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Agonist activity at full length human ERbeta receptor assessed as transcriptional activity incubated for 22 to 24 hrs by cell based luciferase reporter gene assay
Assay data:13 Active, 5 Activity ≤ 1 nM, 13 Activity ≤ 1 µM, 13 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at full length human ERbeta receptor assessed as inhibition of estradiol-induced activation incubated for 22 to 24 hrs by cell based luciferase reporter gene assay
Assay data:3 Activity ≤ 1 µM, 12 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at full length human ERalpha receptor assessed as inhibition of estradiol-induced activation incubated for 22 to 24 hrs by cell based luciferase reporter gene assay
Assay data:5 Activity ≤ 1 µM, 10 Tested
Agonist activity at full length human ERalpha receptor assessed as transcriptional activity incubated for 22 to 24 hrs by cell based luciferase reporter gene assay
Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested
Displacement of fluormone from GST-tagged ERbeta receptor LBD (unknown origin) measured after 60 mins by TR-FRET competitive binding assay
Assay data:14 Active, 5 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 14 Tested
Progesterone receptor (PR) small molecule agonists, qHTS assay: Summary
Assay data:193 Active, 7 Activity ≤ 1 nM, 121 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule agonists of the progesterone receptor (PR) signaling pathway - cell viability counter screen
Assay data:458 Active, 3 Activity ≤ 1 nM, 233 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
qHTS assay to identify small molecule agonists of the progesterone receptor (PR) signaling pathway
Assay data:138 Active, 6 Activity ≤ 1 nM, 166 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule antagonists of the estrogen related receptor signaling pathway with the pleiotropic PPARgamma coactivator (PGC) from Tox21 10K library: Summary
Assay data:462 Active, 149 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor beta (ER-beta) signaling pathway: Summary
Assay data:149 Active, 1 Activity ≤ 1 nM, 52 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line in the presence of 0.5 nM R1881: Summary
Assay data:1108 Active, 2 Activity ≤ 1 nM, 246 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway in the presence of an antagonist
Assay data:257 Active, 66 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor beta (ER-beta) signaling pathway
Assay data:113 Active, 4 Activity ≤ 1 nM, 67 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line in the presence of 0.5 nM R1881
Assay data:1453 Active, 4 Activity ≤ 1 nM, 292 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
BK Channel Variant Modulator Selectivity Assay
Assay data:286 Active, 904 Activity ≤ 1 nM, 951 Activity ≤ 1 µM, 951 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
A CellTox Green Cytotoxicity Assay to monitor cytotoxicity in HepG2 cells - 8 hour
Assay data:390 Active, 34 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Depositor
A CellTox Green Cytotoxicity Assay to monitor cytotoxicity in HEK293 cells - 16 hour
Assay data:413 Active, 35 Activity ≤ 1 µM, 9667 Tested
A CellTox Green Cytotoxicity Assay to monitor cytotoxicity in HEK293 cells - 8 hour
Assay data:327 Active, 30 Activity ≤ 1 µM, 9667 Tested
A CellTox Green Cytotoxicity Assay to monitor cytotoxicity in HepG2 cells - 32 hour
Assay data:900 Active, 77 Activity ≤ 1 µM, 9667 Tested
A CellTox Green Cytotoxicity Assay to monitor cytotoxicity in HepG2 cells - 0 hour
Assay data:120 Active, 17 Activity ≤ 1 µM, 9667 Tested
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