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Items: 11

1.

Thiazolidinone/thiazole based hybrids - New class of antitrypanosomal agents.

Kryshchyshyn A, Kaminskyy D, Karpenko O, Gzella A, Grellier P, Lesyk R.

Eur J Med Chem. 2019 Jul 15;174:292-308. doi: 10.1016/j.ejmech.2019.04.052. Epub 2019 Apr 24.

PMID:
31051403
2.

Synthesis of 5-enamine-4-thiazolidinone derivatives with trypanocidal and anticancer activity.

Holota S, Kryshchyshyn A, Derkach H, Trufin Y, Demchuk I, Gzella A, Grellier P, Lesyk R.

Bioorg Chem. 2019 May;86:126-136. doi: 10.1016/j.bioorg.2019.01.045. Epub 2019 Jan 22.

PMID:
30690336
3.

Isothiochromenothiazoles-A Class of Fused Thiazolidinone Derivatives with Established Anticancer Activity That Inhibits Growth of Trypanosoma brucei brucei.

Kryshchyshyn A, Kaminskyy D, Nektegayev I, Grellier P, Lesyk R.

Sci Pharm. 2018 Oct 19;86(4). pii: E47. doi: 10.3390/scipharm86040047.

4.

Thiopyrano[2,3-d]Thiazoles as New Efficient Scaffolds in Medicinal Chemistry.

Kryshchyshyn A, Roman O, Lozynskyi A, Lesyk R.

Sci Pharm. 2018 Jun 14;86(2). pii: E26. doi: 10.3390/scipharm86020026. Review.

5.

Development of Predictive QSAR Models of 4-Thiazolidinones Antitrypanosomal Activity Using Modern Machine Learning Algorithms.

Kryshchyshyn A, Devinyak O, Kaminskyy D, Grellier P, Lesyk R.

Mol Inform. 2018 May;37(5):e1700078. doi: 10.1002/minf.201700078. Epub 2017 Nov 14.

PMID:
29134756
6.

Anticancer properties of 4-thiazolidinone derivatives depend on peroxisome proliferator-activated receptor gamma (PPARγ).

Szychowski KA, Leja ML, Kaminskyy DV, Kryshchyshyn AP, Binduga UE, Pinyazhko OR, Lesyk RB, Tobiasz J, Gmiński J.

Eur J Med Chem. 2017 Dec 1;141:162-168. doi: 10.1016/j.ejmech.2017.09.071. Epub 2017 Sep 30.

PMID:
29031063
7.

Recent developments with rhodanine as a scaffold for drug discovery.

Kaminskyy D, Kryshchyshyn A, Lesyk R.

Expert Opin Drug Discov. 2017 Dec;12(12):1233-1252. doi: 10.1080/17460441.2017.1388370. Epub 2017 Oct 11. Review.

PMID:
29019278
8.

5-Ene-4-thiazolidinones - An efficient tool in medicinal chemistry.

Kaminskyy D, Kryshchyshyn A, Lesyk R.

Eur J Med Chem. 2017 Nov 10;140:542-594. doi: 10.1016/j.ejmech.2017.09.031. Epub 2017 Sep 20. Review.

PMID:
28987611
9.

Trends in research of antitrypanosomal agents among synthetic heterocycles.

Kryshchyshyn A, Kaminskyy D, Grellier P, Lesyk R.

Eur J Med Chem. 2014 Oct 6;85:51-64. doi: 10.1016/j.ejmech.2014.07.092. Epub 2014 Jul 25. Review.

PMID:
25072876
10.

Isothiocoumarin-3-carboxylic acid derivatives: synthesis, anticancer and antitrypanosomal activity evaluation.

Kaminskyy D, Kryshchyshyn A, Nektegayev I, Vasylenko O, Grellier P, Lesyk R.

Eur J Med Chem. 2014 Mar 21;75:57-66. doi: 10.1016/j.ejmech.2014.01.028. Epub 2014 Jan 25.

PMID:
24530491
11.

Fused Thiopyrano[2,3-d]thiazole Derivatives as Potential Anticancer Agents.

Kryshchyshyn A, Atamanyuk D, Lesyk R.

Sci Pharm. 2012 Jul-Sep;80(3):509-29. Epub 2012 May 3.

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