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Inhibition of human dopamine transporter
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv after 4 mins
Assay data:1 Tested
SummaryPubMed Citation
Drug uptake in Sprague-Dawley rat striatum assessed as reduction of striatal binding potential at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 60 mins
Drug uptake in Sprague-Dawley rat striatum assessed as reduction of striatal binding potential at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 30 mins
Drug uptake in Sprague-Dawley rat striatum assessed as reduction of striatal binding potential at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 15 mins
Ratio of drug uptake in striatum to cerebellum of Sprague-Dawley rat at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 60 mins
Ratio of drug uptake in striatum to cerebellum of Sprague-Dawley rat at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 30 mins
Ratio of drug uptake in striatum to cerebellum of Sprague-Dawley rat at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 15 mins
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 60 mins
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 30 mins
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv treated 45 mins after DAT inhibitor GBR-12909 challenge measured after 15 mins
Ratio of drug uptake in striatum to cerebellum of Sprague-Dawley rat at 37 MBq, iv after 60 mins
Ratio of drug uptake in striatum to cerebellum of Sprague-Dawley rat at 37 MBq, iv after 30 mins
Ratio of drug uptake in striatum to cerebellum of Sprague-Dawley rat at 37 MBq, iv after 15 mins
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv after 60 mins
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv after 30 mins
Drug uptake in Sprague-Dawley rat striatum assessed per cm'3 at 37 MBq, iv after 15 mins
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