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Items: 9

1.

Visualization and quantification of neurokinin-1 (NK1) receptors in the human brain.

Hietala J, Nyman MJ, Eskola O, Laakso A, Grönroos T, Oikonen V, Bergman J, Haaparanta M, Forsback S, Marjamäki P, Lehikoinen P, Goldberg M, Burns D, Hamill T, Eng WS, Coimbra A, Hargreaves R, Solin O.

Mol Imaging Biol. 2005 Jul-Aug;7(4):262-72.

PMID:
16155744
2.

Synthesis and characterization of a potent, selective, radiolabeled substance-P antagonist for NK1 receptor quantitation: ([18F]SPA-RQ).

Solin O, Eskola O, Hamill TG, Bergman J, Lehikoinen P, Grönroos T, Forsback S, Haaparanta M, Viljanen T, Ryan C, Gibson R, Kieczykowski G, Hietala J, Hargreaves R, Burns HD.

Mol Imaging Biol. 2004 Nov-Dec;6(6):373-84.

PMID:
15564148
3.

Substance P: structure, function, and therapeutics.

Datar P, Srivastava S, Coutinho E, Govil G.

Curr Top Med Chem. 2004;4(1):75-103. Review.

PMID:
14754378
4.
5.

Neurobiology of substance P and the NK1 receptor.

Mantyh PW.

J Clin Psychiatry. 2002;63 Suppl 11:6-10. Review.

6.

The tachykinin peptide family.

Severini C, Improta G, Falconieri-Erspamer G, Salvadori S, Erspamer V.

Pharmacol Rev. 2002 Jun;54(2):285-322. Review.

7.

Brain uptake and receptor binding of two [11C]labelled selective high affinity NK1-antagonists, GR203040 and GR205171--PET studies in rhesus monkey.

Bergström M, Fasth KJ, Kilpatrick G, Ward P, Cable KM, Wipperman MD, Sutherland DR, Långström B.

Neuropharmacology. 2000 Feb 14;39(4):664-70.

PMID:
10728887
8.

The pharmacology of GR203040, a novel, potent and selective non-peptide tachykinin NK1 receptor antagonist.

Beattie DT, Beresford IJ, Connor HE, Marshall FH, Hawcock AB, Hagan RM, Bowers J, Birch PJ, Ward P.

Br J Pharmacol. 1995 Dec;116(8):3149-57.

9.

Discovery of an orally bioavailable NK1 receptor antagonist, (2S,3S)-(2-methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with potent antiemetic activity.

Ward P, Armour DR, Bays DE, Evans B, Giblin GM, Heron N, Hubbard T, Liang K, Middlemiss D, Mordaunt J, et al.

J Med Chem. 1995 Dec 22;38(26):4985-92.

PMID:
8544174
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