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Items: 1 to 20 of 40

3.
4.

BindingDB_Patents: Inhibition Assay. For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and analogous enzymes was used.

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
5.

Inhibition of human VAP1

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
6.

Stability of the compound assessed as human full length SSAO-mediated drug metabolism expressed in CHO cells measured as compound remaining after 20 mins

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
7.

Inhibition of human recombinant VAP-1 transfected in CHO cells using 2,4-dichlorophenol/benzylamine as substrate incubated for 30 mins prior to benzylamine addition measured after 1 hr by spectrophotometry

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
8.
9.

Inhibition of rat VAP-1

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; Semicarbazide-sensitive amine oxidase; SSAO; VP97; Vascular adhesion protein 1; VAP-1
10.

Binding affinity to human recombinant VAP-1 by surface plasmon resonance analysis

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
11.

Activity at recombinant human VAP-1 assessed as hydrogen peroxide generation rate preincubated for 30 mins by Amplex Red assay

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
12.

Activity at recombinant human VAP-1 assessed as hydrogen peroxide generation rate per min/mg preincubated for 30 mins by Amplex Red assay relative to control

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
13.

Ratio of relative Vmax to Km for recombinant human VAP-1 assessed as hydrogen peroxide generation rate preincubated for 30 mins by Amplex Red assay relative to control

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
14.

Activity at recombinant human VAP-1 assessed as hydrogen peroxide generation rate per min/mg using benzylamine as substrate at 200 uM preincubated for 30 mins by Amplex Red assay relative to control

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
15.

Ratio of relative Vmax to Km for recombinant human VAP-1 assessed as hydrogen peroxide generation rate using benzylamine as substrate at 200 uM preincubated for 30 mins by Amplex Red assay

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
16.

Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB

Source:
Shanghai Institute of Organic Chemistry
Protein Targets:
Chain 1, E. Coli (Lacz) Beta-Galactosidase (R599a) In Complex With D- Galctopyranosyl-1-One; ...
Total:
3355
AID:
977610
17.

Inhibition of human VAP-1 expressed in CHO cells using [14C]-benzylamine as substrate preincubated for 30 mins prior to substrate addition measured after 1 hr by scintillation spectrometric analysis

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
18.

Inhibition of rat VAP-1 expressed in CHO cells using [14C]-benzylamine as substrate preincubated for 30 mins prior to substrate addition measured after 1 hr by scintillation spectrometric analysis

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; Semicarbazide-sensitive amine oxidase; SSAO; VP97; Vascular adhesion protein 1; VAP-1
19.

Inhibition of human VAP1 expressed in CHO cells using [14C]-benzylamine as substrate incubated for 30 mins prior to substrate addition measured after 1 hr by scintillation counting analysis

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; HPAO; Semicarbazide-sensitive amine oxidase; SSAO; Vascular adhesion protein 1; VAP-1
20.

Inhibition of rat VAP1 expressed in CHO cells using [14C]-benzylamine as substrate incubated for 30 mins prior to substrate addition measured after 1 hr by scintillation counting analysis

Source:
ChEMBL
Protein Target:
Membrane primary amine oxidase; Copper amine oxidase; Semicarbazide-sensitive amine oxidase; SSAO; VP97; Vascular adhesion protein 1; VAP-1
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