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Compound was tested for its ability to inhibit binding of arginine vasopressin to Vasopressin receptor (V1 subtype); ND is no data
Assay data:5 Tested
SummaryRelated BioAssays by Target
Compound was tested for its ability to inhibit binding of arginine vasopressin to Vasopressin receptor (V1 subtype)
Assay data:2 Tested
Tested for inhibition of vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney.
Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.
Affinity towards vasopressin receptor in porcine renal medullary membrane using [3H]LVP
Assay data:9 Active, 10 Activity ≤ 1 µM, 10 Tested
Affinity for vasopressin V2-receptor of porcine renal medullary membrane
Assay data:13 Tested
SummaryPubMed CitationRelated BioAssays by Target
Ability to displace [3H]AVP from Vasopressin V2 receptor
Assay data:1 Tested
In vitro antagonist activity was measured by inhibition of vasopressin-stimulated adenylate cyclase in renal medullary preparation in pig
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Inhibition of LVP-sensitive adenylate cyclase in a pig renal medullary preparation
Assay data:4 Active, 2 Activity ≤ 1 µM, 4 Tested
Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor); NT=Not tested
Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
Binding affinity towards Vasopressin V2 receptor in LLCPK cells
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Vasopressin V2 receptor binding affinity measured by competition with tritiated LVP lysine vasopressin in pig renal medullary preparation
Assay data:2 Active, 2 Activity ≤ 1 µM, 4 Tested
Inhibition constant for [3H]LVP binding to medullary membranes of pig kidney of Vasopressin V2 receptor
Assay data:11 Active, 10 Activity ≤ 1 µM, 11 Tested
In vitro antagonist activity was measured by inhibition of binding of [3H]LVP to renal medullary membrane preparation in pig
Antagonistic activity of the V2 system (Vasopressin V2 receptor) was evaluated bythe adenylate cyclase activity in LLCPK cells at a concentration of 10E-7 M; No activity
Agonistic activity of the V2 system (Vasopressin V2 receptor) was evaluated bythe adenylate cyclase activity in LLCPK cells at a concentration of 10E-7 M; No activity
Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations; nd=Not determined
Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations; e=Partial agonist with a relative Vmax of 14%.
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations.
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