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Items: 11

1.

A π-Halogen Bond of Dibenzofuranones with the Gatekeeper Phe113 in Human Protein Kinase CK2 Leads to Potent Tight Binding Inhibitors.

Schnitzler A, Gratz A, Bollacke A, Weyrich M, Kuckländer U, Wünsch B, Götz C, Niefind K, Jose J.

Pharmaceuticals (Basel). 2018 Feb 17;11(1). pii: E23. doi: 10.3390/ph11010023.

2.

Identification of a Potent Allosteric Inhibitor of Human Protein Kinase CK2 by Bacterial Surface Display Library Screening.

Nienberg C, Garmann C, Gratz A, Bollacke A, Götz C, Jose J.

Pharmaceuticals (Basel). 2017 Jan 5;10(1). pii: E6. doi: 10.3390/ph10010006.

3.

Functional display of heterotetrameric human protein kinase CK2 on Escherichia coli: a novel tool for drug discovery.

Gratz A, Bollacke A, Stephan S, Nienberg C, Le Borgne M, Götz C, Jose J.

Microb Cell Fact. 2015 Jun 3;14:74. doi: 10.1186/s12934-015-0263-z.

4.

Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds.

Bouaziz Z, Issa S, Gentili J, Gratz A, Bollacke A, Kassack M, Jose J, Herfindal L, Gausdal G, Døskeland SO, Mullié C, Sonnet P, Desgrouas C, Taudon N, Valdameri G, Di Pietro A, Baitiche M, Le Borgne M.

J Enzyme Inhib Med Chem. 2015 Apr;30(2):180-8. doi: 10.3109/14756366.2014.899594. Epub 2014 Apr 3.

PMID:
24697298
5.
6.

TF--a novel cell-permeable and selective inhibitor of human protein kinase CK2 induces apoptosis in the prostate cancer cell line LNCaP.

Götz C, Gratz A, Kucklaender U, Jose J.

Biochim Biophys Acta. 2012 Jul;1820(7):970-7. doi: 10.1016/j.bbagen.2012.02.009. Epub 2012 Feb 24.

PMID:
22387500
7.

Identification of novel CK2 inhibitors with a benzofuran scaffold by novel non-radiometric in vitro assays.

Gratz A, Kuckländer U, Bollig R, Götz C, Jose J.

Mol Cell Biochem. 2011 Oct;356(1-2):83-90. doi: 10.1007/s11010-011-0957-4. Epub 2011 Jul 13.

PMID:
21750981
8.

Focusing mutations within random libraries to distinct areas: protein domain library generation by overlap extension.

Gratz A, Jose J.

Methods Mol Biol. 2011;729:153-66. doi: 10.1007/978-1-61779-065-2_10.

PMID:
21365489
9.

A CE-based assay for human protein kinase CK2 activity measurement and inhibitor screening.

Gratz A, Götz C, Jose J.

Electrophoresis. 2010 Jan;31(4):634-40. doi: 10.1002/elps.200900514.

PMID:
20162588
10.

A FRET-based microplate assay for human protein kinase CK2, a target in neoplastic disease.

Gratz A, Götz C, Jose J.

J Enzyme Inhib Med Chem. 2010 Apr;25(2):234-9. doi: 10.3109/14756360903170038.

PMID:
19874207
11.

Protein domain library generation by overlap extension (PDLGO): a tool for enzyme engineering.

Gratz A, Jose J.

Anal Biochem. 2008 Jul 15;378(2):171-6. doi: 10.1016/j.ab.2008.03.051. Epub 2008 Apr 7.

PMID:
18452697

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