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Items: 1 to 20 of 30

1.

Metal chelators for the inhibition of the lymphocytic choriomeningitis virus endonuclease domain.

Saez-Ayala M, Laban Yekwa E, Mondielli C, Roux L, Hernández S, Bailly F, Cotelle P, Rogolino D, Canard B, Ferron F, Alvarez K.

Antiviral Res. 2019 Feb;162:79-89. doi: 10.1016/j.antiviral.2018.12.008. Epub 2018 Dec 14.

PMID:
30557576
2.

Toward the Discovery of a Novel Class of YAP⁻TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP⁻TEAD Protein⁻Protein Interface.

Gibault F, Coevoet M, Sturbaut M, Farce A, Renault N, Allemand F, Guichou JF, Drucbert AS, Foulon C, Magnez R, Thuru X, Corvaisier M, Huet G, Chavatte P, Melnyk P, Bailly F, Cotelle P.

Cancers (Basel). 2018 May 8;10(5). pii: E140. doi: 10.3390/cancers10050140.

3.

Targeting Transcriptional Enhanced Associate Domains (TEADs).

Gibault F, Sturbaut M, Bailly F, Melnyk P, Cotelle P.

J Med Chem. 2018 Jun 28;61(12):5057-5072. doi: 10.1021/acs.jmedchem.7b00879. Epub 2017 Dec 28.

PMID:
29251924
4.

Inhibition of hepatitis B virus replication by N-hydroxyisoquinolinediones and related polyoxygenated heterocycles.

Edwards TC, Lomonosova E, Patel JA, Li Q, Villa JA, Gupta AK, Morrison LA, Bailly F, Cotelle P, Giannakopoulou E, Zoidis G, Tavis JE.

Antiviral Res. 2017 Jul;143:205-217. doi: 10.1016/j.antiviral.2017.04.012. Epub 2017 Apr 25.

5.

Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway.

Gibault F, Bailly F, Corvaisier M, Coevoet M, Huet G, Melnyk P, Cotelle P.

ChemMedChem. 2017 Jun 21;12(12):954-961. doi: 10.1002/cmdc.201700063. Epub 2017 Apr 20.

PMID:
28334506
6.

2-hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs) as human immunodeficiency virus type 1 integrase inhibitors: Influence of the alkylcarboxamide substitution of position 4.

Billamboz M, Suchaud V, Bailly F, Lion C, Andréola ML, Christ F, Debyser Z, Cotelle P.

Eur J Med Chem. 2016 Jul 19;117:256-68. doi: 10.1016/j.ejmech.2016.03.083. Epub 2016 Mar 28.

PMID:
27105029
7.

Non-Photoinduced Biological Properties of Verteporfin.

Gibault F, Corvaisier M, Bailly F, Huet G, Melnyk P, Cotelle P.

Curr Med Chem. 2016;23(11):1171-84. Review.

PMID:
26980565
8.

The preclinical discovery and development of dolutegravir for the treatment of HIV.

Bailly F, Cotelle P.

Expert Opin Drug Discov. 2015;10(11):1243-53. doi: 10.1517/17460441.2015.1064896. Epub 2015 Sep 7. Review.

PMID:
26517818
9.

4-Substituted 2-Hydroxyisoquinoline-1,3(2H,4H)-diones as a Novel Class of HIV-1 Integrase Inhibitors.

Billamboz M, Suchaud V, Bailly F, Lion C, Demeulemeester J, Calmels C, Andréola ML, Christ F, Debyser Z, Cotelle P.

ACS Med Chem Lett. 2013 May 17;4(7):606-11. doi: 10.1021/ml400009t. eCollection 2013 Jul 11.

10.

Hepatitis B virus replication is blocked by a 2-hydroxyisoquinoline-1,3(2H,4H)-dione (HID) inhibitor of the viral ribonuclease H activity.

Cai CW, Lomonosova E, Moran EA, Cheng X, Patel KB, Bailly F, Cotelle P, Meyers MJ, Tavis JE.

Antiviral Res. 2014 Aug;108:48-55. doi: 10.1016/j.antiviral.2014.05.007. Epub 2014 May 20.

11.

Investigation of a novel series of 2-hydroxyisoquinoline-1,3(2H,4H)-diones as human immunodeficiency virus type 1 integrase inhibitors.

Suchaud V, Bailly F, Lion C, Calmels C, Andréola ML, Christ F, Debyser Z, Cotelle P.

J Med Chem. 2014 Jun 12;57(11):4640-60. doi: 10.1021/jm500109z. Epub 2014 May 14.

PMID:
24793360
12.

2-Hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs), novel inhibitors of HIV integrase with a high barrier to resistance.

Desimmie BA, Demeulemeester J, Suchaud V, Taltynov O, Billamboz M, Lion C, Bailly F, Strelkov SV, Debyser Z, Cotelle P, Christ F.

ACS Chem Biol. 2013;8(6):1187-94. doi: 10.1021/cb4000426. Epub 2013 Apr 2.

PMID:
23517458
13.

Antiproliferative and apoptotic effects of the oxidative dimerization product of methyl caffeate on human breast cancer cells.

Bailly F, Toillon RA, Tomavo O, Jouy N, Hondermarck H, Cotelle P.

Bioorg Med Chem Lett. 2013 Jan 15;23(2):574-8. doi: 10.1016/j.bmcl.2012.11.009. Epub 2012 Nov 22.

PMID:
23228470
14.

Development of a series of 3-hydroxyquinolin-2(1H)-ones as selective inhibitors of HIV-1 reverse transcriptase associated RNase H activity.

Suchaud V, Bailly F, Lion C, Tramontano E, Esposito F, Corona A, Christ F, Debyser Z, Cotelle P.

Bioorg Med Chem Lett. 2012 Jun 15;22(12):3988-92. doi: 10.1016/j.bmcl.2012.04.096. Epub 2012 Apr 30.

PMID:
22607675
15.

Magnesium chelating 2-hydroxyisoquinoline-1,3(2H,4H)-diones, as inhibitors of HIV-1 integrase and/or the HIV-1 reverse transcriptase ribonuclease H domain: discovery of a novel selective inhibitor of the ribonuclease H function.

Billamboz M, Bailly F, Lion C, Touati N, Vezin H, Calmels C, Andréola ML, Christ F, Debyser Z, Cotelle P.

J Med Chem. 2011 Mar 24;54(6):1812-24. doi: 10.1021/jm1014692. Epub 2011 Mar 2.

PMID:
21366258
16.

2-hydroxyisoquinoline-1,3(2H,4H)-diones as inhibitors of HIV-1 integrase and reverse transcriptase RNase H domain: influence of the alkylation of position 4.

Billamboz M, Bailly F, Lion C, Calmels C, Andréola ML, Witvrouw M, Christ F, Debyser Z, De Luca L, Chimirri A, Cotelle P.

Eur J Med Chem. 2011 Feb;46(2):535-46. doi: 10.1016/j.ejmech.2010.11.033. Epub 2010 Nov 27.

PMID:
21185110
17.

New 2-arylnaphthalenediols and triol inhibitors of HIV-1 integrase--discovery of a new polyhydroxylated antiviral agent.

Maurin C, Lion C, Bailly F, Touati N, Vezin H, Mbemba G, Mouscadet JF, Debyser Z, Witvrouw M, Cotelle P.

Bioorg Med Chem. 2010 Jul 15;18(14):5194-201. doi: 10.1016/j.bmc.2010.05.059. Epub 2010 May 26.

PMID:
20541944
18.

Evaluation of aldose reductase inhibition and docking studies of 6'-nitro and 6',6''-dinitrorosmarinic acids.

Koukoulitsa C, Bailly F, Pegklidou K, Demopoulos VJ, Cotelle P.

Eur J Med Chem. 2010 Apr;45(4):1663-6. doi: 10.1016/j.ejmech.2009.12.007. Epub 2010 Jan 13.

PMID:
20071057
19.

Design, synthesis, and biological evaluation of a series of 2-hydroxyisoquinoline-1,3(2H,4H)-diones as dual inhibitors of human immunodeficiency virus type 1 integrase and the reverse transcriptase RNase H domain.

Billamboz M, Bailly F, Barreca ML, De Luca L, Mouscadet JF, Calmels C, Andréola ML, Witvrouw M, Christ F, Debyser Z, Cotelle P.

J Med Chem. 2008 Dec 25;51(24):7717-30. doi: 10.1021/jm8007085.

PMID:
19053754
20.

Synthesis and antiviral properties of some polyphenols related to Salvia genus.

Queffélec C, Bailly F, Mbemba G, Mouscadet JF, Hayes S, Debyser Z, Witvrouw M, Cotelle P.

Bioorg Med Chem Lett. 2008 Aug 15;18(16):4736-40. doi: 10.1016/j.bmcl.2008.06.063. Epub 2008 Jun 21.

PMID:
18674899

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