Mezilamine, a new dopamine antagonist, blocks presynaptic but stimulates postsynaptic alpha-adrenoceptors

Eur J Pharmacol. 1979 Oct 15;58(4):359-67. doi: 10.1016/0014-2999(79)90306-6.
No abstract available

MeSH terms

  • Adrenergic alpha-Agonists*
  • Adrenergic alpha-Antagonists*
  • Animals
  • Cerebral Cortex / metabolism
  • Dopamine Antagonists*
  • Drug Interactions
  • Female
  • Muscle Contraction / drug effects
  • Norepinephrine / metabolism
  • Piperazines / pharmacology
  • Pyrimidines / pharmacology*
  • Rats
  • Spinal Cord / physiology
  • Synapses / drug effects*
  • Synaptosomes / metabolism

Substances

  • Adrenergic alpha-Agonists
  • Adrenergic alpha-Antagonists
  • Dopamine Antagonists
  • Piperazines
  • Pyrimidines
  • mezilamine
  • Norepinephrine