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Items: 16

1.

Inhibition of PKR (unknown origin)

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
2.

Inhibition of PRKR (unknown origin) at 1 uM relative to control

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
3.

Inhibition of EIF2AK2 (unknown origin) at 1 uM after 1 hr

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
4.

Inhibition of PKR (unknown origin) assessed as EIF2AK2 phosphorylation

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
5.

Binding affinity to PRKR (unknown origin)

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
6.

Competitive binding affinity to PRKR (unknown origin) at 10 uM in presence of ATP relative to control

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
7.

Inhibition of PKR in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
8.

Inhibition of human PKR in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
9.

Binding constant for PRKR kinase domain

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
10.

Inhibition of human PKR in HL60 cells lysate at 10 uM using post probe-labeling by LC-MS/MS analysis relative to control

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
11.

Competitive inhibition of human recombinant PKR

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
12.

Inhibition of human recombinant PKR autophosphorylation using poly[I:C] after 10 mins by luminescent assay

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
13.

Binding constant for PRKR kinase domain

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
14.

Inhibition of E2K2

Source:
ChEMBL
Protein Target:
Interferon-induced, double-stranded RNA-activated protein kinase; Eukaryotic translation initiation factor 2-alpha kinase 2; eIF-2A protein kinase 2; Interferon-inducible RNA-dependent protein kinase; P1/eIF-2A protein kinase; Protein kinase RNA-activated; PKR; Protein kinase R; Tyrosine-protein kinase EIF2AK2; p68 kinase
15.

Kinase inhibition selectivity assay for compound SID-48409448

Source:
Burnham Center for Chemical Genomics
Protein Targets:
3-phosphoinositide-dependent protein kinase 1 isoform 1 [Homo sapiens]; ...
Total:
314
16.

Kinase Inhibitor Selectivity Profiling Assay

Source:
Ambit Biosciences
Protein Targets:
3-phosphoinositide-dependent protein kinase 1 isoform 1 [Homo sapiens]; ...
Total:
287
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