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8P07:
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 5-((3-(4H-1,2,4-triazol-4-yl)phenyl)amino)-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile
PDB ID:
8P07
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MMDB ID:
230344
PDB Deposition Date:
2023/5/9
Updated in MMDB:
2024/08
Experimental Method:
x-ray diffraction
Resolution:
2.4 Å
Source Organism:
Homo sapiens
Similar Structures:
VAST+
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Biological Unit for 8P07: dimeric; determined by author
Molecular Components in 8P07
Label
Count
Molecule
Proteins (2 molecules)
A
B
2
Casein Kinase II Subunit Alpha
(Gene symbol:
CSNK2A1
)
Chemicals and Non-standard biopolymers (18 molecules)
1
12
SULFATE ION
2
2
7-(cyclopropylamino)-5-[[3-(1,2,4-triazol-4-yl)phenyl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
3
4
1,2-ETHANEDIOL
* Click molecule labels to explore molecular sequence information.
Citing MMDB
Madej T, Lanczycki CJ, Zhang D, Thiessen PA, Geer RC, Marchler-Bauer A, Bryant SH.
"
MMDB and VAST+: tracking structural similarities between macromolecular complexes.
Nucleic Acids Res. 2014 Jan; 42(Database issue)
:D297-303