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Items: 18

1.

Synthesis, In Vitro Screening and Docking Studies of New Thiosemicarbazide Derivatives as Antitubercular Agents.

Pitucha M, Karczmarzyk Z, Swatko-Ossor M, Wysocki W, Wos M, Chudzik K, Ginalska G, Fruzinski A.

Molecules. 2019 Jan 11;24(2). pii: E251. doi: 10.3390/molecules24020251.

2.

Polysubstituted 3-trifluoromethylpyrazoles: regioselective (3 + 2)-cycloaddition of trifluoroacetonitrile imines with enol ethers and functional group transformations.

Utecht G, Fruziński A, Jasiński M.

Org Biomol Chem. 2018 Feb 21;16(8):1252-1257. doi: 10.1039/c7ob03126b.

PMID:
29392253
3.

Synthesis, Structure and Antiproliferative Activity of New pyrazolo[4,3- e]triazolo[4,5-b][1,2,4]triazine Derivatives.

Mojzych M, Tarasiuk P, Karczmarzyk Z, Juszczak M, Rzeski W, Fruzinski A, Wozny A.

Med Chem. 2018;14(1):53-59. doi: 10.2174/1573406413666171020114924.

PMID:
29065838
4.

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

Kuder KJ, Łażewska D, Kaleta M, Latacz G, Kottke T, Olejarz A, Karcz T, Fruziński A, Szczepańska K, Karolak-Wojciechowska J, Stark H, Kieć-Kononowicz K.

Bioorg Med Chem. 2017 May 15;25(10):2701-2712. doi: 10.1016/j.bmc.2017.03.031. Epub 2017 Mar 21.

PMID:
28372935
5.

Similarities and differences in affinity and binding modes of tricyclic pyrimido- and pyrazinoxanthines at human and rat adenosine receptors.

Szymańska E, Drabczyńska A, Karcz T, Müller CE, Köse M, Karolak-Wojciechowska J, Fruziński A, Schabikowski J, Doroz-Płonka A, Handzlik J, Kieć-Kononowicz K.

Bioorg Med Chem. 2016 Sep 15;24(18):4347-4362. doi: 10.1016/j.bmc.2016.07.028. Epub 2016 Jul 18.

PMID:
27485602
6.

Discovery of nitroaryl urea derivatives with antiproliferative properties.

Wróbel TM, Kiełbus M, Kaczor AA, Kryštof V, Karczmarzyk Z, Wysocki W, Fruziński A, Król SK, Grabarska A, Stepulak A, Matosiuk D.

J Enzyme Inhib Med Chem. 2016 Aug;31(4):608-18. doi: 10.3109/14756366.2015.1057716. Epub 2015 Jun 26.

PMID:
26114307
7.

Captopril and its dimer captopril disulfide: comparative structural and conformational studies.

Bojarska J, Maniukiewicz W, Fruziński A, Sieroń L, Remko M.

Acta Crystallogr C Struct Chem. 2015 Mar;71(Pt 3):199-203. doi: 10.1107/S2053229615002582. Epub 2015 Feb 18.

PMID:
25734850
8.

Structural studies, homology modeling and molecular docking of novel non-competitive antagonists of GluK1/GluK2 receptors.

Kaczor AA, Karczmarzyk Z, Fruziński A, Pihlaja K, Sinkkonen J, Wiinämaki K, Kronbach C, Unverferth K, Poso A, Matosiuk D.

Bioorg Med Chem. 2014 Jan 15;22(2):787-95. doi: 10.1016/j.bmc.2013.12.013. Epub 2013 Dec 12.

PMID:
24368028
9.

Synthesis of novel isothiazolopyridines and their in vitro evaluation against Mycobacterium and Propionibacterium acnes.

Malinka W, Swiątek P, Sliwińska M, Szponar B, Gamian A, Karczmarzyk Z, Fruziński A.

Bioorg Med Chem. 2013 Sep 1;21(17):5282-91. doi: 10.1016/j.bmc.2013.06.027. Epub 2013 Jun 19.

10.

2-(5,6-Diphenyl-1,2,4-triazin-3-yl)aniline.

Mojzych M, Karczmarzyk Z, Fruziński A.

Acta Crystallogr Sect E Struct Rep Online. 2012 Dec 1;68(Pt 12):o3278. doi: 10.1107/S1600536812044194. Epub 2012 Nov 3.

11.

Ethyl 2-(3-methyl-5-sulfanyl-idene-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetate.

Karczmarzyk Z, Pitucha M, Wysocki W, Fruziński A, Olender E.

Acta Crystallogr Sect E Struct Rep Online. 2012 Dec 1;68(Pt 12):o3264-5. doi: 10.1107/S1600536812044716. Epub 2012 Nov 3.

12.

Novel pseudopolymorph of the active metabolite of perindopril.

Bojarska J, Maniukiewicz W, Sieroń L, Fruziński A, Kopczacki P, Walczyński K, Remko M.

Acta Crystallogr C. 2012 Sep;68(Pt 9):o341-3. doi: 10.1107/S0108270112032349. Epub 2012 Aug 1.

PMID:
22935500
13.

Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with α₁-adrenoceptor antagonistic properties.

Handzlik J, Szymańska E, Wójcik R, Dela A, Jastrzębska-Więsek M, Karolak-Wojciechowska J, Fruziński A, Siwek A, Filipek B, Kieć-Kononowicz K.

Bioorg Med Chem. 2012 Jul 15;20(14):4245-57. doi: 10.1016/j.bmc.2012.05.064. Epub 2012 Jun 5.

PMID:
22739084
14.

5,6,7,8-Tetra-hydro-quinolin-8-one.

Lipińska TM, Karczmarzyk Z, Wysocki W, Gruba E, Fruziński A.

Acta Crystallogr Sect E Struct Rep Online. 2011 Jun 1;67(Pt 6):o1365. doi: 10.1107/S1600536811016175. Epub 2011 May 7.

15.

N-{2-[(4S)-4-tert-Butyl-4,5-dihydro-1,3-oxazol-2-yl]phen-yl}-5,6-diphenyl-1,2,4-triazin-3-amine.

Karczmarzyk Z, Wolińska E, Fruziński A.

Acta Crystallogr Sect E Struct Rep Online. 2011 Feb 19;67(Pt 3):o651. doi: 10.1107/S1600536811005411.

16.

1-(3-Chloro-phen-yl)-3-(1-p-tolyl-imidazolidin-2-yl-idene)urea.

Wysocki W, Matosiuk D, Karczmarzyk Z, Fidecka S, Fruziński A.

Acta Crystallogr Sect E Struct Rep Online. 2008 Dec 6;65(Pt 1):o40. doi: 10.1107/S1600536808040701.

17.

(E)-1-(Pyridin-2-yl)ethanone O-acryloyloxime.

Mojzych M, Karczmarzyk Z, Fruziński A.

Acta Crystallogr Sect E Struct Rep Online. 2008 Mar 5;64(Pt 4):o653. doi: 10.1107/S1600536808005436.

18.

Phenylethyl-substituted pyrimido[2,1-f]purinediones and related compounds: structure-activity relationships as adenosine A(1) and A(2A) receptor ligands.

Drabczyńska A, Müller CE, Schiedel A, Schumacher B, Karolak-Wojciechowska J, Fruziński A, Zobnina W, Yuzlenko O, Kieć-Kononowicz K.

Bioorg Med Chem. 2007 Nov 15;15(22):6956-74. Epub 2007 Aug 22.

PMID:
17827019

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