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Antagonist activity at rat P2X4R expressed in HEK293 cells preincubated for 2 mins followed by ATP addition and measured after 4 mins
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Purinergic P2X Eurofins-Panlabs radioligand binding assay
Assay data:5 Tested
SummaryRelated BioAssays by Target
P2X Eurofins-Cerep binding assay
Assay data:2 Tested
P2X CEREP ligand profiling
Assay data:1 Tested
P2X-purinergic receptor CEREP ligand profiling
P2X Ligand binding assay
rP2X Cerep panel
Antagonist activity at rat P2X4 receptor expressed in Xenopus laevis oocytes assessed as reduction in ATP-induced channel currents at 100 uM by TEVC electrophysiology assay relative to control
SummaryPubMed CitationRelated BioAssays by Target
Displacement of [3H]alpha, beta-methylene ATP from P2X receptor in rat urinary bladder at 10 uM incubated for 120 mins by scintillation counting analysis relative to control
Displacement of [3H] alpha, beta-Methylene-ATP from P2X receptor in Wistar rat urinary bladder assessed as residual binding level for radioligand at 10 uM incubated for 120 mins by liquid scintillation counting method relative to control
Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 10 mins by Fluo2-AM staining based inverted fluorescence microscopic method
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 mins and measured every 2 secs for 120 secs by Fluo8-AM staining based FLIPR assay
Displacement of [3H]alpha, beta-MeATP from rat bladder P2X at 10 uM after 120 mins by scintillation counting analysis relative to control
Inhibition of rat P2X4 receptor expressed in xenopus lavies oocytes assessed as inhibition of ATP-induced peak current at 3 mM by two electrode voltage clamp
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