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Items: 1 to 20 of 29

1.

Efficacy of a Selective Binder of αVβ3 Integrin Linked to the Tyrosine Kinase Inhibitor Sunitinib in Ovarian Carcinoma Preclinical Models.

Sartori A, Corno C, De Cesare M, Scanziani E, Minoli L, Battistini L, Zanardi F, Perego P.

Cancers (Basel). 2019 Apr 13;11(4). pii: E531. doi: 10.3390/cancers11040531.

2.

Integrin-targeted AmpRGD sunitinib liposomes as integrated antiangiogenic tools.

Bianchini F, De Santis A, Portioli E, Russo Krauss I, Battistini L, Curti C, Peppicelli S, Calorini L, D'Errico G, Zanardi F, Sartori A.

Nanomedicine. 2019 Mar 6;18:135-145. doi: 10.1016/j.nano.2019.02.015. [Epub ahead of print]

PMID:
30849548
3.

Cell-targeted c(AmpRGD)-sunitinib molecular conjugates impair tumor growth of melanoma.

Bianchini F, Portioli E, Ferlenghi F, Vacondio F, Andreucci E, Biagioni A, Ruzzolini J, Peppicelli S, Lulli M, Calorini L, Battistini L, Zanardi F, Sartori A.

Cancer Lett. 2019 Apr 1;446:25-37. doi: 10.1016/j.canlet.2018.12.021. Epub 2019 Jan 11.

PMID:
30639534
4.

Synthesis of Novel c(AmpRGD)-Sunitinib Dual Conjugates as Molecular Tools Targeting the αvβ3 Integrin/VEGFR2 Couple and Impairing Tumor-Associated Angiogenesis.

Sartori A, Portioli E, Battistini L, Calorini L, Pupi A, Vacondio F, Arosio D, Bianchini F, Zanardi F.

J Med Chem. 2017 Jan 12;60(1):248-262. doi: 10.1021/acs.jmedchem.6b01266. Epub 2016 Dec 20.

PMID:
27997164
5.

Organocatalytic, Asymmetric Eliminative [4+2] Cycloaddition of Allylidene Malononitriles with Enals: Rapid Entry to Cyclohexadiene-Embedding Linear and Angular Polycycles.

Brindani N, Rassu G, Dell'Amico L, Zambrano V, Pinna L, Curti C, Sartori A, Battistini L, Casiraghi G, Pelosi G, Greco D, Zanardi F.

Angew Chem Int Ed Engl. 2015 Jun 15;54(25):7386-90. doi: 10.1002/anie.201501894. Epub 2015 May 7.

PMID:
25950770
6.

Pushing the boundaries of vinylogous reactivity: catalytic enantioselective mukaiyama aldol reactions of highly unsaturated 2-silyloxyindoles.

Curti C, Sartori A, Battistini L, Brindani N, Rassu G, Pelosi G, Lodola A, Mor M, Casiraghi G, Zanardi F.

Chemistry. 2015 Apr 20;21(17):6433-42. doi: 10.1002/chem.201500083. Epub 2015 Mar 3.

PMID:
25735832
7.

Exploring the vinylogous reactivity of cyclohexenylidene malononitriles: switchable regioselectivity in the organocatalytic asymmetric addition to enals giving highly enantioenriched carbabicyclic structures.

Dell'Amico L, Rassu G, Zambrano V, Sartori A, Curti C, Battistini L, Pelosi G, Casiraghi G, Zanardi F.

J Am Chem Soc. 2014 Aug 6;136(31):11107-14. doi: 10.1021/ja5054576. Epub 2014 Jul 24.

PMID:
25032901
8.

Enhancement of the uptake and cytotoxic activity of doxorubicin in cancer cells by novel cRGD-semipeptide-anchoring liposomes.

Battistini L, Burreddu P, Sartori A, Arosio D, Manzoni L, Paduano L, D'Errico G, Sala R, Reia L, Bonomini S, Rassu G, Zanardi F.

Mol Pharm. 2014 Jul 7;11(7):2280-93. doi: 10.1021/mp400718j. Epub 2014 May 22.

PMID:
24819754
9.

3-Alkenyl-2-silyloxyindoles in vinylogous Mannich reactions: synthesis of aminated indole-based scaffolds and products.

Ranieri B, Sartori A, Curti C, Battistini L, Rassu G, Pelosi G, Casiraghi G, Zanardi F.

Org Lett. 2014 Feb 7;16(3):932-5. doi: 10.1021/ol4036598. Epub 2014 Jan 16.

PMID:
24432768
10.

Synthesis, structure and inhibitory activity of a stereoisomer of oseltamivir carboxylate.

Sartori A, Dell'Amico L, Battistini L, Curti C, Rivara S, Pala D, Kerry PS, Pelosi G, Casiraghi G, Rassu G, Zanardi F.

Org Biomol Chem. 2014 Mar 14;12(10):1561-9. doi: 10.1039/c3ob42069h.

PMID:
24425043
11.

Design, synthesis, and biological evaluation of novel cRGD-paclitaxel conjugates for integrin-assisted drug delivery.

Pilkington-Miksa M, Arosio D, Battistini L, Belvisi L, De Matteo M, Vasile F, Burreddu P, Carta P, Rassu G, Perego P, Carenini N, Zunino F, De Cesare M, Castiglioni V, Scanziani E, Scolastico C, Casiraghi G, Zanardi F, Manzoni L.

Bioconjug Chem. 2012 Aug 15;23(8):1610-22. doi: 10.1021/bc300164t. Epub 2012 Jul 20.

PMID:
22770429
12.

Bifunctional cinchona alkaloid/thiourea catalyzes direct and enantioselective vinylogous Michael addition of 3-alkylidene oxindoles to nitroolefins.

Curti C, Rassu G, Zambrano V, Pinna L, Pelosi G, Sartori A, Battistini L, Zanardi F, Casiraghi G.

Angew Chem Int Ed Engl. 2012 Jun 18;51(25):6200-4. doi: 10.1002/anie.201202027. Epub 2012 May 8. No abstract available.

PMID:
22565658
13.

Diastereo- and enantioselective catalytic vinylogous Mukaiyama-Mannich reactions of pyrrole-based silyl dienolates with alkyl-substituted aldehydes.

Ranieri B, Curti C, Battistini L, Sartori A, Pinna L, Casiraghi G, Zanardi F.

J Org Chem. 2011 Dec 16;76(24):10291-8. doi: 10.1021/jo201875a. Epub 2011 Nov 22.

PMID:
22059699
14.

Catalytic, asymmetric hypervinylogous Mukaiyama aldol reactions of extended furan-based silyl enolates.

Curti C, Battistini L, Sartori A, Lodola A, Mor M, Rassu G, Pelosi G, Zanardi F, Casiraghi G.

Org Lett. 2011 Sep 2;13(17):4738-41. doi: 10.1021/ol2020626. Epub 2011 Aug 11.

PMID:
21834551
15.

The vinylogous aldol and related addition reactions: ten years of progress.

Casiraghi G, Battistini L, Curti C, Rassu G, Zanardi F.

Chem Rev. 2011 May 11;111(5):3076-154. doi: 10.1021/cr100304n. Epub 2011 Mar 24. Review. No abstract available.

PMID:
21434642
16.

anti-Selective, catalytic asymmetric vinylogous Mukaiyama Mannich reactions of pyrrole-based silyl dienolates with N-aryl aldimines.

Curti C, Battistini L, Ranieri B, Pelosi G, Rassu G, Casiraghi G, Zanardi F.

J Org Chem. 2011 Apr 1;76(7):2248-52. doi: 10.1021/jo1021234. Epub 2011 Mar 7.

PMID:
21381711
17.

Uncatalyzed, diastereoselective vinylogous Mukaiyama aldol reactions on aqueous media: pyrrole vs furan 2-silyloxy dienes.

Curti C, Battistini L, Zanardi F, Rassu G, Zambrano V, Pinna L, Casiraghi G.

J Org Chem. 2010 Dec 17;75(24):8681-4. doi: 10.1021/jo101799e. Epub 2010 Nov 18.

PMID:
21086960
18.

Asymmetric total synthesis of 1-deoxy-7,8-di-epi-castanospermine.

Zambrano V, Rassu G, Roggio A, Pinna L, Zanardi F, Curti C, Casiraghi G, Battistini L.

Org Biomol Chem. 2010 Apr 7;8(7):1725-30. doi: 10.1039/b924721a. Epub 2010 Feb 9.

PMID:
20237688
19.

4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation.

Battistini L, Burreddu P, Carta P, Rassu G, Auzzas L, Curti C, Zanardi F, Manzoni L, Araldi EM, Scolastico C, Casiraghi G.

Org Biomol Chem. 2009 Dec 7;7(23):4924-35. doi: 10.1039/b914836a. Epub 2009 Oct 6.

PMID:
19907783
20.

Vicarious silylative Mukaiyama aldol reaction: a vinylogous extension.

Curti C, Sartori A, Battistini L, Rassu G, Burreddu P, Zanardi F, Casiraghi G.

J Org Chem. 2008 Jul 18;73(14):5446-51. doi: 10.1021/jo800741c. Epub 2008 Jun 13.

PMID:
18549289

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