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Bioorg Med Chem Lett. 1999 Sep 6;9(17):2579-82.

Preparation and receptor binding affinities of cyclic C-terminal neurotensin (8-13) and (9-13) analogues.

Author information

1
Department of Pharmaceutical Sciences, Medical University of South Carolina, Charleston 29425, USA.

Abstract

Cyclic analogues of neurotensin (NT) C-terminal fragments NT(8-13) and NT(9-13) were produced via intramolecular nucleophilic substitution of the Tyr(11) phenoxide anion on a 6-bromohexanoyl side chain substituted at position 8 or 9 and tested for NT receptor binding affinity.

PMID:
10498212
DOI:
10.1016/s0960-894x(99)00420-5
[Indexed for MEDLINE]

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