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Items: 4

1.

Naltrexone

A noroxymorphone derivative with competitive opioid antagonistic property. Naltrexone reverses the effects of opioid analgesics by binding to the various opioid receptors in the central nervous system, including the mu-, kappa- and gamma-opioid receptors. This leads to an inhibition of the typical actions of opioid analgesics, including analgesia, euphoria, sedation, respiratory depression, miosis, bradycardia, and physical dependence. Naltrexone is longer-acting and more potent compared to naloxone. [from NCI]

MedGen UID:
6516
Concept ID:
C0027360
Organic Chemical; Pharmacologic Substance
2.

Related

MedGen UID:
619805
Concept ID:
C0445223
Finding
3.

Agonist

An agent that has affinity for a receptor and intrinsic activity at that receptor. [from NCI]

MedGen UID:
459858
Concept ID:
C2987634
Pharmacologic Substance
4.

Drug Inverse Agonism

Phenomena and pharmaceutics of compounds that bind to the same receptor binding-site as an agonist (DRUG AGONISM) for that receptor but exerts the opposite pharmacological effect. [from MeSH]

MedGen UID:
363051
Concept ID:
C1955884
Molecular Function
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