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Items: 1 to 20 of 85

1.

Induction of cell killing and autophagy by amphiphilic pyrrolidine derivatives on human pancreatic cancer cells.

Bello C, Bai J, Zambron BK, Elías-Rodríguez P, Gajate C, Robina I, Caffa I, Cea M, Montecucco F, Nencioni A, Nahimana A, Aubry D, Breton C, Duchosal MA, Mollinedo F, Vogel P.

Eur J Med Chem. 2018 Apr 25;150:457-478. doi: 10.1016/j.ejmech.2018.02.086. Epub 2018 Mar 2.

PMID:
29547833
2.

1,2,3-Triazoles as inhibitors of indoleamine 2,3-dioxygenase 2 (IDO2).

Röhrig UF, Majjigapu SR, Caldelari D, Dilek N, Reichenbach P, Ascencao K, Irving M, Coukos G, Vogel P, Zoete V, Michielin O.

Bioorg Med Chem Lett. 2016 Sep 1;26(17):4330-3. doi: 10.1016/j.bmcl.2016.07.031. Epub 2016 Jul 16.

PMID:
27469130
3.

Synthesis and Applications of Silyl 2-Methylprop-2-ene-1-sulfinates in Preparative Silylation and GC-Derivatization Reactions of Polyols and Carbohydrates.

Marković D, Tchawou WA, Novosjolova I, Laclef S, Stepanovs D, Turks M, Vogel P.

Chemistry. 2016 Mar 14;22(12):4196-205. doi: 10.1002/chem.201504380. Epub 2016 Feb 11.

PMID:
26864218
4.

Challenges in the Discovery of Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors.

Röhrig UF, Majjigapu SR, Vogel P, Zoete V, Michielin O.

J Med Chem. 2015 Dec 24;58(24):9421-37. doi: 10.1021/acs.jmedchem.5b00326. Epub 2015 May 26. Review.

PMID:
25970480
5.

Detailed analysis and follow-up studies of a high-throughput screening for indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors.

Röhrig UF, Majjigapu SR, Chambon M, Bron S, Pilotte L, Colau D, Van den Eynde BJ, Turcatti G, Vogel P, Zoete V, Michielin O.

Eur J Med Chem. 2014 Sep 12;84:284-301. doi: 10.1016/j.ejmech.2014.06.078. Epub 2014 Jul 10.

PMID:
25036789
6.

A critical role of autophagy in antileukemia/lymphoma effects of APO866, an inhibitor of NAD biosynthesis.

Ginet V, Puyal J, Rummel C, Aubry D, Breton C, Cloux AJ, Majjigapu SR, Sordat B, Vogel P, Bruzzone S, Nencioni A, Duchosal MA, Nahimana A.

Autophagy. 2014 Apr;10(4):603-17. doi: 10.4161/auto.27722. Epub 2014 Jan 17.

7.

Amides in one pot from carboxylic acids and amines via sulfinylamides.

Bai J, Zambroń BK, Vogel P.

Org Lett. 2014 Jan 17;16(2):604-7. doi: 10.1021/ol403508j. Epub 2014 Jan 3.

PMID:
24387286
8.

The anti-lymphoma activity of APO866, an inhibitor of nicotinamide adenine dinucleotide biosynthesis, is potentialized when used in combination with anti-CD20 antibody.

Nahimana A, Aubry D, Breton CS, Majjigapu SR, Sordat B, Vogel P, Duchosal MA.

Leuk Lymphoma. 2014 Sep;55(9):2141-50. doi: 10.3109/10428194.2013.869325. Epub 2014 Jan 24.

PMID:
24283753
9.

Amide formation in one pot from carboxylic acids and amines via carboxyl and sulfinyl mixed anhydrides.

Zambroń BK, Dubbaka SR, Marković D, Moreno-Clavijo E, Vogel P.

Org Lett. 2013 May 17;15(10):2550-3. doi: 10.1021/ol401053y. Epub 2013 May 3.

PMID:
23642170
10.

A C-linked disaccharide analogue of Thomsen-Friedenreich epitope induces a strong immune response in mice.

Awad L, Madani R, Gillig A, Kolympadi M, Philgren M, Muhs A, Gérard C, Vogel P.

Chemistry. 2012 Jul 9;18(28):8578-82. doi: 10.1002/chem.201200364. Epub 2012 Jun 12. No abstract available.

PMID:
22692824
11.

Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition.

Röhrig UF, Majjigapu SR, Grosdidier A, Bron S, Stroobant V, Pilotte L, Colau D, Vogel P, Van den Eynde BJ, Zoete V, Michielin O.

J Med Chem. 2012 Jun 14;55(11):5270-90. doi: 10.1021/jm300260v. Epub 2012 May 22.

PMID:
22616902
12.

Determining the Role of the Aromatic Ring of N-Arylmethyl ent-conduramine F-1 in their Interactions with α-Glucosidases by Saturation Transfer Difference NMR Spectroscopy Experiments.

Hernández Daranas A, Koteich Khatib S, Lysek R, Vogel P, Gavín JA.

ChemistryOpen. 2012 Feb;1(1):13-6. doi: 10.1002/open.201100004. Epub 2012 Jan 2. No abstract available.

13.

Synthesis of branched seven-membered 1-N-iminosugars and their evaluation as glycosidase inhibitors.

Li H, Zhang Y, Favre S, Vogel P, Sollogoub M, Blériot Y.

Carbohydr Res. 2012 Jul 15;356:110-4. doi: 10.1016/j.carres.2011.10.039. Epub 2011 Nov 9.

PMID:
22129839
14.

Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols.

Bello C, Dal Bello G, Cea M, Nahimana A, Aubry D, Garuti A, Motta G, Moran E, Fruscione F, Pronzato P, Grossi F, Patrone F, Ballestrero A, Dupuis M, Sordat B, Zimmermann K, Loretan J, Wartmann M, Duchosal MA, Nencioni A, Vogel P.

Bioorg Med Chem. 2011 Dec 15;19(24):7720-7. doi: 10.1016/j.bmc.2011.07.053. Epub 2011 Jul 30.

PMID:
22079865
15.

Glycochemistry today.

Vogel P.

Chimia (Aarau). 2011;65(1-2):7-9. No abstract available.

PMID:
21469436
16.

Concise synthesis of complicated polypropionates through one-pot dissymmetrical two-directional chain elongation.

Exner CJ, Turks M, Fonquerne F, Vogel P.

Chemistry. 2011 Apr 4;17(15):4246-53. doi: 10.1002/chem.201003264. Epub 2011 Mar 8.

PMID:
21387431
17.

Total asymmetric syntheses of β-hydroxy-δ-lactones via Umpolung with sulfur dioxide.

Exner CJ, Laclef S, Poli F, Turks M, Vogel P.

J Org Chem. 2011 Feb 4;76(3):840-5. doi: 10.1021/jo102035d. Epub 2011 Jan 10.

PMID:
21218837
18.
19.

Total synthesis and determination of the absolute configuration of (-)-dolabriferol.

Laclef S, Turks M, Vogel P.

Angew Chem Int Ed Engl. 2010 Nov 2;49(45):8525-7. doi: 10.1002/anie.201003735. No abstract available.

PMID:
20865714
20.

Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity.

Borcard F, Baud M, Bello C, Dal Bello G, Grossi F, Pronzato P, Cea M, Nencioni A, Vogel P.

Bioorg Med Chem Lett. 2010 Sep 1;20(17):5353-6. doi: 10.1016/j.bmcl.2009.09.019. Epub 2009 Sep 10.

PMID:
20688516

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