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Org Lett. 2010 May 21;12(10):2314-7. doi: 10.1021/ol100671v.

General method for synthesis of 2-heterocyclic N-methyliminodiacetic acid boronates.

Author information

1
Howard Hughes Medical Institute, Roger Adams Lab, University of Illinois at Urbana-Champaign, Urbana, Illinois 61801, USA.

Abstract

A wide range of 2-pyridyl and other difficult-to-access heterocyclic N-methyliminodiacetic acid boronates can be readily prepared from the corresponding bromides via a new method involving direct transligation of 2-heterocyclic trialkoxyborate salts with N-methyliminodiacetic acid (MIDA) at elevated temperatures.

PMID:
20465293
PMCID:
PMC5127601
DOI:
10.1021/ol100671v
[Indexed for MEDLINE]
Free PMC Article

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