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Items: 13

1.

Identification of highly potent and selective MMP2 inhibitors addressing the S1' subsite with d-proline-based compounds.

Lenci E, Innocenti R, Di Francescantonio T, Menchi G, Bianchini F, Contini A, Trabocchi A.

Bioorg Med Chem. 2019 May 1;27(9):1891-1902. doi: 10.1016/j.bmc.2019.03.043. Epub 2019 Mar 22.

PMID:
30926311
2.

Bicyclic acetals: biological relevance, scaffold analysis, and applications in diversity-oriented synthesis.

Lenci E, Menchi G, Saldívar-Gonzalez FI, Medina-Franco JL, Trabocchi A.

Org Biomol Chem. 2019 Jan 31;17(5):1037-1052. doi: 10.1039/c8ob02808g. Review.

PMID:
30620036
3.

Smart Design of Small-Molecule Libraries: When Organic Synthesis Meets Cheminformatics.

Lenci E, Trabocchi A.

Chembiochem. 2019 May 2;20(9):1115-1123. doi: 10.1002/cbic.201800751. Epub 2019 Mar 19. Review.

PMID:
30589187
4.

Diversity-Oriented Synthesis and Chemoinformatic Analysis of the Molecular Diversity of sp3-Rich Morpholine Peptidomimetics.

Lenci E, Innocenti R, Menchi G, Trabocchi A.

Front Chem. 2018 Oct 30;6:522. doi: 10.3389/fchem.2018.00522. eCollection 2018.

5.

Short synthesis of polyfunctional sp3-rich threonine-derived morpholine scaffolds.

Lenci E, Rossi A, Menchi G, Trabocchi A.

Org Biomol Chem. 2017 Nov 22;15(45):9710-9717. doi: 10.1039/c7ob02454a.

PMID:
29125175
6.

Corrigendum to "Design and synthesis of bicyclic acetals as Beta Secretase (BACE1) inhibitors" [Bioorg. Med. Chem. 25 (2017) 5077-5083].

Innocenti R, Lenci E, Menchi G, Pupi A, Trabocchi A.

Bioorg Med Chem. 2017 Dec 15;25(24):6724-6725. doi: 10.1016/j.bmc.2017.10.019. Epub 2017 Nov 1. No abstract available.

PMID:
29111366
7.

Design and synthesis of bicyclic acetals as Beta Secretase (BACE1) inhibitors.

Innocenti R, Lenci E, Menchi G, Pupi A, Trabocchi A.

Bioorg Med Chem. 2017 Oct 1;25(19):5077-5083. doi: 10.1016/j.bmc.2017.03.030. Epub 2017 Mar 18. Erratum in: Bioorg Med Chem. 2017 Dec 15;25(24):6724-6725.

PMID:
28359674
8.

Iridium-Catalyzed Reductive Strecker Reaction for Late-Stage Amide and Lactam Cyanation.

Fuentes de Arriba ÁL, Lenci E, Sonawane M, Formery O, Dixon DJ.

Angew Chem Int Ed Engl. 2017 Mar 20;56(13):3655-3659. doi: 10.1002/anie.201612367. Epub 2017 Feb 24.

PMID:
28233919
9.

Identification of Novel Human Breast Carcinoma (MDA-MB-231) Cell Growth Modulators from a Carbohydrate-Based Diversity Oriented Synthesis Library.

Lenci E, Innocenti R, Biagioni A, Menchi G, Bianchini F, Trabocchi A.

Molecules. 2016 Oct 20;21(10). pii: E1405.

10.

Insight to the binding mode of triazole RGD-peptidomimetics to integrin-rich cancer cells by NMR and molecular modeling.

Vasile F, Menchi G, Lenci E, Guarna A, Potenza D, Trabocchi A.

Bioorg Med Chem. 2016 Mar 1;24(5):989-94. doi: 10.1016/j.bmc.2016.01.023. Epub 2016 Jan 14.

PMID:
26818999
11.

Two-step one-pot synthesis of dihydropyrazinones as Xaa-Ser dipeptide isosteres through morpholine acetal rearrangement.

Lenci E, Innocenti R, Menchi G, Faggi C, Trabocchi A.

Org Biomol Chem. 2015 Jul 7;13(25):7013-9. doi: 10.1039/c5ob00783f. Epub 2015 Jun 1.

PMID:
26030011
12.

Skeletal diversity from carbohydrates: use of mannose for the diversity-oriented synthesis of polyhydroxylated compounds.

Lenci E, Menchi G, Guarna A, Trabocchi A.

J Org Chem. 2015 Feb 20;80(4):2182-91. doi: 10.1021/jo502701c. Epub 2015 Feb 11.

PMID:
25636147
13.

Diversity-oriented synthesis as a tool for chemical genetics.

Lenci E, Guarna A, Trabocchi A.

Molecules. 2014 Oct 14;19(10):16506-28. doi: 10.3390/molecules191016506. Review.

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