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Items: 1 to 20 of 21

1.

Synthesis and Fluorescent Properties of Novel Isoquinoline Derivatives.

Balewski Ł, Sączewski F, Gdaniec M, Kornicka A, Cicha K, Jalińska A.

Molecules. 2019 Nov 10;24(22). pii: E4070. doi: 10.3390/molecules24224070.

2.

Synthesis, Structure, Chemical Stability, and In Vitro Cytotoxic Properties of Novel Quinoline-3-Carbaldehyde Hydrazones Bearing a 1,2,4-Triazole or Benzotriazole Moiety.

Korcz M, Sączewski F, Bednarski PJ, Kornicka A.

Molecules. 2018 Jun 20;23(6). pii: E1497. doi: 10.3390/molecules23061497.

3.

COMPARISON OF THE EFFECTS OF MARSANIDINE DERIVATIVES ON RAT CARDIOVASCULAR SYSTEM.

Boblewski K, Lehmann A, Marchwinska A, Kornicka A, Wasilewska A, Saczewski F, Rybczynska A.

Acta Pol Pharm. 2017 Mar;74(2):579-586.

4.

Are Alpha-2D Adrenoceptor Subtypes Involved in Rat Mydriasis Evoked by New Imidazoline Derivatives: Marsanidine and 7-Methylmarsanidine?

Raczak-Gutknecht J, Frąckowiak T, Nasal A, Kornicka A, Sączewski F, Kaliszan R.

Dose Response. 2017 Apr 18;15(2):1559325817701213. doi: 10.1177/1559325817701213. eCollection 2017 Apr-Jun.

5.

Comparative pharmacodynamic analysis of imidazoline compounds using rat model of ocular mydriasis with a test of quantitative structure-activity relationships.

Raczak-Gutknecht J, Nasal A, Frąckowiak T, Kornicka A, Sączewski F, Wawrzyniak R, Kubik Ł, Kaliszan R.

J Pharm Biomed Anal. 2017 Sep 10;144:122-128. doi: 10.1016/j.jpba.2017.03.053. Epub 2017 Apr 6.

PMID:
28420580
6.

Synthesis and Preliminary Cytotoxicity Studies of 1-[1-(4,5-Dihydrooxazol- 2-yl)-1H-indazol-3-yl]-3-phenylurea and 3-phenylthiourea Derivatives.

Kornicka A, Saczewski F, Bednarski PJ, Korcz M, Szumlas P, Romejko E, Sakowicz A, Sitek L, Wojciechowska M.

Med Chem. 2017;13(7):616-624. doi: 10.2174/1573406413666170306114401.

PMID:
28266278
7.

1-[(Imidazolidin-2-yl)imino]-1H-indoles as new hypotensive agents: synthesis and in vitro and in vivo biological studies.

Kornicka A, Wasilewska A, Sączewski J, Hudson AL, Boblewski K, Lehmann A, Gzella K, Belka M, Sączewski F, Gdaniec M, Rybczyńska A, Bączek T.

Chem Biol Drug Des. 2017 Mar;89(3):400-410. doi: 10.1111/cbdd.12846. Epub 2016 Sep 26.

PMID:
27566285
8.

Imidazoline scaffold in medicinal chemistry: a patent review (2012-2015).

Sączewski F, Kornicka A, Balewski Ł.

Expert Opin Ther Pat. 2016 Sep;26(9):1031-48. doi: 10.1080/13543776.2016.1210128. Epub 2016 Jul 20. Review. Erratum in: Expert Opin Ther Pat. 2017 Feb;27(2):227.

PMID:
27382975
9.

Circulatory effect of TCS-80, a new imidazoline compound, in rats.

Boblewski K, Lehmann A, Sączewski F, Sączewski J, Kornicka A, Marchwińska A, Rybczyńska A.

Pharmacol Rep. 2016 Aug;68(4):715-9. doi: 10.1016/j.pharep.2016.03.008. Epub 2016 Mar 23.

PMID:
27127910
10.

Vagotomy reveals the importance of the imidazoline receptors in the cardiovascular effects of marsanidine and 7-ME-marsanidine in rats.

Boblewski K, Lehmann A, Sączewski F, Kornicka A, Rybczyńska A.

Pharmacol Rep. 2014 Oct;66(5):874-9. doi: 10.1016/j.pharep.2014.05.009. Epub 2014 Jun 6.

PMID:
25149994
11.

Marsanidine and 7-Me-marsanidine, the new hypotensive imidazolines augment sodium and urine excretion in rats.

Wróblewska M, Kasprzyk J, Sączewski F, Kornicka A, Boblewski K, Lehmann A, Rybczyńska A.

Pharmacol Rep. 2013;65(4):1025-32.

12.

Synthesis, cytotoxicity testing, and structure-activity relationships of novel 6-chloro-7-(4-phenylimino-4H-3,1-benzoxazin-2-yl)-3-(substituted)-1,4,2-benzodithiazine 1,1-dioxides.

Pomarnacka E, Kornicka A, Kuchnio A, Heinrichs M, Grünert R, Gdaniec M, Bednarski PJ.

Arch Pharm (Weinheim). 2011 Jul;344(7):431-41. doi: 10.1002/ardp.201000183. Epub 2011 May 25.

PMID:
21618270
13.

3-[(Imidazolidin-2-yl)imino]indazole ligands with selectivity for the α(2)-adrenoceptor compared to the imidazoline I(1) receptor.

Sączewski F, Kornicka A, Hudson AL, Laird S, Scheinin M, Laurila JM, Rybczyńska A, Boblewski K, Lehmann A, Gdaniec M.

Bioorg Med Chem. 2011 Jan 1;19(1):321-9. doi: 10.1016/j.bmc.2010.11.020. Epub 2010 Nov 11.

PMID:
21129985
14.

Synthesis and biological activity of some 2-imidazolinylhydrazone derivatives.

Kornicka A, Hudson AL, Bednarski PJ.

Acta Pol Pharm. 2009 Sep-Oct;66(5):523-34.

15.

1-[(Imidazolidin-2-yl)imino]indazole. Highly alpha 2/I1 selective agonist: synthesis, X-ray structure, and biological activity.

Saczewski F, Kornicka A, Rybczyńska A, Hudson AL, Miao SS, Gdaniec M, Boblewski K, Lehmann A.

J Med Chem. 2008 Jun 26;51(12):3599-608. doi: 10.1021/jm800112s. Epub 2008 Jun 3.

PMID:
18517187
16.

Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.

Saczewski F, Innocenti A, Sławiński J, Kornicka A, Brzozowski Z, Pomarnacka E, Scozzafava A, Temperini C, Supuran CT.

Bioorg Med Chem. 2008 Apr 1;16(7):3933-40. doi: 10.1016/j.bmc.2008.01.034. Epub 2008 Jan 26.

PMID:
18242998
17.
18.

Carbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides.

Saczewski F, Innocenti A, Brzozowski Z, Slawiński J, Pomarnacka E, Kornicka A, Scozzafava A, Supuran CT.

J Enzyme Inhib Med Chem. 2006 Oct;21(5):563-8.

PMID:
17194028
19.

Carbonic anhydrase inhibitors. Inhibition of the cytosolic human isozymes I and II, and the transmembrane, tumor-associated isozymes IX and XII with substituted aromatic sulfonamides activatable in hypoxic tumors.

Saczewski F, Sławiński J, Kornicka A, Brzozowski Z, Pomarnacka E, Innocenti A, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett. 2006 Sep 15;16(18):4846-51. Epub 2006 Jun 30.

PMID:
16809036
20.

2-(4,5-Dihydroimidazol-2-yl)benzimidazoles as highly selective imidazoline I2/adrenergic alpha2 receptor ligands.

Saczewski F, Tabin P, Tyacke RJ, Maconie A, Saczewski J, Kornicka A, Nutt DJ, Hudson AL.

Bioorg Med Chem. 2006 Oct 1;14(19):6679-85. Epub 2006 Jun 16.

PMID:
16782348

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