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Items: 1 to 20 of 33

1.

Stapled peptide targeting the CDK4/Cyclin D interface combined with Abemaciclib inhibits KRAS mutant lung cancer growth.

Bouclier C, Simon M, Laconde G, Pellerano M, Diot S, Lantuejoul S, Busser B, Vanwonterghem L, Vollaire J, Josserand V, Legrand B, Coll JL, Amblard M, Hurbin A, Morris MC.

Theranostics. 2020 Jan 12;10(5):2008-2028. doi: 10.7150/thno.40971. eCollection 2020.

2.

Prospect of Thiazole-based γ-Peptide Foldamers in Enamine Catalysis: Exploration of the Nitro-Michael Addition.

Aguesseau-Kondrotas J, Simon M, Legrand B, Bantigniès JL, Kang YK, Dumitrescu D, Van der Lee A, Campagne JM, de Figueiredo RM, Maillard LT.

Chemistry. 2019 May 28;25(30):7396-7401. doi: 10.1002/chem.201901221. Epub 2019 May 7.

PMID:
30946485
3.

The HslV Protease from Leishmania major and Its Activation by C-terminal HslU Peptides.

Kebe NM, Samanta K, Singh P, Lai-Kee-Him J, Apicella V, Payrot N, Lauraire N, Legrand B, Lisowski V, Mbang-Benet DE, Pages M, Bastien P, Kajava AV, Bron P, Hernandez JF, Coux O.

Int J Mol Sci. 2019 Feb 26;20(5). pii: E1021. doi: 10.3390/ijms20051021.

4.

12/10-Helix in Mixed β-Peptides Alternating Bicyclic and Acyclic β-Amino Acids: Probing the Relationship between Bicyclic Side Chain and Helix Stability.

Simon M, Milbeo P, Liu H, André C, Wenger E, Martinez J, Amblard M, Aubert E, Legrand B, Calmès M.

Chemistry. 2018 Dec 12;24(70):18795-18800. doi: 10.1002/chem.201804404. Epub 2018 Nov 15.

PMID:
30277633
5.

Synthesis of [1,2,4]Triazolo[4,3- a]piperazin-6-ones: An Approach to the Triazole-Fused Ketopiperazine Scaffold.

Ben Haj Salah K, Legrand B, Bibian M, Wenger E, Fehrentz JA, Denoyelle S.

Org Lett. 2018 Jun 1;20(11):3250-3254. doi: 10.1021/acs.orglett.8b01112. Epub 2018 May 15.

PMID:
29763330
6.

How are 1,2,3-triazoles accommodated in helical secondary structures?

Ben Haj Salah K, Das S, Ruiz N, Andreu V, Martinez J, Wenger E, Amblard M, Didierjean C, Legrand B, Inguimbert N.

Org Biomol Chem. 2018 May 15;16(19):3576-3583. doi: 10.1039/c8ob00686e.

PMID:
29693098
7.

Selectivity Modulation and Structure of α/aza-β3 Cyclic Antimicrobial Peptides.

Laurencin M, Simon M, Fleury Y, Baudy-Floc'h M, Bondon A, Legrand B.

Chemistry. 2018 Apr 20;24(23):6191-6201. doi: 10.1002/chem.201800152. Epub 2018 Mar 26.

PMID:
29411917
8.

Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds.

Van der Poorten O, Legrand B, Vezenkov LL, García-Pindado J, Bettache N, Knuhtsen A, Pedersen DS, Sánchez-Navarro M, Martinez J, Teixidó M, Garcia M, Tourwé D, Amblard M, Ballet S.

Chembiochem. 2018 Apr 4;19(7):696-705. doi: 10.1002/cbic.201700678. Epub 2018 Feb 28.

PMID:
29377388
9.

C9/12 Ribbon-Like Structures in Hybrid Peptides Alternating α- and Thiazole-Based γ-Amino Acids.

Bonnel C, Legrand B, Simon M, Martinez J, Bantignies JL, Kang YK, Wenger E, Hoh F, Masurier N, Maillard LT.

Chemistry. 2017 Dec 11;23(69):17584-17591. doi: 10.1002/chem.201704001. Epub 2017 Nov 15.

PMID:
28990697
10.

Enhancing the Antimicrobial Activity of Alamethicin F50/5 by Incorporating N-terminal Hydrophobic Triazole Substituents.

Das S, Ben Haj Salah K, Wenger E, Martinez J, Kotarba J, Andreu V, Ruiz N, Savini F, Stella L, Didierjean C, Legrand B, Inguimbert N.

Chemistry. 2017 Dec 19;23(71):17964-17972. doi: 10.1002/chem.201703569. Epub 2017 Nov 23.

PMID:
28922505
11.

Ribbon-like Foldamers for Cellular Uptake and Drug Delivery.

Vezenkov LL, Martin V, Bettache N, Simon M, Messerschmitt A, Legrand B, Bantignies JL, Subra G, Maynadier M, Bellet V, Garcia M, Martinez J, Amblard M.

Chembiochem. 2017 Nov 2;18(21):2110-2114. doi: 10.1002/cbic.201700455. Epub 2017 Sep 22.

PMID:
28863239
12.

A General Approach to the Aza-Diketomorpholine Scaffold.

Berthet M, Legrand B, Martinez J, Parrot I.

Org Lett. 2017 Feb 3;19(3):492-495. doi: 10.1021/acs.orglett.6b03656. Epub 2017 Jan 17.

PMID:
28093918
13.

Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases.

Knuhtsen A, Legrand B, Van der Poorten O, Amblard M, Martinez J, Ballet S, Kristensen JL, Pedersen DS.

Chemistry. 2016 Sep 19;22(39):14022-14028. doi: 10.1002/chem.201602518. Epub 2016 Aug 12.

PMID:
27515561
14.

LEON-BIS: multiple alignment evaluation of sequence neighbours using a Bayesian inference system.

Vanhoutreve R, Kress A, Legrand B, Gass H, Poch O, Thompson JD.

BMC Bioinformatics. 2016 Jul 7;17(1):271. doi: 10.1186/s12859-016-1146-y.

15.

12/14/14-Helix Formation in 2:1 α/β-Hybrid Peptides Containing Bicyclo[2.2.2]octane Ring Constraints.

Legrand B, André C, Moulat L, Didierjean C, Hermet P, Bantignies JL, Martinez J, Amblard M, Calmès M.

Chemistry. 2016 Aug 16;22(34):11986-90. doi: 10.1002/chem.201602746. Epub 2016 Jul 14.

PMID:
27311099
16.

A switchable stapled peptide.

Kalistratova A, Legrand B, Verdié P, Naydenova E, Amblard M, Martinez J, Subra G.

J Pept Sci. 2016 Mar;22(3):143-8. doi: 10.1002/psc.2851. Epub 2016 Jan 19.

PMID:
26785930
17.

Crystal structure of Boc-(S)-ABOC-(S)-Ala-(S)-ABOC-(S)-Phe-OBn chloro-form monosolvate.

Wenger E, Moulat L, Legrand B, Amblard M, Calmès M, Didierjean C.

Acta Crystallogr E Crystallogr Commun. 2015 Sep 17;71(Pt 10):1193-5. doi: 10.1107/S2056989015016941. eCollection 2015 Oct 1.

18.

Turning Peptide Sequences into Ribbon Foldamers by a Straightforward Multicyclization Reaction.

Martin V, Legrand B, Vezenkov LL, Berthet M, Subra G, Calmès M, Bantignies JL, Martinez J, Amblard M.

Angew Chem Int Ed Engl. 2015 Nov 16;54(47):13966-70. doi: 10.1002/anie.201506955. Epub 2015 Sep 23.

PMID:
26398631
19.

Straightforward strategy to substitute amide bonds by 1,2,3-triazoles in peptaibols analogs using Aibψ[Tz]-Xaa dipeptides.

Ben Haj Salah K, Legrand B, Das S, Martinez J, Inguimbert N.

Biopolymers. 2015 Sep;104(5):611-21. doi: 10.1002/bip.22641.

PMID:
25784277
20.

Unprecedented chain-length-dependent conformational conversion between 11/9 and 18/16 helix in α/β-hybrid peptides.

Legrand B, André C, Moulat L, Wenger E, Didierjean C, Aubert E, Averlant-Petit MC, Martinez J, Calmes M, Amblard M.

Angew Chem Int Ed Engl. 2014 Nov 24;53(48):13131-5. doi: 10.1002/anie.201407329. Epub 2014 Sep 26.

PMID:
25258017

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