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Mobility-Shift Assay from US Patent US11912663: "Multi-targeted tyrosine kinase inhibitors and their pharmaceutical uses"
Assay data:14 Active, 15 Activity ≤ 1 µM, 15 Tested
SummaryRelated BioAssays by Target
In Vitro Kinase Binding Assay from US Patent US20240058459: "DENDRIMER COMPOSITIONS AND METHODS FOR DRUG DELIVERY TO THE EYE"
Assay data:3 Active, 2 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
Safety47 Scan (DiscoverX - Eurofins)
Assay data:1 Tested
SRC SGC Tm panel (DSF)
SRC Invitrogen Lab (UK) kinase screen (BI)
LYN A Invitrogen Lab (UK) kinase screen (BI)
KDR Invitrogen Lab (UK) kinase screen (BI)
Compound was evaluated for inhibition of human KDR in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:12 Active, 3 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 101 Tested
Assay data:19 Active, 11 Activity ≤ 1 µM, 692 Tested
Inhibition of LYN (unknown origin) at 10 uM by biochemical hotspot kinase assay
Inhibition of c-Src (unknown origin) at 10 uM by biochemical hotspot kinase assay
Inhibition of VEGFR2 (unknown origin) at 10 uM by biochemical hotspot kinase assay
Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 60 mins by ELISA
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of VEGFR-2 (unknown origin)
Assay data:9 Active, 8 Activity ≤ 1 µM, 10 Tested
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