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Best matches for A. Dömling:

MCR synthesis of a tetracyclic tetrazole scaffold. Patil P et al. Bioorg Med Chem. (2015)

Various cyclization scaffolds by a truly Ugi 4-CR. Sinha MK et al. Org Biomol Chem. (2013)

A universal isocyanide for diverse heterocycle syntheses. Patil P et al. Org Lett. (2014)

Search results

Items: 1 to 20 of 143

1.

A patent review on PD-1/PD-L1 antagonists: small molecules, peptides, and macrocycles (2015-2018).

Shaabani S, Huizinga HPS, Butera R, Kouchi A, Guzik K, Magiera-Mularz K, Holak TA, Dömling A.

Expert Opin Ther Pat. 2018 Sep 10:1-14. doi: 10.1080/13543776.2018.1512706. [Epub ahead of print]

PMID:
30107136
2.

Multicomponent Reaction Based Synthesis of 1-Tetrazolylimidazo[1,5- a]pyridines.

Kurhade S, Diekstra E, Sutanto F, Kurpiewska K, Kalinowska-Tłuścik J, Dömling A.

Org Lett. 2018 Jul 6;20(13):3871-3874. doi: 10.1021/acs.orglett.8b01452. Epub 2018 Jun 26.

3.

Triglyceride profiling in adipose tissues from obese insulin sensitive, insulin resistant and type 2 diabetes mellitus individuals.

Al-Sulaiti H, Diboun I, Banu S, Al-Emadi M, Amani P, Harvey TM, Dömling AS, Latiff A, Elrayess MA.

J Transl Med. 2018 Jun 26;16(1):175. doi: 10.1186/s12967-018-1548-x.

4.

Artificial Macrocycles as IL-17A/IL-17RA Antagonists.

Wang W, Groves MR, Dömling A.

Medchemcomm. 2018 Jan 1;9(1):22-26. doi: 10.1039/C7MD00464H. Epub 2017 Oct 25.

PMID:
29750108
5.

Isolation and molecular characterization of novel glucarpidases: Enzymes to improve the antibody directed enzyme pro-drug therapy for cancer treatment.

Rashidi FB, AlQhatani AD, Bashraheel SS, Shaabani S, Groves MR, Dömling A, Goda SK.

PLoS One. 2018 Apr 26;13(4):e0196254. doi: 10.1371/journal.pone.0196254. eCollection 2018.

6.

Guide for Selection of Relevant Cell Lines During the Evaluation of New Anti-Cancer Compounds.

Ruiz-Moreno AJ, Torres-Barrera P, Velazquez-Paniagua M, Domling A, Velasco-Velazquez MA.

Anticancer Agents Med Chem. 2018 Feb 20. doi: 10.2174/1871520618666180220120544. [Epub ahead of print]

PMID:
29697026
7.

Identification of a non-competitive inhibitor of Plasmodium falciparum aspartate transcarbamoylase.

Lunev S, Bosch SS, Batista FA, Wang C, Li J, Linzke M, Kruithof P, Chamoun G, Dömling ASS, Wrenger C, Groves MR.

Biochem Biophys Res Commun. 2018 Mar 11;497(3):835-842. doi: 10.1016/j.bbrc.2018.02.112. Epub 2018 Feb 21.

PMID:
29476738
8.

Synthesis of Highly Substituted Imidazole Uracil Containing Molecules via Ugi-4CR and Passerini-3CR.

Madhavachary R, Zarganes-Tzitzikas T, Patil P, Kurpiewska K, Kalinowska-Tłuścik J, Dömling A.

ACS Comb Sci. 2018 Apr 9;20(4):192-196. doi: 10.1021/acscombsci.7b00145. Epub 2018 Feb 26.

9.

Diastereoselective One Pot Five-Component Reaction toward 4-(Tetrazole)-1,3-Oxazinanes.

Chandgude AL, Narducci D, Kurpiewska K, Kalinowska-Tłuścik J, Dömling A.

RSC Adv. 2017;7(79):49995-49998. doi: 10.1039/C7RA07392E. Epub 2017 Oct 26.

PMID:
29430295
10.

Discovery of chromenes as inhibitors of macrophage migration inhibitory factor.

Kok T, Wapenaar H, Wang K, Neochoritis CG, Zarganes-Tzitzikas T, Proietti G, Eleftheriadis N, Kurpiewska K, Kalinowska-Tłuścik J, Cool RH, Poelarends GJ, Dömling A, Dekker FJ.

Bioorg Med Chem. 2018 Mar 1;26(5):999-1005. doi: 10.1016/j.bmc.2017.12.032. Epub 2017 Dec 24.

PMID:
29428527
11.

Two-Step Macrocycle Synthesis by Classical Ugi Reaction.

Abdelraheem EMM, Khaksar S, Kurpiewska K, Kalinowska-Tłuścik J, Shaabani S, Dömling A.

J Org Chem. 2018 Feb 2;83(3):1441-1447. doi: 10.1021/acs.joc.7b02984. Epub 2018 Jan 24.

12.

Library-to-Library Synthesis of Highly Substituted α-Aminomethyl Tetrazoles via Ugi Reaction.

Patil P, Mishra B, Sheombarsing G, Kurpiewska K, Kalinowska-Tłuścik J, Dömling A.

ACS Comb Sci. 2018 Feb 12;20(2):70-74. doi: 10.1021/acscombsci.7b00137. Epub 2018 Jan 4. Review.

13.

Immune Checkpoint PD-1/PD-L1: Is There Life Beyond Antibodies?

Konstantinidou M, Zarganes-Tzitzikas T, Magiera-Mularz K, Holak TA, Dömling A.

Angew Chem Int Ed Engl. 2018 Apr 23;57(18):4840-4848. doi: 10.1002/anie.201710407. Epub 2018 Feb 23. Review.

PMID:
29178534
14.

Ugi Multicomponent Reaction Based Synthesis of Medium-Sized Rings.

Abdelraheem EMM, Madhavachary R, Rossetti A, Kurpiewska K, Kalinowska-Tłuścik J, Shaabani S, Dömling A.

Org Lett. 2017 Nov 17;19(22):6176-6179. doi: 10.1021/acs.orglett.7b03094. Epub 2017 Oct 30.

15.

Small-molecule inhibitors of PD-1/PD-L1 immune checkpoint alleviate the PD-L1-induced exhaustion of T-cells.

Skalniak L, Zak KM, Guzik K, Magiera K, Musielak B, Pachota M, Szelazek B, Kocik J, Grudnik P, Tomala M, Krzanik S, Pyrc K, Dömling A, Dubin G, Holak TA.

Oncotarget. 2017 Aug 7;8(42):72167-72181. doi: 10.18632/oncotarget.20050. eCollection 2017 Sep 22.

16.

Artificial Macrocycles as Potent p53-MDM2 Inhibitors.

Estrada-Ortiz N, Neochoritis CG, Twarda-Clapa A, Musielak B, Holak TA, Dömling A.

ACS Med Chem Lett. 2017 Sep 20;8(10):1025-1030. doi: 10.1021/acsmedchemlett.7b00219. eCollection 2017 Oct 12.

17.

Scaffold hopping via ANCHOR.QUERY: β-lactams as potent p53-MDM2 antagonists.

Shaabani S, Neochoritis CG, Twarda-Clapa A, Musielak B, Holak TA, Dömling A.

Medchemcomm. 2017 May 1;8(5):1046-1052. doi: 10.1039/C7MD00058H. Epub 2017 Mar 15.

18.

Abnormal Tin-Boron Exchange in the Attempted Synthesis of a Borylated Borole.

Braunschweig H, Dömling M, Kachel S, Kelch H, Kramer T, Krummenacher I, Lenczyk C, Lin S, Lin Z, Possiel C, Radacki K.

Chemistry. 2017 Nov 16;23(64):16167-16170. doi: 10.1002/chem.201703810. Epub 2017 Oct 25.

PMID:
28960516
19.

AnchorQuery: Rapid online virtual screening for small-molecule protein-protein interaction inhibitors.

Koes DR, Dömling A, Camacho CJ.

Protein Sci. 2018 Jan;27(1):229-232. doi: 10.1002/pro.3303. Epub 2017 Oct 24.

PMID:
28921842
20.

Concise Synthesis of Tetrazole Macrocycle.

Abdelraheem EMM, de Haan MP, Patil P, Kurpiewska K, Kalinowska-Tłuścik J, Shaabani S, Dömling A.

Org Lett. 2017 Oct 6;19(19):5078-5081. doi: 10.1021/acs.orglett.7b02319. Epub 2017 Sep 13.

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