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Items: 1 to 20 of 72

1.

Exploring the antimalarial potential of the methoxy-thiazinoquinone scaffold: Identification of a new lead candidate.

Imperatore C, Persico M, Senese M, Aiello A, Casertano M, Luciano P, Basilico N, Parapini S, Paladino A, Fattorusso C, Menna M.

Bioorg Chem. 2019 Apr;85:240-252. doi: 10.1016/j.bioorg.2018.12.031. Epub 2019 Jan 3.

PMID:
30640072
2.

Interplay between Plasmodium falciparum haemozoin and L-arginine: implication for nitric oxide production.

Corbett Y, D'Alessandro S, Parapini S, Scaccabarozzi D, Kalantari P, Zava S, Giavarini F, Caruso D, Colombo I, Egan TJ, Basilico N.

Malar J. 2018 Dec 6;17(1):456. doi: 10.1186/s12936-018-2602-0.

3.

Malaria pigment accelerates MTT - formazan exocytosis in human endothelial cells.

D'Alessandro S, Corbett Y, Parapini S, Perego F, Cavicchini L, Signorini L, Delbue S, Perego C, Ferrante P, Taramelli D, Basilico N.

Parasitology. 2019 Mar;146(3):399-406. doi: 10.1017/S0031182018001579. Epub 2018 Oct 1.

PMID:
30269694
4.

Novel Aminoquinoline Derivatives Significantly Reduce Parasite Load in Leishmania infantum Infected Mice.

Konstantinović J, Videnović M, Orsini S, Bogojević K, D'Alessandro S, Scaccabarozzi D, Terzić Jovanović N, Gradoni L, Basilico N, Šolaja BA.

ACS Med Chem Lett. 2018 May 4;9(7):629-634. doi: 10.1021/acsmedchemlett.8b00053. eCollection 2018 Jul 12.

PMID:
30034591
5.

Facile Preparation of N-Glycosylated 10-Piperazinyl Artemisinin Derivatives and Evaluation of Their Antimalarial and Cytotoxic Activities.

Wu Y, Parapini S, Williams ID, Misiano P, Wong HN, Taramelli D, Basilico N, Haynes RK.

Molecules. 2018 Jul 13;23(7). pii: E1713. doi: 10.3390/molecules23071713.

6.

Metabolic Responses in Endothelial Cells Following Exposure to Ketone Bodies.

Meroni E, Papini N, Criscuoli F, Casiraghi MC, Massaccesi L, Basilico N, Erba D.

Nutrients. 2018 Feb 22;10(2). pii: E250. doi: 10.3390/nu10020250.

7.

Benzimidazole derivatives endowed with potent antileishmanial activity.

Tonelli M, Gabriele E, Piazza F, Basilico N, Parapini S, Tasso B, Loddo R, Sparatore F, Sparatore A.

J Enzyme Inhib Med Chem. 2018 Dec;33(1):210-226. doi: 10.1080/14756366.2017.1410480.

8.

In Vivo and In Vitro Activities and ADME-Tox Profile of a Quinolizidine-Modified 4-Aminoquinoline: A Potent Anti-P. falciparum and Anti-P. vivax Blood-Stage Antimalarial.

Basilico N, Parapini S, Sparatore A, Romeo S, Misiano P, Vivas L, Yardley V, Croft SL, Habluetzel A, Lucantoni L, Renia L, Russell B, Suwanarusk R, Nosten F, Dondio G, Bigogno C, Jabes D, Taramelli D.

Molecules. 2017 Dec 1;22(12). pii: E2102. doi: 10.3390/molecules22122102.

9.

Malaria pigment stimulates chemokine production by human microvascular endothelium.

Basilico N, Corbett Y, D' Alessandro S, Parapini S, Prato M, Girelli D, Misiano P, Olliaro P, Taramelli D.

Acta Trop. 2017 Aug;172:125-131. doi: 10.1016/j.actatropica.2017.05.002. Epub 2017 May 2.

PMID:
28476599
10.

Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents.

Pieroni M, Azzali E, Basilico N, Parapini S, Zolkiewski M, Beato C, Annunziato G, Bruno A, Vacondio F, Costantino G.

J Med Chem. 2017 Mar 9;60(5):1959-1970. doi: 10.1021/acs.jmedchem.6b01685. Epub 2017 Feb 14.

PMID:
28128956
11.

Chloroquine-containing organoruthenium complexes are fast-acting multistage antimalarial agents.

Macedo TS, Colina-Vegas L, DA Paixão M, Navarro M, Barreto BC, Oliveira PC, Macambira SG, Machado M, Prudêncio M, D'Alessandro S, Basilico N, Moreira DR, Batista AA, Soares MB.

Parasitology. 2016 Oct;143(12):1543-56. doi: 10.1017/S0031182016001153. Epub 2016 Jul 21.

PMID:
27439976
12.

Exploring clotrimazole-based pharmacophore: 3D-QSAR studies and synthesis of novel antiplasmodial agents.

Brogi S, Brindisi M, Joshi BP, Sanna Coccone S, Parapini S, Basilico N, Novellino E, Campiani G, Gemma S, Butini S.

Bioorg Med Chem Lett. 2015 Nov 15;25(22):5412-8. doi: 10.1016/j.bmcl.2015.09.007. Epub 2015 Sep 5.

PMID:
26428874
13.

Dextran-shelled oxygen-loaded nanodroplets reestablish a normoxia-like pro-angiogenic phenotype and behavior in hypoxic human dermal microvascular endothelium.

Basilico N, Magnetto C, D'Alessandro S, Panariti A, Rivolta I, Genova T, Khadjavi A, Gulino GR, Argenziano M, Soster M, Cavalli R, Giribaldi G, Guiot C, Prato M.

Toxicol Appl Pharmacol. 2015 Nov 1;288(3):330-8. doi: 10.1016/j.taap.2015.08.005. Epub 2015 Aug 12.

14.

Synthesis and Antiplasmodial Activity of Novel Chloroquine Analogues with Bulky Basic Side Chains.

Tasso B, Novelli F, Tonelli M, Barteselli A, Basilico N, Parapini S, Taramelli D, Sparatore A, Sparatore F.

ChemMedChem. 2015 Sep;10(9):1570-83. doi: 10.1002/cmdc.201500195. Epub 2015 Jul 24.

PMID:
26213237
15.

Modified quaternary ammonium salts as potential antimalarial agents.

Basilico N, Migotto M, Ilboudo DP, Taramelli D, Stradi R, Pini E.

Bioorg Med Chem. 2015 Aug 1;23(15):4681-7. doi: 10.1016/j.bmc.2015.05.055. Epub 2015 Jun 3.

PMID:
26081764
16.

Salinomycin and other ionophores as a new class of antimalarial drugs with transmission-blocking activity.

D'Alessandro S, Corbett Y, Ilboudo DP, Misiano P, Dahiya N, Abay SM, Habluetzel A, Grande R, Gismondo MR, Dechering KJ, Koolen KM, Sauerwein RW, Taramelli D, Basilico N, Parapini S.

Antimicrob Agents Chemother. 2015 Sep;59(9):5135-44. doi: 10.1128/AAC.04332-14. Epub 2015 Jun 8.

17.

Glycosyl hydroperoxides: a new class of potential antimalarial agents.

Szechner B, Jaromin A, Parapini S, Basilico N, Grzeszczyk B, Furman B, Chmielewski M.

Bioorg Med Chem. 2015 Jul 1;23(13):3033-9. doi: 10.1016/j.bmc.2015.05.009. Epub 2015 May 14.

PMID:
26022082
18.

Stability of the antimalarial drug dihydroartemisinin under physiologically relevant conditions: implications for clinical treatment and pharmacokinetic and in vitro assays.

Parapini S, Olliaro P, Navaratnam V, Taramelli D, Basilico N.

Antimicrob Agents Chemother. 2015 Jul;59(7):4046-52. doi: 10.1128/AAC.00183-15. Epub 2015 Apr 27.

19.

Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents.

De Monte C, Bizzarri B, Gidaro MC, Carradori S, Mollica A, Luisi G, Granese A, Alcaro S, Costa G, Basilico N, Parapini S, Scaltrito MM, Masia C, Sisto F.

J Enzyme Inhib Med Chem. 2015 Dec;30(6):1027-33. doi: 10.3109/14756366.2014.1001755. Epub 2015 Sep 4.

PMID:
25766747
20.

Clofazimine analogs with antileishmanial and antiplasmodial activity.

Barteselli A, Casagrande M, Basilico N, Parapini S, Rusconi CM, Tonelli M, Boido V, Taramelli D, Sparatore F, Sparatore A.

Bioorg Med Chem. 2015 Jan 1;23(1):55-65. doi: 10.1016/j.bmc.2014.11.028. Epub 2014 Nov 26.

PMID:
25497962

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