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Items: 1 to 20 of 88

1.

Synthesis of indole based acetohydrazide analogs: Their in vitro and in silico thymidine phosphorylase studies.

Taha M, Aldhamin EAJ, Almandil NB, Anouar EH, Uddin N, Alomari M, Rahim F, Adalat B, Ibrahim M, Nawaz F, Iqbal N, Alghanem B, Altolayyan A, Khan KM.

Bioorg Chem. 2020 Mar 12;98:103745. doi: 10.1016/j.bioorg.2020.103745. [Epub ahead of print]

PMID:
32200327
2.

Exploring efficacy of indole-based dual inhibitors for α-glucosidase and α-amylase enzymes: In silico, biochemical and kinetic studies.

Kawde AN, Taha M, Alansari RS, Almandil NB, Anouar EH, Uddin N, Rahim F, Chigurupati S, Nawaz M, Hayat S, Ibrahim M, Elakurthy PK, Vijayan V, Morsy M, Ibrahim H, Baig N, Khan KM.

Int J Biol Macromol. 2020 Mar 12;154:217-232. doi: 10.1016/j.ijbiomac.2020.03.090. [Epub ahead of print]

PMID:
32173438
3.

Synthesis, α-glycosidase inhibitory potential and molecular docking study of benzimidazole derivatives.

Taha M, Rahim F, Zaman K, Selvaraj M, Uddin N, Farooq RK, Nawaz M, Sajid M, Nawaz F, Ibrahim M, Khan KM.

Bioorg Chem. 2020 Jan;95:103555. doi: 10.1016/j.bioorg.2019.103555. Epub 2019 Dec 26.

PMID:
31911306
4.

Synthesis, in vitro alpha-glucosidase inhibitory potential of benzimidazole bearing bis-Schiff bases and their molecular docking study.

Rahim F, Zaman K, Taha M, Ullah H, Ghufran M, Wadood A, Rehman W, Uddin N, Shah SAA, Sajid M, Nawaz F, Khan KM.

Bioorg Chem. 2020 Jan;94:103394. doi: 10.1016/j.bioorg.2019.103394. Epub 2019 Oct 23.

PMID:
31699396
5.

Synthesis of new isoquinoline-base-oxadiazole derivatives as potent inhibitors of thymidine phosphorylase and molecular docking study.

Zaman K, Rahim F, Taha M, Wadood A, Shah SAA, Ahmed QU, Zakaria ZA.

Sci Rep. 2019 Nov 5;9(1):16015. doi: 10.1038/s41598-019-52100-0.

6.

Synthesis of Novel Triazinoindole-Based Thiourea Hybrid: A Study on α-Glucosidase Inhibitors and Their Molecular Docking.

Taha M, Alshamrani FJ, Rahim F, Hayat S, Ullah H, Zaman K, Imran S, Khan KM, Naz F.

Molecules. 2019 Oct 23;24(21). pii: E3819. doi: 10.3390/molecules24213819.

7.

New triazinoindole bearing thiazole/oxazole analogues: Synthesis, α-amylase inhibitory potential and molecular docking study.

Rahim F, Tariq S, Taha M, Ullah H, Zaman K, Uddin I, Wadood A, Khan AA, Rehman AU, Uddin N, Zafar S, Shah SAA.

Bioorg Chem. 2019 Nov;92:103284. doi: 10.1016/j.bioorg.2019.103284. Epub 2019 Sep 17.

PMID:
31546207
8.

Design, synthesis, in vitro evaluation, molecular docking and ADME properties studies of hybrid bis-coumarin with thiadiazole as a new inhibitor of Urease.

Alomari M, Taha M, Imran S, Jamil W, Selvaraj M, Uddin N, Rahim F.

Bioorg Chem. 2019 Nov;92:103235. doi: 10.1016/j.bioorg.2019.103235. Epub 2019 Aug 30.

PMID:
31494327
9.

Synthesis, anti-leishmanial and molecular docking study of bis-indole derivatives.

Taha M, Uddin I, Gollapalli M, Almandil NB, Rahim F, Farooq RK, Nawaz M, Ibrahim M, Alqahtani MA, Bamarouf YA, Selvaraj M.

BMC Chem. 2019 Aug 6;13(1):102. doi: 10.1186/s13065-019-0617-4. eCollection 2019 Dec.

10.

Indole bearing thiadiazole analogs: synthesis, β-glucuronidase inhibition and molecular docking study.

Almandil NB, Taha M, Gollapalli M, Rahim F, Ibrahim M, Mosaddik A, Anouar EH.

BMC Chem. 2019 Feb 4;13(1):14. doi: 10.1186/s13065-019-0522-x. eCollection 2019 Dec.

11.

Synthesis of quinoline derivatives as diabetic II inhibitors and molecular docking studies.

Taha M, Sultan S, Imran S, Rahim F, Zaman K, Wadood A, Ur Rehman A, Uddin N, Mohammed Khan K.

Bioorg Med Chem. 2019 Sep 15;27(18):4081-4088. doi: 10.1016/j.bmc.2019.07.035. Epub 2019 Jul 20.

PMID:
31378594
12.

Synthesis of new arylhydrazide bearing Schiff bases/thiazolidinone: α-Amylase, urease activities and their molecular docking studies.

Rahim F, Taha M, Ullah H, Wadood A, Selvaraj M, Rab A, Sajid M, Shah SAA, Uddin N, Gollapalli M.

Bioorg Chem. 2019 Oct;91:103112. doi: 10.1016/j.bioorg.2019.103112. Epub 2019 Jul 9.

PMID:
31349115
13.

Synthesis of oxadiazole-coupled-thiadiazole derivatives as a potent β-glucuronidase inhibitors and their molecular docking study.

Taha M, Imran S, Alomari M, Rahim F, Wadood A, Mosaddik A, Uddin N, Gollapalli M, Alqahtani MA, Bamarouf YA.

Bioorg Med Chem. 2019 Jul 15;27(14):3145-3155. doi: 10.1016/j.bmc.2019.05.049. Epub 2019 Jun 4.

PMID:
31196753
14.

Synthesis, In vitro α-Glucosidase Inhibitory Potential and Molecular Docking Studies of 2-Amino-1,3,4-Oxadiazole Derivatives.

Ullah H, Rahim F, Taha M, Hussain R, Wadood A, Nawaz M, Wahab Z, Kanwal, Khan KM.

Med Chem. 2019 Jun 12. doi: 10.2174/1573406415666190612150447. [Epub ahead of print]

PMID:
31195948
15.

Synthesis, in vitro urease inhibitory potential and molecular docking study of Benzimidazole analogues.

Zaman K, Rahim F, Taha M, Ullah H, Wadood A, Nawaz M, Khan F, Wahab Z, Shah SAA, Rehman AU, Kawde AN, Gollapalli M.

Bioorg Chem. 2019 Aug;89:103024. doi: 10.1016/j.bioorg.2019.103024. Epub 2019 May 31.

PMID:
31176853
16.

Synthesis, thymidine phosphorylase, angiogenic inhibition and molecular docking study of isoquinoline derivatives.

Zaman K, Rahim F, Taha M, Wadood A, Adnan Ali Shah S, Gollapalli M, Ullah F, Ahmed A.

Bioorg Chem. 2019 Aug;89:102999. doi: 10.1016/j.bioorg.2019.102999. Epub 2019 May 21.

PMID:
31151055
17.

Synthesis of Chromen-4-One-Oxadiazole Substituted Analogs as Potent β-Glucuronidase Inhibitors.

Taha M, Rahim F, Ali M, Khan MN, Alqahtani MA, Bamarouf YA, Gollapalli M, Farooq RK, Shah SAA, Ahmed QU, Zakaria ZA.

Molecules. 2019 Apr 18;24(8). pii: E1528. doi: 10.3390/molecules24081528.

18.

A mutation in the major autophagy gene, WIPI2, associated with global developmental abnormalities.

Jelani M, Dooley HC, Gubas A, Mohamoud HSA, Khan MTM, Ali Z, Kang C, Rahim F, Jan A, Vadgama N, Khan MI, Al-Aama JY, Khan A, Tooze SA, Nasir J.

Brain. 2019 May 1;142(5):1242-1254. doi: 10.1093/brain/awz075.

19.

Synthesis of Thymidine Phosphorylase Inhibitor Based on Quinoxaline Derivatives and Their Molecular Docking Study.

Almandil NB, Taha M, Farooq RK, Alhibshi A, Ibrahim M, Anouar EH, Gollapalli M, Rahim F, Nawaz M, Shah SAA, Ahmed QU, Zakaria ZA.

Molecules. 2019 Mar 13;24(6). pii: E1002. doi: 10.3390/molecules24061002.

20.

Synthesis, Molecular Docking and β-Glucuronidase Inhibitory Potential of Indole Base Oxadiazole Derivatives.

Anouar EH, Moustapha ME, Taha M, Geesi MH, Farag ZR, Rahim F, Almandil NB, Farooq RK, Nawaz M, Mosaddik A.

Molecules. 2019 Mar 8;24(5). pii: E963. doi: 10.3390/molecules24050963.

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