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8CYI:
Cryo-EM structures and computational analysis for enhanced potency in MTA-synergic inhibition of human protein arginine methyltransferase 5
PDB ID:
8CYI
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MMDB ID:
228961
PDB Deposition Date:
2022/5/23
Updated in MMDB:
2024/06
Experimental Method:
electron microscopy
Resolution:
3.14 Å
Source Organism:
Homo sapiens
Similar Structures:
VAST+
Download sequence data
Biological Unit for 8CYI: dimeric; determined by author
Molecular Components in 8CYI
Label
Count
Molecule
Proteins (2 molecules)
A
1
Protein Arginine N-methyltransferase 5
(Gene symbol:
PRMT5
)
B
1
Methylosome Protein 50
(Gene symbol:
WDR77
)
Chemicals and Non-standard biopolymers (2 molecules)
1
1
N-[(2-aminoquinolin-7-yl)methyl]-9-(2-hydroxyethyl)-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
2
1
5'-DEOXY-5'-METHYLTHIOADENOSINE
* Click molecule labels to explore molecular sequence information.
Citing MMDB
Madej T, Lanczycki CJ, Zhang D, Thiessen PA, Geer RC, Marchler-Bauer A, Bryant SH.
"
MMDB and VAST+: tracking structural similarities between macromolecular complexes.
Nucleic Acids Res. 2014 Jan; 42(Database issue)
:D297-303