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Cytochrome P450 Family 3 Subfamily A Member 4 (CYP3A4) small molecule antagonists: luciferase reporter qHTS assay
Assay data:1792 Active, 248 Activity ≤ 1 µM, 9667 Tested
Summary
Cytochrome P450 family 2 subfamily C member 9 (CYP2C9) small molecule antagonists: luciferase cell-based qHTS assay
Assay data:2039 Active, 244 Activity ≤ 1 µM, 5242 Tested
Cytochrome P450 family 3 subfamily A member 4 (CYP3A4) small molecule antagonists: luciferase cell-based qHTS assay
Assay data:2147 Active, 1 Activity ≤ 1 nM, 377 Activity ≤ 1 µM, 5242 Tested
Inhibition of human GSTO1-1 by MMA (V) reductase assay
Assay data:2 Active, 5 Tested
Reversible inhibition of PTP1B (1 to 298 residues) (unknown origin) using 10 fold excess DifMUP as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by fluorescence assay
Assay data:1 Active, 1 Tested
Human pregnane X receptor (PXR) small molecule agonists, qHTS assay
Assay data:2218 Active, 1 Activity ≤ 1 nM, 106 Activity ≤ 1 µM, 9667 Tested
Drug repurposing screens with cells derived from glioblastoma tumor samples
Assay data:1237 Active, 3 Activity ≤ 1 nM, 360 Activity ≤ 1 µM, 3733 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor beta (ER-beta) signaling pathway - cell viability counter screen
Assay data:1136 Active, 121 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway in the presence of an antagonist - cell viability counter screen
Assay data:756 Active, 46 Activity ≤ 1 µM, 9667 Tested
AlphaScreen-based biochemical high throughput primary assay to identify inhibitors of Unc-51 Like Autophagy Activating Kinase 1 (ULK1).
Assay data:575 Active, 30318 Tested
qHTS RealTime-Glo MT Cell Viability Assay in HepG2 cells - 32 hour
Assay data:444 Active, 40 Activity ≤ 1 µM, 9667 Tested
qHTS RealTime-Glo MT Cell Viability Assay in HepG2 cells - 40 hour
Assay data:442 Active, 39 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule agonists of the hypoxia (HIF-1) signaling pathway - cell viability counter screen
Assay data:617 Active, 94 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway
Assay data:1034 Active, 2 Activity ≤ 1 nM, 491 Activity ≤ 1 µM, 9667 Tested
qHTS assay to identify small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway - cell viability counter screen
Assay data:498 Active, 61 Activity ≤ 1 µM, 9667 Tested
DLD-1 viability from Cell TiterGlo-screen
Assay data:479 Active, 2458 Tested
SW480 viability from Cell TiterGlo-screen
Assay data:746 Active, 2458 Tested
HCT116 viability from Cell TiterGlo-screen
Assay data:509 Active, 2458 Tested
VEGF stimulated ADSC/ECFC co-culture CD31-stained tube area decrease-screen
Assay data:357 Active, 2422 Tested
Induction of apoptosis in Homo sapiens (human) HCT116 cells assessed as caspase9 cleavage at 52.3 uM at 16 hr by Western blot analysis
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