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Accession: PRJNA345242 ID: 345242

Homo sapiens (human)

A novel LSD1 inhibitor T-3775440 induces transdifferentiation in AML cell lines

See Genome Information for Homo sapiens
We describe the anti-leukemic activity and mechanism of action of T-3775440, a novel irreversible LSD1 inhibitor. More...
AccessionPRJNA345242; GEO: GSE87580
Data TypeTranscriptome or Gene expression
ScopeMultiisolate
OrganismHomo sapiens[Taxonomy ID: 9606]
Eukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi; Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini; Catarrhini; Hominidae; Homo; Homo sapiens
PublicationsIshikawa Y et al., "A Novel LSD1 Inhibitor T-3775440 Disrupts GFI1B-Containing Complex Leading to Transdifferentiation and Impaired Growth of AML Cells.", Mol Cancer Ther, 2017 Feb;16(2):273-284
SubmissionRegistration date: 3-Oct-2016
Oncology Drug Discovery Unit, Takeda Pharmaceutical Company Ltd.
RelevanceMedical
Project Data:
Resource NameNumber
of Links
Publications
PubMed1
Other datasets
GEO DataSets1
GEO Data Details
ParameterValue
Data volume, Spots755712
Data volume, Processed Mbytes9
Data volume, Supplementary Mbytes40

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