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J Org Chem. 2002 May 17;67(10):3365-73.

"Fleximers". Design and synthesis of a new class of novel shape-modified nucleosides(1).

Author information

1
School of Chemistry and Biochemistry, Georgia Institute of Technology, Atlanta, Georgia 30332-0400, USA. katherine.seley@chemistry.gatech.edu

Abstract

A new class of shape-modified nucleosides is introduced. These novel "fleximers" feature the purine ring systems of adenosine, inosine, and guanosine split into their individual imidazole and pyrimidine components (as in 1-3). This structural modification serves to introduce flexibility into the nucleoside while still retaining the elements essential for recognition. As a consequence, these novel fleximers should find use as bioprobes for investigating enzyme-coenzyme binding sites as well as nucleic acid and protein interactions. Their design and synthesis are described.

PMID:
12003548
[Indexed for MEDLINE]

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