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Items: 1 to 20 of 35

1.

Nor-Lignans: Occurrence in Plants and Biological Activities-A Review.

Frezza C, Venditti A, Toniolo C, De Vita D, Franceschin M, Ventrone A, Tomassini L, Foddai S, Guiso M, Nicoletti M, Serafini M, Bianco A.

Molecules. 2020 Jan 3;25(1). pii: E197. doi: 10.3390/molecules25010197. Review.

2.

Anti-Inflammatory and Antioxidant Properties of Dehydrated Potato-Derived Bioactive Compounds in Intestinal Cells.

Basilicata MG, Pepe G, Rapa SF, Merciai F, Ostacolo C, Manfra M, Di Sarno V, Autore G, De Vita D, Marzocco S, Campiglia P.

Int J Mol Sci. 2019 Dec 3;20(23). pii: E6087. doi: 10.3390/ijms20236087.

3.

Towards a new application of amaranth seed oil as an agent against Candida albicans.

De Vita D, Messore A, Toniolo C, Frezza C, Scipione L, Bertea CM, Micera M, Di Sarno V, Madia VN, Pindinello I, Roscilli P, Botto A, Simonetti G, Orekhova A, Manfredini S, Costi R, Di Santo R.

Nat Prod Res. 2019 Dec 4:1-6. doi: 10.1080/14786419.2019.1696335. [Epub ahead of print]

PMID:
31795749
4.

Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement.

Gomes JC, Cianni L, Ribeiro J, Dos Reis Rocho F, da Costa Martins Silva S, Batista PHJ, Moraes CB, Franco CH, Freitas-Junior LHG, Kenny PW, Leitão A, Burtoloso ACB, de Vita D, Montanari CA.

Bioorg Med Chem. 2019 Nov 15;27(22):115083. doi: 10.1016/j.bmc.2019.115083. Epub 2019 Aug 28.

PMID:
31561938
5.

Tegaserod for the Treatment of Irritable Bowel Syndrome.

Madia VN, Messore A, Saccoliti F, Tudino V, De Leo A, De Vita D, Bortolami M, Scipione L, Pindinello I, Costi R, Di Santo R.

Antiinflamm Antiallergy Agents Med Chem. 2019 Sep 11. doi: 10.2174/1871523018666190911121306. [Epub ahead of print]

PMID:
31518227
6.

Pedicularis L. Genus: Systematics, Botany, Phytochemistry, Chemotaxonomy, Ethnopharmacology, and Other.

Frezza C, Venditti A, Toniolo C, Vita D, Serafini I, Ciccòla A, Franceschin M, Ventrone A, Tomassini L, Foddai S, Guiso M, Nicoletti M, Bianco A, Serafini M.

Plants (Basel). 2019 Aug 27;8(9). pii: E306. doi: 10.3390/plants8090306. Review.

7.

Comparison of different methods for the extraction of cannabinoids from cannabis.

De Vita D, Madia VN, Tudino V, Saccoliti F, De Leo A, Messore A, Roscilli P, Botto A, Pindinello I, Santilli G, Scipione L, Costi R, Di Santo R.

Nat Prod Res. 2019 Apr 29:1-7. doi: 10.1080/14786419.2019.1601194. [Epub ahead of print]

PMID:
31035854
8.

Searching for new agents active against Candida albicans biofilm: A series of indole derivatives, design, synthesis and biological evaluation.

Pandolfi F, D'Acierno F, Bortolami M, De Vita D, Gallo F, De Meo A, Di Santo R, Costi R, Simonetti G, Scipione L.

Eur J Med Chem. 2019 Mar 1;165:93-106. doi: 10.1016/j.ejmech.2019.01.012. Epub 2019 Jan 9.

PMID:
30660829
9.

Secondary metabolites of Tilia tomentosa Moench inflorescences collected in Central Italy: chemotaxonomy relevance and phytochemical rationale of traditional use.

Frezza C, De Vita D, Spinaci G, Sarandrea M, Venditti A, Bianco A.

Nat Prod Res. 2019 Jan 12:1-8. doi: 10.1080/14786419.2018.1550487. [Epub ahead of print]

PMID:
30638062
10.

Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents.

Saccoliti F, Madia VN, Tudino V, De Leo A, Pescatori L, Messore A, De Vita D, Scipione L, Brun R, Kaiser M, Mäser P, Calvet CM, Jennings GK, Podust LM, Pepe G, Cirilli R, Faggi C, Di Marco A, Battista MR, Summa V, Costi R, Di Santo R.

J Med Chem. 2019 Feb 14;62(3):1330-1347. doi: 10.1021/acs.jmedchem.8b01464. Epub 2019 Jan 23.

PMID:
30615444
11.

Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity.

Messore A, Madia VN, Pescatori L, Saccoliti F, Tudino V, De Leo A, Bortolami M, De Vita D, Scipione L, Pepi F, Costi R, Rivara S, Scalvini L, Mor M, Ferrara FF, Pavoni E, Roscilli G, Cassinelli G, Milazzo FM, Battistuzzi G, Di Santo R, Giannini G.

J Med Chem. 2018 Dec 13;61(23):10834-10859. doi: 10.1021/acs.jmedchem.8b01497. Epub 2018 Nov 29.

PMID:
30412404
12.

Experimental study and computational modelling of cruzain cysteine protease inhibition by dipeptidyl nitriles.

Dos Santos AM, Cianni L, De Vita D, Rosini F, Leitão A, Laughton CA, Lameira J, Montanari CA.

Phys Chem Chem Phys. 2018 Sep 26;20(37):24317-24328. doi: 10.1039/c8cp03320j.

PMID:
30211406
13.

Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents.

Saccoliti F, Madia VN, Tudino V, De Leo A, Pescatori L, Messore A, De Vita D, Scipione L, Brun R, Kaiser M, Mäser P, Calvet CM, Jennings GK, Podust LM, Costi R, Di Santo R.

Eur J Med Chem. 2018 Aug 5;156:53-60. doi: 10.1016/j.ejmech.2018.06.063. Epub 2018 Jun 28.

PMID:
30006174
14.

Leveraging the cruzain S3 subsite to increase affinity for reversible covalent inhibitors.

Cianni L, Sartori G, Rosini F, De Vita D, Pires G, Lopes BR, Leitão A, Burtoloso ACB, Montanari CA.

Bioorg Chem. 2018 Sep;79:285-292. doi: 10.1016/j.bioorg.2018.04.006. Epub 2018 Apr 26.

PMID:
29783099
15.

Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents.

Carradori S, Ortuso F, Petzer A, Bagetta D, De Monte C, Secci D, De Vita D, Guglielmi P, Zengin G, Aktumsek A, Alcaro S, Petzer JP.

Eur J Med Chem. 2018 Jan 1;143:1543-1552. doi: 10.1016/j.ejmech.2017.10.050. Epub 2017 Oct 19.

PMID:
29126727
16.

A comparative study of warheads for design of cysteine protease inhibitors.

Silva DG, Ribeiro JFR, De Vita D, Cianni L, Franco CH, Freitas-Junior LH, Moraes CB, Rocha JR, Burtoloso ACB, Kenny PW, Leitão A, Montanari CA.

Bioorg Med Chem Lett. 2017 Nov 15;27(22):5031-5035. doi: 10.1016/j.bmcl.2017.10.002. Epub 2017 Oct 3.

PMID:
29054358
17.

New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation.

Pandolfi F, De Vita D, Bortolami M, Coluccia A, Di Santo R, Costi R, Andrisano V, Alabiso F, Bergamini C, Fato R, Bartolini M, Scipione L.

Eur J Med Chem. 2017 Dec 1;141:197-210. doi: 10.1016/j.ejmech.2017.09.022. Epub 2017 Sep 18.

PMID:
29031067
18.

Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties.

De Vita D, Angeli A, Pandolfi F, Bortolami M, Costi R, Di Santo R, Suffredini E, Ceruso M, Del Prete S, Capasso C, Scipione L, Supuran CT.

J Enzyme Inhib Med Chem. 2017 Dec;32(1):798-804. doi: 10.1080/14756366.2017.1327522.

19.

Exploring the anti-biofilm activity of cinnamic acid derivatives in Candida albicans.

De Vita D, Simonetti G, Pandolfi F, Costi R, Di Santo R, D'Auria FD, Scipione L.

Bioorg Med Chem Lett. 2016 Dec 15;26(24):5931-5935. doi: 10.1016/j.bmcl.2016.10.091. Epub 2016 Nov 1.

PMID:
27838185
20.

New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation.

De Vita D, Pandolfi F, Ornano L, Feroci M, Chiarotto I, Sileno I, Pepi F, Costi R, Di Santo R, Scipione L.

J Enzyme Inhib Med Chem. 2016;31(sup4):106-113. Epub 2016 Sep 3.

PMID:
27594053

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