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Antiviral activity against RSV A2 infected in african green monkey assessed as reduction in viral replication in lung lavage samples at 10 mg/kg, iv administered 4 hrs prior to viral infection and daily upto 5 days post infection and measured every other day until day 15 by RT-qPCR analysis
Assay data:1 Tested
SummaryPubMed Citation
Terminal half life in African green monkey at 10 mg/kg, iv after 30 mins by LC-MS/MS analysis
Antitrypanosomal activity against bloodstream Trypanosoma vivax STIB 719/ ILRAD 560 infected in Fulani Zebu cattle assessed as reduction in parasitemia at 10 mg/kg, IM administered twice daily and measured after 4 days
Drug level in Swiss-Webster mouse plasma infected with Trypanosoma brucei brucei TREU667 at 50 mg/kg, po bid administered via gavage for 10 days starting from 21 days post infection measured at 1 hr post last dose
Drug level in Swiss-Webster mouse plasma infected with Trypanosoma brucei brucei TREU667 at 50 mg/kg, po bid administered via gavage for 10 days starting from 21 days post infection measured on day 7 prior to dose 15
Drug level in Swiss-Webster mouse plasma infected with Trypanosoma brucei rhodesiense STIB900 at 50 mg/kg, po bid administered via gavage for 4 days starting from 2 days post infection measured at 1 hr post last dose
Drug level in Swiss-Webster mouse plasma infected with Trypanosoma brucei rhodesiense STIB900 at 50 mg/kg, po bid administered via gavage for 4 days starting from 2 days post infection measured on day 3 prior to dose 7
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
AUC (0 to infinity) in mouse at 50 mg/kg, po administered as single dose via gavage as 0.5% methylcellulose cP400/0.5% Tween 80 formulation by liquid chromatography/tandem mass spectrometric analysis
Drug level in mouse plasma at 50 mg/kg, po administered as single dose via gavage measured at 24 hrs post dose by liquid chromatography/tandem mass spectrometric analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Drug level in mouse plasma at 50 mg/kg, po administered as single dose via gavage measured at 8 hrs post dose by liquid chromatography/tandem mass spectrometric analysis
Drug level in mouse plasma at 50 mg/kg, po administered as single dose via gavage measured at 4 hrs post dose by liquid chromatography/tandem mass spectrometric analysis
Drug level in mouse plasma at 50 mg/kg, po administered as single dose via gavage measured at 1 hr post dose by liquid chromatography/tandem mass spectrometric analysis
Drug level in mouse plasma at 5 mg/kg, ip administered as single dose measured at 1 hr post dose by liquid chromatography/tandem mass spectrometric analysis
Assay data:17 Active, 4 Activity ≤ 1 µM, 17 Tested
AUC (0 to infinity) in mouse at 50 mg/kg, po administered as single dose via gavage as 7% Tween 80/3% EtOH/5% DMSO formulation by liquid chromatography/tandem mass spectrometric analysis
Assay data:4 Tested
AUC in mouse plasma at 50 mg/kg, po by LC-MS analysis
Assay data:2 Tested
Antitrypanosomal activity against bloodstream Trypanosoma congolense KONT 2/133 infected in Friesian-Holstein calf assessed as reduction in parasitemia at 5 mg/kg, sc BID and measured after 3 days
Bioavailability in Fresian-Holstein cattle at 10 mg/kg,IM measured upto 120 hrs
AUC (0 to infinity) in Fresian-Holstein cattle at 2 mg/kg, iv measured upto 120 hrs
Antitrypanosomal activity against bloodstream Trypanosoma congolense IL3000 assessed as parasite growth inhibition incubated for 69 hrs by resazurin dye based fluorescence analysis
Assay data:8 Active, 2 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 8 Tested
Antitrypanosomal activity against bloodstream Trypanosoma brucei brucei assessed as parasite growth inhibition incubated for 3 days by resazurin dye based fluorescence analysis
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