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Items: 1 to 20 of 36

1.

Efficacy of a Selective Binder of αVβ3 Integrin Linked to the Tyrosine Kinase Inhibitor Sunitinib in Ovarian Carcinoma Preclinical Models.

Sartori A, Corno C, De Cesare M, Scanziani E, Minoli L, Battistini L, Zanardi F, Perego P.

Cancers (Basel). 2019 Apr 13;11(4). pii: E531. doi: 10.3390/cancers11040531.

2.

Integrin-targeted AmpRGD sunitinib liposomes as integrated antiangiogenic tools.

Bianchini F, De Santis A, Portioli E, Russo Krauss I, Battistini L, Curti C, Peppicelli S, Calorini L, D'Errico G, Zanardi F, Sartori A.

Nanomedicine. 2019 Mar 6;18:135-145. doi: 10.1016/j.nano.2019.02.015. [Epub ahead of print]

PMID:
30849548
3.

Acetaldehyde Silyl Enol Ethers in Enantioselective Mukaiyama Aldol Reactions: Enzyme-Like Organocatalysis in Action.

Dell'Amico L, Zanardi F.

Angew Chem Int Ed Engl. 2019 Mar 11;58(11):3264-3266. doi: 10.1002/anie.201812964. Epub 2019 Feb 7. Review.

PMID:
30730598
4.

Cell-targeted c(AmpRGD)-sunitinib molecular conjugates impair tumor growth of melanoma.

Bianchini F, Portioli E, Ferlenghi F, Vacondio F, Andreucci E, Biagioni A, Ruzzolini J, Peppicelli S, Lulli M, Calorini L, Battistini L, Zanardi F, Sartori A.

Cancer Lett. 2019 Apr 1;446:25-37. doi: 10.1016/j.canlet.2018.12.021. Epub 2019 Jan 11.

PMID:
30639534
5.

Gold Nanoparticles Functionalized with RGD-Semipeptides: A Simple yet Highly Effective Targeting System for αV β3 Integrins.

Maggi V, Bianchini F, Portioli E, Peppicelli S, Lulli M, Bani D, Sole RD, Zanardi F, Sartori A, Fiammengo R.

Chemistry. 2018 Aug 14;24(46):12093-12100. doi: 10.1002/chem.201801823. Epub 2018 Jul 16.

PMID:
29923243
6.

Synthetic and analytical strategies for the quantification of phenyl-γ-valerolactone conjugated metabolites in human urine.

Brindani N, Mena P, Calani L, Benzie I, Choi SW, Brighenti F, Zanardi F, Curti C, Del Rio D.

Mol Nutr Food Res. 2017 Sep;61(9). doi: 10.1002/mnfr.201700077. Epub 2017 Jun 9.

PMID:
28440064
7.

Synthesis of Novel c(AmpRGD)-Sunitinib Dual Conjugates as Molecular Tools Targeting the αvβ3 Integrin/VEGFR2 Couple and Impairing Tumor-Associated Angiogenesis.

Sartori A, Portioli E, Battistini L, Calorini L, Pupi A, Vacondio F, Arosio D, Bianchini F, Zanardi F.

J Med Chem. 2017 Jan 12;60(1):248-262. doi: 10.1021/acs.jmedchem.6b01266. Epub 2016 Dec 20.

PMID:
27997164
8.

Exploiting the Distal Reactivity of Indolyl Methylenemalononitriles: An Asymmetric Organocatalyzed [4+2] Cycloaddition with Enals Enables the Assembly of Elusive Dihydrocarbazoles.

Rassu G, Curti C, Zambrano V, Pinna L, Brindani N, Pelosi G, Zanardi F.

Chemistry. 2016 Aug 26;22(36):12637-40. doi: 10.1002/chem.201602793. Epub 2016 Jul 28.

PMID:
27348410
9.

Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines.

Spadoni G, Bedini A, Lucarini S, Mari M, Caignard DH, Boutin JA, Delagrange P, Lucini V, Scaglione F, Lodola A, Zanardi F, Pala D, Mor M, Rivara S.

J Med Chem. 2015 Sep 24;58(18):7512-25. doi: 10.1021/acs.jmedchem.5b01066.

PMID:
26334942
10.

Organocatalytic, Asymmetric Eliminative [4+2] Cycloaddition of Allylidene Malononitriles with Enals: Rapid Entry to Cyclohexadiene-Embedding Linear and Angular Polycycles.

Brindani N, Rassu G, Dell'Amico L, Zambrano V, Pinna L, Curti C, Sartori A, Battistini L, Casiraghi G, Pelosi G, Greco D, Zanardi F.

Angew Chem Int Ed Engl. 2015 Jun 15;54(25):7386-90. doi: 10.1002/anie.201501894. Epub 2015 May 7.

PMID:
25950770
11.

Pushing the boundaries of vinylogous reactivity: catalytic enantioselective mukaiyama aldol reactions of highly unsaturated 2-silyloxyindoles.

Curti C, Sartori A, Battistini L, Brindani N, Rassu G, Pelosi G, Lodola A, Mor M, Casiraghi G, Zanardi F.

Chemistry. 2015 Apr 20;21(17):6433-42. doi: 10.1002/chem.201500083. Epub 2015 Mar 3.

PMID:
25735832
12.

Exploring the vinylogous reactivity of cyclohexenylidene malononitriles: switchable regioselectivity in the organocatalytic asymmetric addition to enals giving highly enantioenriched carbabicyclic structures.

Dell'Amico L, Rassu G, Zambrano V, Sartori A, Curti C, Battistini L, Pelosi G, Casiraghi G, Zanardi F.

J Am Chem Soc. 2014 Aug 6;136(31):11107-14. doi: 10.1021/ja5054576. Epub 2014 Jul 24.

PMID:
25032901
13.

Enhancement of the uptake and cytotoxic activity of doxorubicin in cancer cells by novel cRGD-semipeptide-anchoring liposomes.

Battistini L, Burreddu P, Sartori A, Arosio D, Manzoni L, Paduano L, D'Errico G, Sala R, Reia L, Bonomini S, Rassu G, Zanardi F.

Mol Pharm. 2014 Jul 7;11(7):2280-93. doi: 10.1021/mp400718j. Epub 2014 May 22.

PMID:
24819754
14.

3-Alkenyl-2-silyloxyindoles in vinylogous Mannich reactions: synthesis of aminated indole-based scaffolds and products.

Ranieri B, Sartori A, Curti C, Battistini L, Rassu G, Pelosi G, Casiraghi G, Zanardi F.

Org Lett. 2014 Feb 7;16(3):932-5. doi: 10.1021/ol4036598. Epub 2014 Jan 16.

PMID:
24432768
15.

Synthesis, structure and inhibitory activity of a stereoisomer of oseltamivir carboxylate.

Sartori A, Dell'Amico L, Battistini L, Curti C, Rivara S, Pala D, Kerry PS, Pelosi G, Casiraghi G, Rassu G, Zanardi F.

Org Biomol Chem. 2014 Mar 14;12(10):1561-9. doi: 10.1039/c3ob42069h.

PMID:
24425043
16.

Design, synthesis, and biological evaluation of novel cRGD-paclitaxel conjugates for integrin-assisted drug delivery.

Pilkington-Miksa M, Arosio D, Battistini L, Belvisi L, De Matteo M, Vasile F, Burreddu P, Carta P, Rassu G, Perego P, Carenini N, Zunino F, De Cesare M, Castiglioni V, Scanziani E, Scolastico C, Casiraghi G, Zanardi F, Manzoni L.

Bioconjug Chem. 2012 Aug 15;23(8):1610-22. doi: 10.1021/bc300164t. Epub 2012 Jul 20.

PMID:
22770429
17.

Bifunctional cinchona alkaloid/thiourea catalyzes direct and enantioselective vinylogous Michael addition of 3-alkylidene oxindoles to nitroolefins.

Curti C, Rassu G, Zambrano V, Pinna L, Pelosi G, Sartori A, Battistini L, Zanardi F, Casiraghi G.

Angew Chem Int Ed Engl. 2012 Jun 18;51(25):6200-4. doi: 10.1002/anie.201202027. Epub 2012 May 8. No abstract available.

PMID:
22565658
18.

Diastereo- and enantioselective catalytic vinylogous Mukaiyama-Mannich reactions of pyrrole-based silyl dienolates with alkyl-substituted aldehydes.

Ranieri B, Curti C, Battistini L, Sartori A, Pinna L, Casiraghi G, Zanardi F.

J Org Chem. 2011 Dec 16;76(24):10291-8. doi: 10.1021/jo201875a. Epub 2011 Nov 22.

PMID:
22059699
19.

Catalytic, asymmetric hypervinylogous Mukaiyama aldol reactions of extended furan-based silyl enolates.

Curti C, Battistini L, Sartori A, Lodola A, Mor M, Rassu G, Pelosi G, Zanardi F, Casiraghi G.

Org Lett. 2011 Sep 2;13(17):4738-41. doi: 10.1021/ol2020626. Epub 2011 Aug 11.

PMID:
21834551
20.

The vinylogous aldol and related addition reactions: ten years of progress.

Casiraghi G, Battistini L, Curti C, Rassu G, Zanardi F.

Chem Rev. 2011 May 11;111(5):3076-154. doi: 10.1021/cr100304n. Epub 2011 Mar 24. Review. No abstract available.

PMID:
21434642

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