IDBrain Penetration Studies
Plasma Concentration (μM)Brain Concentration (μM)Ratio [B]/[P] (%)
SID-17507305 8.5 ± 3.33.7 ± 1.744
SID-17413392 1.1 ± 0.10.4 ± 0.0336
SID-17413034 1.6 ± 0.61.7 ± 0.6106
SID-4242079 9.0 ± 0.74.5 ± 0.350
SID-22413249 1.3 ± 0.31.5 ± 0.2115
BIIE-0246 12 ± 20.2 ± 0.12

From: Probe Report for NPY-Y2 Receptor Antagonists

Cover of Probe Reports from the NIH Molecular Libraries Program
Probe Reports from the NIH Molecular Libraries Program [Internet].

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