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Binding affinity to C9orf72 (G4C2)2 G4 quadruplex RNA (unknown origin) assessed as change in chemical shift by one-dimensional 1H-NMR analysis
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed Citation
Binding affinity to C9orf72 (G4C2)4 G4 quadruplex DNA (unknown origin) assessed as change in chemical shift at pH 6 in 25 to 45 degree C by one-dimensional 1H-NMR analysis
Assay data:3 Active, 3 Tested
Neuroprotective activity in mouse Neuro2a cells transfected DNA (G4C2)29 C9orf 72 ALS/FTD cell model assessed as increase in cell viability at 1 ug/ml by DAPI staining based immunofluorescence analysis
Assay data:2 Active, 3 Tested
Binding affinity to (GGCCCC)5 motif-containing duplex DNA (unknown origin) at 80 uM by ESI-TOF-MS analysis
Assay data:1 Active, 1 Tested
Binding affinity to (GGCCCC)9 motif-containing duplex DNA (unknown origin) assessed as formation of CD bands at 20 uM at 245 to 282 nm by CD spectrometry
Binding affinity to (GGCCCC)9 motif-containing duplex DNA (unknown origin) assessed as melting temperature at 20 uM by UV-spectrophotometric method
Assay data:1 Tested
SummaryPubMed Citation
Binding affinity to GGCCCC/GGGGCC motif-containing duplex DNA (unknown origin) at 40 uM by ESI-TOF-MS analysis
Binding affinity to GGCCCC/GGCCCC motif-containing duplex DNA (unknown origin) at 80 uM by ESI-TOF-MS analysis
Binding affinity to GGCCCC/GGCCCC motif-containing duplex DNA (unknown origin) at 40 uM by ESI-TOF-MS analysis
Binding affinity to GGCTCC/GGCTCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
Binding affinity to GGTTCC/GGCCCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
Binding affinity to GGTCCC/GGTCCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
Binding affinity to GGTCCC/GGCTCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
Binding affinity to GGCTCC/GGCCCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
Binding affinity to GGTCCC/GGCCCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
Binding affinity to GGTCCC/GGTCCC motif-containing duplex DNA (unknown origin) assessed as formation of CD bands at 20 uM at 310 to 345 nm by CD spectrometry
Binding affinity to GGCTCC/GGCCCC motif-containing duplex DNA (unknown origin) assessed as formation of CD bands at 20 uM at 310 to 345 nm by CD spectrometry
Binding affinity to GGTCCC/GGCCCC motif-containing duplex DNA (unknown origin) assessed as formation of CD bands at 20 uM at 300 to 345 nm by CD spectrometry
Binding affinity to GGCCCC/GGCCCC motif-containing duplex DNA (unknown origin) assessed as formation of CD bands at 20 uM at 310 to 345 nm by CD spectrometry
Binding affinity to GGCCC/GGCCC motif-containing duplex DNA (unknown origin) assessed as change in melting temperature at 20 uM by UV-spectrophotometric method
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