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Links from PubChem BioAssay

Items: 1 to 20 of 30

1.

Inhibition of KHS (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
2.

Inhibition of GLK (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 3; Germinal center kinase-related protein kinase; GLK; MAPK/ERK kinase kinase kinase 3; MEK kinase kinase 3; MEKKK 3
3.

Inhibition of recombinant human KHS1 at 1 uM relative to control

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
4.

Competitive binding affinity to KHS1 in human A375 cells after 15 mins in presence of ATP analogue

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
5.

Inhibition of MAP4K5 (unknown origin) at 1 uM in presence of 100 uM ATP

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
6.

Inhibition of KHS1 (unknown origin) at 100 nM

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
7.

Inhibition of KHS1 (unknown origin) at 1 uM

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
8.

Inhibition of MAP4K5 (unknown origin) in presence of 1 mM ATP

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
9.

Inhibition of MAP4K5 (unknown origin) assessed as remaining enzyme activity at 10 uM by radioactive [33P]-ATP filter binding assay

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
10.

Inhibition of MAP4K3 (unknown origin) assessed as remaining enzyme activity at 10 uM by radioactive [33P]-ATP filter binding assay

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 3; Germinal center kinase-related protein kinase; GLK; MAPK/ERK kinase kinase kinase 3; MEK kinase kinase 3; MEKKK 3
11.

Inhibition of KHS1 (unknown origin) at 1 uM

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
12.

Inhibition of KHS1 (unknown origin) at 10 uM

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
13.

Competitive binding affinity to MAP4K5 (unknown origin) at 10 uM in presence of ATP relative to control

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
14.

Competitive binding affinity to MAP4K3 (unknown origin) at 10 uM in presence of ATP relative to control

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 3; Germinal center kinase-related protein kinase; GLK; MAPK/ERK kinase kinase kinase 3; MEK kinase kinase 3; MEKKK 3
15.

Inhibition of MAP4K5 (unknown origin) at 50 times TAK1 Ki

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
16.

Inhibition of MAP4K5 (unknown origin) at 10 uM relative to control

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
17.

Inhibition of KHS1 (unknown origin) assessed as remaining activity at 1 uM relative to control

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
18.

Inhibition of KHS1 (unknown origin) assessed as remaining activity at 10 uM relative to control

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
19.

Inhibition of human KHS1 in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
20.

Binding constant for MAP4K5 kinase domain

Source:
ChEMBL
Protein Target:
Mitogen-activated protein kinase kinase kinase kinase 5; Kinase homologous to SPS1/STE20; KHS; MAPK/ERK kinase kinase kinase 5; MEK kinase kinase 5; MEKKK 5
AID:
625061
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