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Antagonist activity at PAC1R in rat RG2 cells assessed as inhibition of Maxadilan-induced cAMP accumulation pre-incubated for 30 mins followed by agonist addition and measured after 75 mins by Eu-cAMP tracer based LANCE ultra cAMP assay
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at PAC1R in rat RG2 cells assessed as inhibition of PACAP38-induced cAMP accumulation pre-incubated for 30 mins followed by agonist addition and measured after 75 mins by Eu-cAMP tracer based LANCE ultra cAMP assay
Rat PAC1 receptor (VIP and PACAP receptors)
Assay data:9 Active, 9 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Antagonist activity at PAC1R in rat AR42J cells assessed as PACAP-induced calcium mobilization by FLIPR assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
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