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Items: 1 to 20 of 21

1.

Organic Diselenides: Versatile Reagents, Precursors, and Intriguing Biologically Active Compounds.

Santi C, Tomassini C, Sancineto L.

Chimia (Aarau). 2017 Sep 27;71(9):592-595. doi: 10.2533/chimia.2017.592. Review.

PMID:
30188290
2.

2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors.

Nkizinkiko Y, Desantis J, Koivunen J, Haikarainen T, Murthy S, Sancineto L, Massari S, Ianni F, Obaji E, Loza MI, Pihlajaniemi T, Brea J, Tabarrini O, Lehtiö L.

Sci Rep. 2018 Jan 26;8(1):1680. doi: 10.1038/s41598-018-19872-3.

3.

NCp7: targeting a multitask protein for next-generation anti-HIV drug development part 2. Noncovalent inhibitors and nucleic acid binders.

Iraci N, Tabarrini O, Santi C, Sancineto L.

Drug Discov Today. 2018 Mar;23(3):687-695. doi: 10.1016/j.drudis.2018.01.022. Epub 2018 Jan 8. Review.

PMID:
29326078
4.

NCp7: targeting a multitasking protein for next-generation anti-HIV drug development part 1: covalent inhibitors.

Sancineto L, Iraci N, Tabarrini O, Santi C.

Drug Discov Today. 2018 Feb;23(2):260-271. doi: 10.1016/j.drudis.2017.10.017. Epub 2017 Oct 28. Review.

PMID:
29107765
5.

Selenocompounds in Cancer Therapy: An Overview.

Bartolini D, Sancineto L, Fabro de Bem A, Tew KD, Santi C, Radi R, Toquato P, Galli F.

Adv Cancer Res. 2017;136:259-302. doi: 10.1016/bs.acr.2017.07.007. Epub 2017 Sep 28. Review.

PMID:
29054421
6.

Induction of reactive oxygen species by diphenyl diselenide is preceded by changes in cell morphology and permeability in Saccharomyces cerevisiae.

Galant LS, Braga MM, de Souza D, de Bem AF, Sancineto L, Santi C, da Rocha JBT.

Free Radic Res. 2017 Jul-Aug;51(7-8):657-668. doi: 10.1080/10715762.2017.1355054. Epub 2017 Aug 25.

PMID:
28840761
7.

Atom Efficient Preparation of Zinc Selenates for the Synthesis of Selenol Esters under "On Water" Conditions.

Sancineto L, Pinto Vargas J, Monti B, Arca M, Lippolis V, Perin G, Lenardao EJ, Santi C.

Molecules. 2017 Jun 8;22(6). pii: E953. doi: 10.3390/molecules22060953.

8.

Green Hydroselenation of Aryl Alkynes: Divinyl Selenides as a Precursor of Resveratrol.

Perin G, Barcellos AM, Luz EQ, Borges EL, Jacob RG, Lenardão EJ, Sancineto L, Santi C.

Molecules. 2017 Feb 20;22(2). pii: E327. doi: 10.3390/molecules22020327.

9.

Water and Aqueous Mixtures as Convenient Alternative Media for Organoselenium Chemistry.

Santi C, Jacob RG, Monti B, Bagnoli L, Sancineto L, Lenardão EJ.

Molecules. 2016 Nov 6;21(11). pii: E1482. Review.

10.

Diphenyl diselenide derivatives inhibit microbial biofilm formation involved in wound infection.

Sancineto L, Piccioni M, De Marco S, Pagiotti R, Nascimento V, Braga AL, Santi C, Pietrella D.

BMC Microbiol. 2016 Sep 21;16(1):220.

11.

Organoselenium Compounds as Phytochemicals from the Natural Kingdom.

Achibat H, AlOmari NA, Messina F, Sancineto L, Khouili M, Santi C.

Nat Prod Commun. 2015 Nov;10(11):1885-92. Review.

PMID:
26749817
12.

Design and Synthesis of DiselenoBisBenzamides (DISeBAs) as Nucleocapsid Protein 7 (NCp7) Inhibitors with anti-HIV Activity.

Sancineto L, Mariotti A, Bagnoli L, Marini F, Desantis J, Iraci N, Santi C, Pannecouque C, Tabarrini O.

J Med Chem. 2015 Dec 24;58(24):9601-14. doi: 10.1021/acs.jmedchem.5b01183. Epub 2015 Dec 10.

PMID:
26613134
13.

Selenium Catalyzed Oxidation of Aldehydes: Green Synthesis of Carboxylic Acids and Esters.

Sancineto L, Tidei C, Bagnoli L, Marini F, Lenardão EJ, Santi C.

Molecules. 2015 Jun 8;20(6):10496-510. doi: 10.3390/molecules200610496.

14.

Synthesis and biological evaluation of new nitrogen-containing diselenides.

Nascimento V, Ferreira NL, Canto RF, Schott KL, Waczuk EP, Sancineto L, Santi C, Rocha JB, Braga AL.

Eur J Med Chem. 2014 Nov 24;87:131-9. doi: 10.1016/j.ejmech.2014.09.022. Epub 2014 Sep 8.

PMID:
25244678
15.

Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands.

Sancineto L, Iraci N, Barreca ML, Massari S, Manfroni G, Corazza G, Cecchetti V, Marcello A, Daelemans D, Pannecouque C, Tabarrini O.

Bioorg Med Chem. 2014 Sep 1;22(17):4658-66. doi: 10.1016/j.bmc.2014.07.018. Epub 2014 Jul 22.

PMID:
25127466
16.

Structural investigation of cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly.

Massari S, Nannetti G, Goracci L, Sancineto L, Muratore G, Sabatini S, Manfroni G, Mercorelli B, Cecchetti V, Facchini M, Palù G, Cruciani G, Loregian A, Tabarrini O.

J Med Chem. 2013 Dec 27;56(24):10118-31. doi: 10.1021/jm401560v. Epub 2013 Dec 13.

PMID:
24313730
17.

Computer-aided design, synthesis and validation of 2-phenylquinazolinone fragments as CDK9 inhibitors with anti-HIV-1 Tat-mediated transcription activity.

Sancineto L, Iraci N, Massari S, Attanasio V, Corazza G, Barreca ML, Sabatini S, Manfroni G, Avanzi NR, Cecchetti V, Pannecouque C, Marcello A, Tabarrini O.

ChemMedChem. 2013 Dec;8(12):1941-53. doi: 10.1002/cmdc.201300287. Epub 2013 Oct 21.

PMID:
24150998
18.

Design, synthesis, and evaluation of WC5 analogues as inhibitors of human cytomegalovirus Immediate-Early 2 protein, a promising target for anti-HCMV treatment.

Massari S, Mercorelli B, Sancineto L, Sabatini S, Cecchetti V, Gribaudo G, Palù G, Pannecouque C, Loregian A, Tabarrini O.

ChemMedChem. 2013 Aug;8(8):1403-14. doi: 10.1002/cmdc.201300106. Epub 2013 Jun 11.

PMID:
23757191
19.

Re-evolution of the 2-phenylquinolines: ligand-based design, synthesis, and biological evaluation of a potent new class of Staphylococcus aureus NorA efflux pump inhibitors to combat antimicrobial resistance.

Sabatini S, Gosetto F, Iraci N, Barreca ML, Massari S, Sancineto L, Manfroni G, Tabarrini O, Dimovska M, Kaatz GW, Cecchetti V.

J Med Chem. 2013 Jun 27;56(12):4975-89. doi: 10.1021/jm400262a. Epub 2013 Jun 13.

PMID:
23710549
20.

From small to powerful: the fragments universe and its "chem-appeal".

Sancineto L, Massari S, Iraci N, Tabarrini O.

Curr Med Chem. 2013;20(11):1355-81. Review.

PMID:
23410157

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