th, Sun D, Prasad BAB, Di Francesco ME, Czako B, Asara JM, Wang YA, Bornmann W, DePinho RA, Muller FL.

Nat Chem Biol. 2016 Dec;12(12):1053-1058. doi: 10.1038/nchembio.2195. Epub 2016 Oct 10.

8.

Identification of ABC Transporter Interaction of a Novel Cyanoquinoline Radiotracer and Implications for Tumour Imaging by Positron Emission Tomography.

Slade RL, Pisaneschi F, Nguyen QD, Smith G, Carroll L, Beckley A, Kaliszczak MA, Aboagye EO.

PLoS One. 2016 Aug 23;11(8):e0161427. doi: 10.1371/journal.pone.0161427. eCollection 2016.

9.

Positron emission tomographic imaging of CXCR4 in cancer: challenges and promises.

George GP, Pisaneschi F, Nguyen QD, Aboagye EO.

Mol Imaging. 2014;13. doi: 10.2310/7290.2014.00041. Review.

PMID:
25341373
10.

Scavenging strategy for specific activity improvement: application to a new CXCR4-specific cyclopentapeptide positron emission tomography tracer.

George GP, Pisaneschi F, Stevens E, Nguyen QD, Åberg O, Spivey AC, Aboagye EO.

J Labelled Comp Radiopharm. 2013 Nov;56(13):679-85. doi: 10.1002/jlcr.3095. Epub 2013 Jul 16.

PMID:
25196030
11.

Preclinical evaluation of 3-18F-fluoro-2,2-dimethylpropionic acid as an imaging agent for tumor detection.

Witney TH, Pisaneschi F, Alam IS, Trousil S, Kaliszczak M, Twyman F, Brickute D, Nguyen QD, Schug Z, Gottlieb E, Aboagye EO.

J Nucl Med. 2014 Sep;55(9):1506-12. doi: 10.2967/jnumed.114.140343. Epub 2014 Jul 10. Erratum in: J Nucl Med. 2014 Nov;55(11):1914.

12.

Preclinical evaluation of a CXCR4-specific (68)Ga-labelled TN14003 derivative for cancer PET imaging.

George GP, Stevens E, Åberg O, Nguyen QD, Pisaneschi F, Spivey AC, Aboagye EO.

Bioorg Med Chem. 2014 Jan 15;22(2):796-803. doi: 10.1016/j.bmc.2013.12.012. Epub 2013 Dec 11.

PMID:
24365390
13.

Synthesis of a new fluorine-18 glycosylated 'click' cyanoquinoline for the imaging of epidermal growth factor receptor.

Pisaneschi F, Slade RL, Iddon L, George GP, Nguyen QD, Spivey AC, Aboagye EO.

J Labelled Comp Radiopharm. 2014 Feb;57(2):92-6. doi: 10.1002/jlcr.3170. Epub 2013 Dec 5.

PMID:
24307532
14.

Development of a new epidermal growth factor receptor positron emission tomography imaging agent based on the 3-cyanoquinoline core: synthesis and biological evaluation.

Pisaneschi F, Nguyen QD, Shamsaei E, Glaser M, Robins E, Kaliszczak M, Smith G, Spivey AC, Aboagye EO.

Bioorg Med Chem. 2010 Sep 15;18(18):6634-45. doi: 10.1016/j.bmc.2010.08.004. Epub 2010 Aug 6.

15.

Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin alphavbeta3 and alphavbeta5 ligands.

Salvati M, Cordero FM, Pisaneschi F, Melani F, Gratteri P, Cini N, Bottoncetti A, Brandi A.

Bioorg Med Chem. 2008 Apr 15;16(8):4262-71. doi: 10.1016/j.bmc.2008.02.080. Epub 2008 Feb 29.

PMID:
18343671
16.

Application of Mosher's method for absolute configuration assignment and resolution of 2-hydroxypyrrolizidinones.

Cordero FM, Pisaneschi F, Salvati M, Valenza S, Faggi C, Brandi A.

Chirality. 2005 Mar;17(3):149-53.

PMID:
15704198
17.

A new bicyclic dipeptide isostere with pyrrolizidinone skeleton.

Cordero FM, Pisaneschi F, Meschini Batista K, Valenza S, Machetti F, Brandi A.

J Org Chem. 2005 Feb 4;70(3):856-67.

PMID:
15675843
18.

Selective ring contraction of 5-spirocyclopropane isoxazolidines mediated by acids.

Cordero FM, Pisaneschi F, Salvati M, Paschetta V, Ollivier J, Salaün J, Brandi A.

J Org Chem. 2003 Apr 18;68(8):3271-80.

PMID:
12688801

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