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Items: 1 to 20 of 171

1.

Novel method of treating macular degeneration: a patent evaluation (WO2018/107005).

Capasso C, Winum JY.

Expert Opin Ther Pat. 2019 Sep 1:1-4. doi: 10.1080/13543776.2019.1661991. [Epub ahead of print]

PMID:
31456444
2.

Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases.

Distinto S, Meleddu R, Ortuso F, Cottiglia F, Deplano S, Sequeira L, Melis C, Fois B, Angeli A, Capasso C, Angius R, Alcaro S, Supuran CT, Maccioni E.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):1526-1533. doi: 10.1080/14756366.2019.1654470.

3.

Anion Inhibition Profile of the β-Carbonic Anhydrase from the Opportunist Pathogenic Fungus Malassezia Restricta Involved in Dandruff and Seborrheic Dermatitis.

Prete SD, Angeli A, Ghobril C, Hitce J, Clavaud C, Marat X, Supuran CT, Capasso C.

Metabolites. 2019 Jul 18;9(7). pii: E147. doi: 10.3390/metabo9070147.

4.

The first activation study of the β-carbonic anhydrases from the pathogenic bacteria Brucella suis and Francisella tularensis with amines and amino acids.

Angeli A, Del Prete S, Pinteala M, Maier SS, Donald WA, Simionescu BC, Capasso C, Supuran CT.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):1178-1185. doi: 10.1080/14756366.2019.1630617.

5.

Seeking new approach for therapeutic treatment of cholera disease via inhibition of bacterial carbonic anhydrases: experimental and theoretical studies for sixteen benzenesulfonamide derivatives.

Gitto R, De Luca L, Mancuso F, Del Prete S, Vullo D, Supuran CT, Capasso C.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):1186-1192. doi: 10.1080/14756366.2019.1618292.

6.

Cloning, Purification, and Characterization of a β-Carbonic Anhydrase from Malassezia restricta, an Opportunistic Pathogen Involved in Dandruff and Seborrheic Dermatitis.

Del Prete S, Vullo D, Ghobril C, Hitce J, Clavaud C, Marat X, Capasso C, Supuran CT.

Int J Mol Sci. 2019 May 17;20(10). pii: E2447. doi: 10.3390/ijms20102447.

7.

Thermostability enhancement of the α-carbonic anhydrase from Sulfurihydrogenibium yellowstonense by using the anchoring-and-self-labelling-protein-tag system (ASLtag).

Del Prete S, Merlo R, Valenti A, Mattossovich R, Rossi M, Carginale V, Supuran CT, Perugino G, Capasso C.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):946-954. doi: 10.1080/14756366.2019.1605991.

8.

Activation Studies of the γ-Carbonic Anhydrases from the Antarctic Marine Bacteria Pseudoalteromonas haloplanktis and Colwellia psychrerythraea with Amino Acids and Amines.

Angeli A, Del Prete S, Osman SM, AlOthman Z, Donald WA, Capasso C, Supuran CT.

Mar Drugs. 2019 Apr 22;17(4). pii: E238. doi: 10.3390/md17040238.

9.

Comparison of the Sulfonamide Inhibition Profiles of the α-Carbonic Anhydrase Isoforms (SpiCA1, SpiCA2 and SpiCA3) Encoded by the Genome of the Scleractinian Coral Stylophora pistillata.

Del Prete S, Bua S, Alasmary FAS, AlOthman Z, Tambutté S, Zoccola D, Supuran CT, Capasso C.

Mar Drugs. 2019 Mar 1;17(3). pii: E146. doi: 10.3390/md17030146.

10.

Identification and characterization of the α-CA in the outer membrane vesicles produced by Helicobacter pylori.

Ronci M, Del Prete S, Puca V, Carradori S, Carginale V, Muraro R, Mincione G, Aceto A, Sisto F, Supuran CT, Grande R, Capasso C.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):189-195. doi: 10.1080/14756366.2018.1539716.

11.

Inhibition of bacterial α-, β- and γ-class carbonic anhydrases with selenazoles incorporating benzenesulfonamide moieties.

Angeli A, Pinteala M, Maier SS, Del Prete S, Capasso C, Simionescu BC, Supuran CT.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):244-249. doi: 10.1080/14756366.2018.1547287.

12.

Prostate cancer cells and exosomes in acidic condition show increased carbonic anhydrase IX expression and activity.

Logozzi M, Capasso C, Di Raimo R, Del Prete S, Mizzoni D, Falchi M, Supuran CT, Fais S.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):272-278. doi: 10.1080/14756366.2018.1538980.

13.

Inhibition of α-, β-, γ-, δ-, ζ- and η-class carbonic anhydrases from bacteria, fungi, algae, diatoms and protozoans with famotidine.

Angeli A, Pinteala M, Maier SS, Del Prete S, Capasso C, Simionescu BC, Supuran CT.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):644-650. doi: 10.1080/14756366.2019.1571273.

14.

An AGT-based protein-tag system for the labelling and surface immobilization of enzymes on E. coli outer membrane.

Merlo R, Del Prete S, Valenti A, Mattossovich R, Carginale V, Supuran CT, Capasso C, Perugino G.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):490-499. doi: 10.1080/14756366.2018.1559161.

15.

Click-tailed benzenesulfonamides as potent bacterial carbonic anhydrase inhibitors for targeting Mycobacterium tuberculosis and Vibrio cholerae.

Bua S, Osman SM, Del Prete S, Capasso C, AlOthman Z, Nocentini A, Supuran CT.

Bioorg Chem. 2019 May;86:183-186. doi: 10.1016/j.bioorg.2019.01.065. Epub 2019 Jan 29.

PMID:
30716618
16.

Phaeodactylum tricornutum as a model organism for testing the membrane penetrability of sulphonamide carbonic anhydrase inhibitors.

Rogato A, Del Prete S, Nocentini A, Carginale V, Supuran CT, Capasso C.

J Enzyme Inhib Med Chem. 2019 Dec;34(1):510-518. doi: 10.1080/14756366.2018.1559840.

17.

Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates.

Küçükbay H, Buğday N, Küçükbay FZ, Berrino E, Bartolucci G, Del Prete S, Capasso C, Supuran CT.

Bioorg Chem. 2019 Mar;83:414-423. doi: 10.1016/j.bioorg.2018.11.003. Epub 2018 Nov 3.

PMID:
30419497
18.

Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides.

Meleddu R, Distinto S, Cottiglia F, Angius R, Gaspari M, Taverna D, Melis C, Angeli A, Bianco G, Deplano S, Fois B, Del Prete S, Capasso C, Alcaro S, Ortuso F, Yanez M, Supuran CT, Maccioni E.

ACS Med Chem Lett. 2018 Sep 17;9(10):1045-1050. doi: 10.1021/acsmedchemlett.8b00352. eCollection 2018 Oct 11.

PMID:
30344915
19.

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases.

Annunziato G, Giovati L, Angeli A, Pavone M, Del Prete S, Pieroni M, Capasso C, Bruno A, Conti S, Magliani W, Supuran CT, Costantino G.

J Enzyme Inhib Med Chem. 2018 Dec;33(1):1537-1544. doi: 10.1080/14756366.2018.1516652.

20.

Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N'-aryl-N-hydroxy-ureas.

Berrino E, Bozdag M, Del Prete S, Alasmary FAS, Alqahtani LS, AlOthman Z, Capasso C, Supuran CT.

J Enzyme Inhib Med Chem. 2018 Dec;33(1):1194-1198. doi: 10.1080/14756366.2018.1490733.

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