PubChem AIDTypeTargetConc. RangeSamples Tested
2551Primary qHTSRORγt46 μM to 3 nM305467
2546Primary qHTSVP1646 μM to 3 nM304088
2762ConfirmatoryRORγt46 μM to 0.26 nM250
2763ConfirmatoryVP1646 μM to 0.26 nM250
489037SecondaryRORγt92 μM to 0.52 nM185
492954OrthogonalTh1720 μM to 0.1 μM37
489039Anti-targetRORα92 μM to 0.52 nM185
489036Anti-targetVP1692 μM to 0.52 nM185
489038Anti-targetDHR392 μM to 0.52 nM185
492962Anti-targetTh130 μM to 3 μM3
2604SummaryRORγt

From: Identification of Potent and Selective RORγ Antagonists

Cover of Probe Reports from the NIH Molecular Libraries Program
Probe Reports from the NIH Molecular Libraries Program [Internet].

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