8DD5: Crystal structure of KAT6A in complex with inhibitor CTx-648 (PF-9363)

PDB ID: 8DD5Download
MMDB ID: 232382
PDB Deposition Date: 2022/6/17
Updated in MMDB: 2023/07
Experimental Method:
x-ray diffraction
Resolution: 2.58  Å
Source Organism:
Similar Structures:
Biological Unit for 8DD5: monomeric; determined by author
Molecular Components in 8DD5
Label Count Molecule
Protein (1 molecule)
1
Histone Acetyltransferase Kat6a
(Gene symbol: KAT6A)
Molecule annotation
Chemicals and Non-standard biopolymers (2 molecules)
1
1
2,6-dimethoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1-sulfonamide2,6-dimethoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1-sulfonamide
2
1
ZINC IONZINC ION
* Click molecule labels to explore molecular sequence information.
Citing MMDB
Madej T, Lanczycki CJ, Zhang D, Thiessen PA, Geer RC, Marchler-Bauer A, Bryant SH. " MMDB and VAST+: tracking structural similarities between macromolecular complexes. Nucleic Acids Res. 2014 Jan; 42(Database issue):D297-303