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Items: 1 to 20 of 47

1.

In vitro and in vivo cytotoxic activity and human serum albumin interaction for a methoxy-styryl-thiosemicarbazone.

Chaves OA, de Castro IS, Goulart CM, Bellieny MSS, Netto-Ferreira JC, Echevarria-Lima J, Echevarria A.

Invest New Drugs. 2019 Jan 19. doi: 10.1007/s10637-018-00722-y. [Epub ahead of print]

PMID:
30661149
2.

Synthesis and biological evaluation of N-aryl-2-phenyl-hydrazinecarbothioamides: Experimental and theoretical analysis on tyrosinase inhibition and interaction with HSA.

Sousa-Pereira D, Chaves OA, Dos Reis CM, de Oliveira MCC, Sant'Anna CMR, Netto-Ferreira JC, Echevarria A.

Bioorg Chem. 2018 Dec;81:79-87. doi: 10.1016/j.bioorg.2018.07.035. Epub 2018 Aug 6.

PMID:
30118988
3.

Novel piperonal 1,3,4-thiadiazolium-2-phenylamines mesoionic derivatives: Synthesis, tyrosinase inhibition evaluation and HSA binding study.

Lopes ND, Chaves OA, de Oliveira MCC, Sant'Anna CMR, Sousa-Pereira D, Netto-Ferreira JC, Echevarria A.

Int J Biol Macromol. 2018 Jun;112:1062-1072. doi: 10.1016/j.ijbiomac.2018.02.050. Epub 2018 Feb 13.

4.

Effects of a new antiprotozoal drug, N,N'-diphenyl-4-methoxy-benzamidine, on energy-linked functions of rat liver mitochondria.

Petiz LL, Pires ADRA, Echevarria A, Rodrigues-Santos CE, Eliane Merlin Rocha M, Acco A, Cadena SMSC.

Chem Biol Interact. 2018 Jan 5;279:34-42. doi: 10.1016/j.cbi.2017.11.006. Epub 2017 Nov 9.

PMID:
29128607
5.

Thiosemicarbazones as inhibitors of tyrosinase enzyme.

Soares MA, Almeida MA, Marins-Goulart C, Chaves OA, Echevarria A, de Oliveira MCC.

Bioorg Med Chem Lett. 2017 Aug 1;27(15):3546-3550. doi: 10.1016/j.bmcl.2017.05.057. Epub 2017 May 18.

PMID:
28583798
6.

Ultrasound-assisted Extraction of Ursolic Acid from the Flowers of Ixora coccinia Linn (Rubiaceae) and Antiproliferative Activity of Ursolic Acid and Synthesized Derivatives.

Alves Monteath SAF, Maciel MAM, Vega RG, de Mello H, de Araújo Martins C, Esteves-Souza A, Gattass CR, Echevarria A.

Pharmacogn Mag. 2017 Apr-Jun;13(50):265-269. doi: 10.4103/0973-1296.204557. Epub 2017 Apr 18.

7.

Impairment of oxidative phosphorylation increases the toxicity of SYD-1 on hepatocarcinoma cells (HepG2).

Brandt AP, Gozzi GJ, Pires Ado R, Martinez GR, Dos Santos Canuto AV, Echevarria A, Di Pietro A, Cadena SM.

Chem Biol Interact. 2016 Aug 25;256:154-60. doi: 10.1016/j.cbi.2016.07.007. Epub 2016 Jul 11.

8.

Sydnone 1: A Mesoionic Compound with Antitumoral and Haematological Effects In Vivo.

Galuppo LF, Dos Reis Lívero FA, Martins GG, Cardoso CC, Beltrame OC, Klassen LM, Canuto AV, Echevarria A, Telles JE, Klassen G, Acco A.

Basic Clin Pharmacol Toxicol. 2016 Jul;119(1):41-50. doi: 10.1111/bcpt.12545. Epub 2016 Jan 25.

9.

Antioxidant effect of 1,3,4-thiadiazolium mesoionic derivatives on isolated mitochondria.

Andrade Pires Ado R, Jabor Gozzi G, Rodrigues Noleto G, Echevarria A, Moretto Reis C, Merlin Rocha ME, Regina Martinez G, Correia Cadena SM.

Eur J Pharmacol. 2016 Jan 5;770:78-84. doi: 10.1016/j.ejphar.2015.12.004. Epub 2015 Dec 5.

PMID:
26667999
10.

Evaluation of Antiplasmodial activity of extracts and constituents from Ampelozizyphus amazonicus.

do Carmo DF, Amaral AC, Machado M, Lopes D, Echevarria A, Rosário VE, Silva JR.

Pharmacogn Mag. 2015 Oct;11(Suppl 2):S244-50. doi: 10.4103/0973-1296.166071.

11.

Antileishmanial activity and trypanothione reductase effects of terpenes from the Amazonian species Croton cajucara Benth (Euphorbiaceae).

Lima GS, Castro-Pinto DB, Machado GC, Maciel MA, Echevarria A.

Phytomedicine. 2015 Nov 15;22(12):1133-7. doi: 10.1016/j.phymed.2015.08.012. Epub 2015 Sep 18.

PMID:
26547537
12.

Quantitative Structure-Property Relationship (QSPR) Models for a Local Quantum Descriptor: Investigation of the 4- and 3-Substituted-Cinnamic Acid Esterification.

Rodrigues-Santos CE, Echevarria A, Sant'Anna CM, Bitencourt TB, Nascimento MG, Bauerfeldt GF.

Molecules. 2015 Sep 22;20(9):17493-510. doi: 10.3390/molecules200917493.

13.

Novel 3,4-methylenedioxyde-6-X-benzaldehyde-thiosemicarbazones: Synthesis and antileishmanial effects against Leishmania amazonensis.

de Melos JL, Torres-Santos EC, Faiões Vdos S, Del Cistia Cde N, Sant'Anna CM, Rodrigues-Santos CE, Echevarria A.

Eur J Med Chem. 2015 Oct 20;103:409-17. doi: 10.1016/j.ejmech.2015.09.009. Epub 2015 Sep 8.

PMID:
26375353
14.

Selective Cytotoxicity of 1,3,4-Thiadiazolium Mesoionic Derivatives on Hepatocarcinoma Cells (HepG2).

Gozzi GJ, Pires Ado R, Valdameri G, Rocha ME, Martinez GR, Noleto GR, Acco A, Alves de Souza CE, Echevarria A, Moretto Dos Reis C, Di Pietro A, Suter Correia Cadena SM.

PLoS One. 2015 Jun 17;10(6):e0130046. doi: 10.1371/journal.pone.0130046. eCollection 2015.

15.

Mesoionic compounds with antifungal activity against Fusarium verticillioides.

Paiva Rde O, Kneipp LF, dos Reis CM, Echevarria A.

BMC Microbiol. 2015 Feb 4;15:11. doi: 10.1186/s12866-015-0340-9.

16.

Sydnone SYD-1 affects the metabolic functions of isolated rat hepatocytes.

Brandt AP, Pires Ado R, Rocha ME, Noleto GR, Acco A, de Souza CE, Echevarria A, Canuto AV, Cadena SM.

Chem Biol Interact. 2014 Jul 25;218:107-14. doi: 10.1016/j.cbi.2014.05.002. Epub 2014 May 15.

17.

1H NMR for quantifying sulfide trapping efficiency by using 1,3,5-tris(2-hydroxyethyl)-1,3,5-triazinane.

Canuto AV, Echevarria A.

Magn Reson Chem. 2014 Jul;52(7):353-7. doi: 10.1002/mrc.4072. Epub 2014 Apr 11.

PMID:
24723368
18.

The antioxidant effect of the mesoionic compound SYD-1 in mitochondria.

Gozzi GJ, Pires Ado R, Martinez GR, Rocha ME, Noleto GR, Echevarria A, Canuto AV, Cadena SM.

Chem Biol Interact. 2013 Oct 5;205(3):181-7. doi: 10.1016/j.cbi.2013.07.004. Epub 2013 Jul 16.

19.

Synthesis, antileishmanial activity and structure-activity relationship of 1-N-X-phenyl-3-N'-Y-phenyl-benzamidines.

Rodrigues-Santos CE, Leon LL, Bortoluzzi AJ, Canto-Cavalheiro MM, Machado GC, Echevarria A.

Eur J Med Chem. 2013 Sep;67:166-74. doi: 10.1016/j.ejmech.2013.06.040. Epub 2013 Jun 27.

PMID:
23851118
20.

In vitro evaluation of 4-phenyl-5-(4'-X-phenyl)-1,3,4-thiadiazolium-2-phenylaminide chlorides and 3[N-4'-X-phenyl]-1,2,3-oxadiazolium-5-olate derivatives on nitric oxide synthase and arginase activities of Leishmania amazonensis.

Soares-Bezerra RJ, Leon LL, Echevarria A, Reis CM, Gomes-Silva L, Agostinho CG, Fernandes RA, Canto-Cavalheiro MM, Genestra MS.

Exp Parasitol. 2013 Sep;135(1):50-4. doi: 10.1016/j.exppara.2013.05.008. Epub 2013 May 18.

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