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Best matches for Šárka Štěpánková:

Cholinesterase-based biosensors. Štěpánková Š et al. J Enzyme Inhib Med Chem. (2016)

Proline-Based Carbamates as Cholinesterase Inhibitors. Pizova H et al. Molecules. (2017)

Salicylanilide diethyl phosphates as cholinesterases inhibitors. Krátký M et al. Bioorg Chem. (2015)

Search results

Items: 1 to 20 of 27

1.

2-Hydroxy-N-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase.

Krátký M, Štěpánková Š, Houngbedji NH, Vosátka R, Vorčáková K, Vinšová J.

Biomolecules. 2019 Nov 5;9(11). pii: E698. doi: 10.3390/biom9110698.

2.

In Vitro and In Silico Acetylcholinesterase Inhibitory Activity of Thalictricavine and Canadine and Their Predicted Penetration across the Blood-Brain Barrier.

Chlebek J, Korábečný J, Doležal R, Štěpánková Š, Pérez DI, Hošťálková A, Opletal L, Cahlíková L, Macáková K, Kučera T, Hrabinová M, Jun D.

Molecules. 2019 Apr 5;24(7). pii: E1340. doi: 10.3390/molecules24071340.

3.

Novel Benzene-Based Carbamates for AChE/BChE Inhibition: Synthesis and Ligand/Structure-Oriented SAR Study.

Bak A, Kozik V, Kozakiewicz D, Gajcy K, Strub DJ, Swietlicka A, Stepankova S, Imramovsky A, Polanski J, Smolinski A, Jampilek J.

Int J Mol Sci. 2019 Mar 27;20(7). pii: E1524. doi: 10.3390/ijms20071524.

4.

Investigation of salicylanilide and 4-chlorophenol-based N-monosubstituted carbamates as potential inhibitors of acetyl- and butyrylcholinesterase.

Krátký M, Štěpánková Š, Vorčáková K, Vinšová J.

Bioorg Chem. 2018 Oct;80:668-673. doi: 10.1016/j.bioorg.2018.07.017. Epub 2018 Jul 17.

PMID:
30059892
5.

Synthesis and characterization of new inhibitors of cholinesterases based on N-phenylcarbamates: In vitro study of inhibitory effect, type of inhibition, lipophilicity and molecular docking.

Vorčáková K, Májeková M, Horáková E, Drabina P, Sedlák M, Štěpánková Š.

Bioorg Chem. 2018 Aug;78:280-289. doi: 10.1016/j.bioorg.2018.03.012. Epub 2018 Mar 28.

PMID:
29621640
6.

Proline-Based Carbamates as Cholinesterase Inhibitors.

Pizova H, Havelkova M, Stepankova S, Bak A, Kauerova T, Kozik V, Oravec M, Imramovsky A, Kollar P, Bobal P, Jampilek J.

Molecules. 2017 Nov 14;22(11). pii: E1969. doi: 10.3390/molecules22111969.

7.

Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity.

Krátký M, Štěpánková Š, Vorčáková K, Navrátilová L, Trejtnar F, Stolaříková J, Vinšová J.

Bioorg Chem. 2017 Apr;71:244-256. doi: 10.1016/j.bioorg.2017.02.010. Epub 2017 Feb 21.

PMID:
28245905
8.

Synthesis, characterization and in vitro evaluation of substituted N-(2-phenylcyclopropyl)carbamates as acetyl- and butyrylcholinesterase inhibitors.

Horáková E, Drabina P, Brož B, Štěpánková Š, Vorčáková K, Královec K, Havelek R, Sedlák M.

J Enzyme Inhib Med Chem. 2016;31(sup3):173-179. Epub 2016 Aug 1.

PMID:
27476673
9.

Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors.

Krátký M, Štěpánková Š, Vorčáková K, Vinšová J.

Bioorg Chem. 2016 Oct;68:23-9. doi: 10.1016/j.bioorg.2016.07.004. Epub 2016 Jul 6.

PMID:
27428597
10.

Cholinesterase-based biosensors.

Štěpánková Š, Vorčáková K.

J Enzyme Inhib Med Chem. 2016;31(sup3):180-193. Epub 2016 Jul 12. Review.

PMID:
27405024
11.

Synthesis, structural characterization, docking, lipophilicity and cytotoxicity of 1-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-3-alkyl carbamates, novel acetylcholinesterase and butyrylcholinesterase pseudo-irreversible inhibitors.

Pejchal V, Štěpánková Š, Pejchalová M, Královec K, Havelek R, Růžičková Z, Ajani H, Lo R, Lepšík M.

Bioorg Med Chem. 2016 Apr 1;24(7):1560-72. doi: 10.1016/j.bmc.2016.02.033. Epub 2016 Feb 26.

PMID:
26947959
12.

Novel Cholinesterase Inhibitors Based on O-Aromatic N,N-Disubstituted Carbamates and Thiocarbamates.

Krátký M, Štěpánková Š, Vorčáková K, Švarcová M, Vinšová J.

Molecules. 2016 Feb 11;21(2). pii: E191. doi: 10.3390/molecules21020191.

13.

In Vitro Inhibitory Effects of 8-O-Demethylmaritidine and Undulatine on Acetylcholinesterase and Their Predicted Penetration across the Blood-Brain Barrier.

Cahlíková L, Pérez DI, Štěpánková Š, Chlebek J, Šafratová M, Hošt'álková A, Opletal L.

J Nat Prod. 2015 Jun 26;78(6):1189-92. doi: 10.1021/acs.jnatprod.5b00191. Epub 2015 Jun 1.

PMID:
26030662
14.

Salicylanilide diethyl phosphates as cholinesterases inhibitors.

Krátký M, Štěpánková Š, Vorčáková K, Vinšová J.

Bioorg Chem. 2015 Feb;58:48-52. doi: 10.1016/j.bioorg.2014.11.005. Epub 2014 Nov 13.

PMID:
25462625
15.

Chemical composition of bioactive alkaloid extracts from some Narcissus species and varieties and their biological activity.

Havlasová J, Safratová M, Siatka T, Stĕpánková S, Novák Z, Locárek M, Opletal L, Hrabinová M, Jun D, Benesová N, Kunes J, Cahlíková L.

Nat Prod Commun. 2014 Aug;9(8):1151-5.

PMID:
25233595
16.

Diethyl 2-(phenylcarbamoyl)phenyl phosphorothioates: synthesis, antimycobacterial activity and cholinesterase inhibition.

Vinšová J, Krátký M, Komlóová M, Dadapeer E, Stěpánková S, Vorčáková K, Stolaříková J.

Molecules. 2014 May 30;19(6):7152-68. doi: 10.3390/molecules19067152.

17.

New method for the determination of the half inhibition concentration (IC50) of cholinesterase inhibitors.

Kovárová M, Komers K, Stepánková S, Parík P, Cegan A.

Z Naturforsch C J Biosci. 2013 Mar-Apr;68(3-4):133-8.

PMID:
23819309
18.

Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors.

Imramovský A, Pejchal V, Štěpánková Š, Vorčáková K, Jampílek J, Vančo J, Šimůnek P, Královec K, Brůčková L, Mandíková J, Trejtnar F.

Bioorg Med Chem. 2013 Apr 1;21(7):1735-48. doi: 10.1016/j.bmc.2013.01.052. Epub 2013 Feb 1.

PMID:
23462716
19.

Acetylcholinesterase-inhibiting activity of salicylanilide N-alkylcarbamates and their molecular docking.

Imramovsky A, Stepankova S, Vanco J, Pauk K, Monreal-Ferriz J, Vinsova J, Jampilek J.

Molecules. 2012 Aug 24;17(9):10142-58. doi: 10.3390/molecules170910142.

20.

1,3-substituted imidazolidine-2,4,5-triones: synthesis and inhibition of cholinergic enzymes.

Pejchal V, Stepankova S, Padelkova Z, Imramovsky A, Jampilek J.

Molecules. 2011 Sep 5;16(9):7565-82. doi: 10.3390/molecules16097565.

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