Format
Items per page
Sort by

Send to:

Choose Destination

Links from

Items: 1 to 20 of 456

1.

Antagonist activity at CCR5 receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of CCl5-induced calcium release at 1 uM by FLIPR assay

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
2.

Displacement of [125I]-MIP-1beta form CCR5 (unknown origin)

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
3.

Displacement of [125I]-MIP-1beta form CCR5 (unknown origin) at 1 mM

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
4.

Displacement of [125I]-MIP-1beta form CCR5 (unknown origin) at 100 uM

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
5.
6.

Antagonist activity at CCR5 (unknown origin) expressed in human MOLT4 cells assessed as inhibition of CCL5-induced calcium mobilization after 1 hr

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
8.

Antagonist activity against human CCR2B expressed in Chem-1 cells assessed as inhibition of human CCL2-induced intracellular calcium flux incubated for 10 mins by Fluo-4 AM dye based intracellular calcium flux assay

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
AID:
1232304
9.

Displacement of [125I]-CCL2 from human CCR2 expressed in U2OS cells incubated for 150 mins by scintillation spectrometry

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
10.

Displacement of [125I]-CCL2 from human CCR2 expressed in U2OS cells at 1 uM incubated for 150 mins by scintillation spectrometry

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
11.

Antagonist activity against CCR5 in whole blood (unknown origin) assessed as reduction in CD11b upregulation

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
12.

Antagonist activity against CCR2 in whole blood (unknown origin) assessed as reduction in CD11b upregulation

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
13.

Inhibition of [125I]MCP1-beta binding to CCR5 in human HT1080 cell membranes incubated for 4 to 6 hrs

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
14.

Antagonist activity against CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis at 37 degC

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
AID:
1226282
15.

Inhibition of [125I]hMCP1 binding to CCR2 in human PBMC incubated for 30 mins at room temperature

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
AID:
1226281
16.

C-C chemokine receptor type 2 antagonist

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
17.

Antagonist activity at CCR5 (unknown origin) at 10 uM relative to control

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
18.

Antagonist activity at CCR2B (unknown origin) at 10 uM relative to control

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
19.

Agonist activity at CCR5 (unknown origin) at 12.5 uM relative to control

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 5; C-C CKR-5; CC-CKR-5; CCR-5; CCR5; CHEMR13; HIV-1 fusion coreceptor; CD_antigen=CD195
20.

Agonist activity at CCR2B (unknown origin) at 12.5 uM relative to control

Source:
ChEMBL
Protein Target:
C-C chemokine receptor type 2; C-C CKR-2; CC-CKR-2; CCR-2; CCR2; Monocyte chemoattractant protein 1 receptor; MCP-1-R; CD_antigen=CD192
Format
Items per page
Sort by

Send to:

Choose Destination

Supplemental Content

Refine your results

• What's this?

Actions on your results

Find related data

Recent activity

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...
Support Center