4TPP: 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors

PDB ID: 4TPPDownload
MMDB ID: 125670
PDB Deposition Date: 2014/6/9
Updated in MMDB: 2023/12
Experimental Method:
x-ray diffraction
Resolution: 2.65  Å
Source Organism:
Similar Structures:
Biological Unit for 4TPP: trimeric; determined by author and by software (PISA)
Molecular Components in 4TPP
Label Count Molecule
Proteins (3 molecules)
3
Camp and Camp-inhibited Cgmp 3',5'-cyclic Phosphodiesterase 10A
(Gene symbol: PDE10A)
Molecule annotation
Chemicals and Non-standard biopolymers (33 molecules)
6
21
3
3
* Click molecule labels to explore molecular sequence information.

Citing MMDB