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Items: 1 to 20 of 61

1.

Directed C-H Functionalization Reactions with a Picolinamide Directing Group: Ni-Catalyzed Cleavage and By-Product Recycling.

Biswas S, Bheemireddy NR, Bal M, Van Steijvoort BF, Maes BUW.

J Org Chem. 2019 Sep 16. doi: 10.1021/acs.joc.9b02299. [Epub ahead of print]

PMID:
31522497
2.

Base Metal-Catalyzed Isocyanide Insertions.

Collet JW, Roose TR, Ruijter E, Maes BUW, Orru R.

Angew Chem Int Ed Engl. 2019 Jul 9. doi: 10.1002/anie.201905838. [Epub ahead of print]

PMID:
31287627
3.

Synthesis of Functionalized Pyrazin-2(1 H)-ones via Tele-Nucleophilic Substitution of Hydrogen Involving Grignard Reactants and Electrophiles.

Mampuys P, Moseev TD, Varaksin MV, De Houwer J, Vande Velde CML, Chupakhin ON, Charushin VN, Maes BUW.

Org Lett. 2019 Apr 19;21(8):2699-2703. doi: 10.1021/acs.orglett.9b00681. Epub 2019 Apr 9.

PMID:
30964690
4.

Carbamate Synthesis Using a Shelf-Stable and Renewable C1 Reactant.

Dobi Z, Reddy BN, Renders E, Van Raemdonck L, Mensch C, De Smet G, Chen C, Bheeter C, Sergeyev S, Herrebout WA, Maes BUW.

ChemSusChem. 2019 Jul 5;12(13):3103-3114. doi: 10.1002/cssc.201900406. Epub 2019 Jun 11.

PMID:
30921504
5.

Ruthenium-Catalyzed Reductive Arylation of N-(2-Pyridinyl)amides with Isopropanol and Arylboronate Esters.

Ronson TO, Renders E, Van Steijvoort BF, Wang X, Wybon CCD, Prokopcová H, Meerpoel L, Maes BUW.

Angew Chem Int Ed Engl. 2019 Jan 8;58(2):482-487. doi: 10.1002/anie.201810947. Epub 2018 Dec 11.

PMID:
30380163
6.

Corrigendum to "Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings" [Bioorg. Med. Chem. Lett. 28(13) (2018) 2320-2323].

Willemse T, Eiselt E, Hollanders K, Schepens W, van Vlijmen HWT, Chung NN, Blais V, Holleran B, Longpré JM, Schiller PW, Maes BUW, Sarret P, Gendron L, Ballet S.

Bioorg Med Chem Lett. 2018 Nov 1;28(20):3418. doi: 10.1016/j.bmcl.2018.08.023. Epub 2018 Sep 5. No abstract available.

PMID:
30195888
7.

Catalytic Aerobic Oxidation of C(sp3 )-H Bonds.

Sterckx H, Morel B, Maes BUW.

Angew Chem Int Ed Engl. 2019 Jun 11;58(24):7946-7970. doi: 10.1002/anie.201804946. Epub 2019 Apr 8. Review.

PMID:
30052305
8.

A comprehensive overview of directing groups applied in metal-catalysed C-H functionalisation chemistry.

Sambiagio C, Schönbauer D, Blieck R, Dao-Huy T, Pototschnig G, Schaaf P, Wiesinger T, Zia MF, Wencel-Delord J, Besset T, Maes BUW, Schnürch M.

Chem Soc Rev. 2018 Aug 28;47(17):6603-6743. doi: 10.1039/c8cs00201k. Review.

9.

Synthesis of Secondary Amides from Thiocarbamates.

Mampuys P, Ruijter E, Orru RVA, Maes BUW.

Org Lett. 2018 Jul 20;20(14):4235-4239. doi: 10.1021/acs.orglett.8b01654. Epub 2018 Jul 5.

PMID:
29975068
10.

Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings.

Willemse T, Eiselt E, Hollanders K, Schepens W, van Vlijmen HWT, Chung NN, Blais V, Holleran B, Longpré JM, Schiller PW, Maes BUW, Sarret P, Gendron L, Ballet S.

Bioorg Med Chem Lett. 2018 Jul 15;28(13):2320-2323. doi: 10.1016/j.bmcl.2018.05.015. Epub 2018 May 12. Erratum in: Bioorg Med Chem Lett. 2018 Nov 1;28(20):3418.

11.

A bifunctional-biased mu-opioid agonist-neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects.

Drieu la Rochelle A, Guillemyn K, Dumitrascuta M, Martin C, Utard V, Quillet R, Schneider S, Daubeuf F, Willemse T, Mampuys P, Maes BUW, Frossard N, Bihel F, Spetea M, Simonin F, Ballet S.

Pain. 2018 Sep;159(9):1705-1718. doi: 10.1097/j.pain.0000000000001262.

PMID:
29708942
12.

Bromotryptophans and their incorporation in cyclic and bicyclic privileged peptides.

García-Pindado J, Willemse T, Goss R, Maes BUW, Giralt E, Ballet S, Teixidó M.

Biopolymers. 2018 Aug;109(10):e23112. doi: 10.1002/bip.23112. Epub 2018 Mar 12.

13.

Modular Three-Component Synthesis of 4-Aminoquinolines via an Imidoylative Sonogashira/Cyclization Cascade.

Collet JW, Ackermans K, Lambregts J, Maes BUW, Orru RVA, Ruijter E.

J Org Chem. 2018 Jan 19;83(2):854-861. doi: 10.1021/acs.joc.7b02844. Epub 2018 Jan 2.

14.

Electrosynthesis: A New Frontier in Aerobic Oxidation?

Sambiagio C, Sterckx H, Maes BUW.

ACS Cent Sci. 2017 Jul 26;3(7):686-688. doi: 10.1021/acscentsci.7b00275. Epub 2017 Jul 5. No abstract available.

15.

"Dark" Singlet Oxygen and Electron Paramagnetic Resonance Spin Trapping as Convenient Tools to Assess Photolytic Drug Degradation.

Persich P, Hostyn S, Joie C, Winderickx G, Pikkemaat J, Romijn EP, Maes BU.

J Pharm Sci. 2017 May;106(5):1310-1316. doi: 10.1016/j.xphs.2017.01.015. Epub 2017 Jan 18.

PMID:
28108379
16.

Concise Xanthine Synthesis through a Double-Amidination Reaction of a 6-Chlorouracil with Amidines using Base-Metal Catalysis.

Morel B, Franck P, Bidange J, Sergeyev S, Smith DA, Moseley JD, Maes BU.

ChemSusChem. 2017 Feb 8;10(3):624-628. doi: 10.1002/cssc.201601483. Epub 2017 Jan 12.

PMID:
27899009
17.

Amine Activation: Synthesis of N-(Hetero)arylamides from Isothioureas and Carboxylic Acids.

Zhu YP, Sergeyev S, Franck P, Orru RV, Maes BU.

Org Lett. 2016 Sep 16;18(18):4602-5. doi: 10.1021/acs.orglett.6b02247. Epub 2016 Aug 29.

PMID:
27570902
18.

Iodide-Catalyzed Synthesis of Secondary Thiocarbamates from Isocyanides and Thiosulfonates.

Mampuys P, Zhu Y, Sergeyev S, Ruijter E, Orru RV, Van Doorslaer S, Maes BU.

Org Lett. 2016 Jun 17;18(12):2808-11. doi: 10.1021/acs.orglett.6b01023. Epub 2016 Jun 8.

PMID:
27276236
19.

Palladium-Catalyzed Construction of Amidines from Arylboronic Acids under Oxidative Conditions.

Zhu F, Li Y, Wang Z, Orru RV, Maes BU, Wu XF.

Chemistry. 2016 Jun 1;22(23):7743-6. doi: 10.1002/chem.201601262. Epub 2016 Apr 27.

PMID:
27061735
20.

Base metal-catalyzed benzylic oxidation of (aryl)(heteroaryl)methanes with molecular oxygen.

Sterckx H, De Houwer J, Mensch C, Herrebout W, Tehrani KA, Maes BU.

Beilstein J Org Chem. 2016 Jan 27;12:144-53. doi: 10.3762/bjoc.12.16. eCollection 2016.

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