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Dopamine Transporter Binding Assay from US Patent US11555013: "Potent and selective inhibitors of monoamine transporters; method of making; and use thereof"
Assay data:50 Active, 35 Activity ≤ 1 µM, 59 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition of dopamine transporter (unknown origin) assessed as inhibition of dopamine reuptake
Assay data:5 Active, 3 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of norepinephrine transporter (unknown origin) assessed as inhibition of norepinephrine reuptake
Assay data:5 Active, 1 Activity ≤ 1 µM, 5 Tested
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000209b SLC6A2
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000295b SLC6A3
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000545a SLC6A3
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Lead profiling screen (Eurofins, GPCRs, ion channels, kinases and transporters)) EUB0000309b SLC6A3
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (CEREP panel (Eurofins, radioligand binding assay, enzymes, GPCRS, transporters, and ion channels)) EUB0000308b SLC6A3
Selectivity interaction (CEREP panel (Eurofins, radioligand binding assay, enzymes, GPCRS, transporters, and ion channels)) EUB0000308b SLC6A2
Selectivity interaction (CEREP ExpressProfile selectivity/specificity profile (human recombinant receptors)) EUB0000213bCl SLC6A3
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000542a SLC6A3
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000541a SLC6A3
Selectivity interaction (PRESTO-Tango GPCR-ome screening) EUB0000539a SLC6A3
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000353a SLC6A3
Selectivity interaction (Eurofins-Panlabs screen (receptors)) EUB0000352a SLC6A3
Selectivity interaction (Prostanoid receptor binding assay) EUB0000334a SLC6A3
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000316b SLC6A3
Selectivity interaction (Prostanoid receptor binding assay) EUB0000297b SLC6A3
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000297b SLC6A3
Selectivity interaction (Radioligand binding assay (MDS Pharma Service)) EUB0000296b SLC6A3
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